Literature DB >> 27736689

Randomized, proof-of-concept trial of low dose naltrexone for patients with breakthrough symptoms of major depressive disorder on antidepressants.

David Mischoulon1, Lindsay Hylek2, Albert S Yeung2, Alisabet J Clain2, Lee Baer2, Cristina Cusin2, Dawn Flosnik Ionescu2, Jonathan E Alpert2, David P Soskin2, Maurizio Fava2.   

Abstract

BACKGROUND: Given the proposed dopaminergic mechanism of low-dose naltrexone (LDN), we examined its efficacy as augmentation for depressive breakthrough on pro-dopaminergic antidepressant regimens.
METHODS: 12 adults (67% female, mean age = 45±12) with recurrent DSM-IV major depressive disorder (MDD) on dopaminergic antidepressant regimens (stimulants, dopamine agonists, bupropion [≥300mg/day], aripiprazole [≤2.5mg/day], or sertraline [≥150mg/day]) were randomized to naltrexone 1mg b.i.d. (n=6) or placebo (n=6) augmentation for 3 weeks.
RESULTS: All subjects completed the trial. Hamilton Depression Rating Scale (HAM-D-17) scores (primary outcome measure) decreased from 21.2±2.0 to 11.7±7.7 for LDN, from 23.7±2.3 to 17.8±5.9 for placebo (Cohen's d=0.62; p=0.3 between treatment groups). HAM-D-28 scores decreased from 26.2±4.0 to 12.0±9.8 for LDN, from 26.3±2.6 to 19.8±6.6 for placebo (d=1.15; p=0.097). Montgomery-Asberg Depression Rating Scale (MADRS-10 item) scores decreased from 30.4±4.9 to 12.2±8.4 for LDN, from 30.7±4.3 to 22.8±8.5) for placebo (d=1.45; p=0.035). MADRS-15 item scores decreased from 36.6±6.2 to 13.2±8.8 for LDN, from 36.7±4.2 to 26.0±10.0 for placebo (d=1.49; p=0.035). Clinical Global Improvement Scale-Severity (CGI-S) scores decreased from 4.3±0.5 to 3.0±1.1 for LDN, from 4.3±0.5 to 4.0±0.6 for placebo (d=1.22; p=0.064). LIMITATIONS: Small study; restrictions on allowed antidepressants.
CONCLUSION: LDN augmentation showed some benefit for MDD relapse on dopaminergic agents. Confirmation in larger studies is needed.
Copyright © 2016 Elsevier B.V. All rights reserved.

Entities:  

Keywords:  Breakthrough; Depression; LDN; Naltrexone; Relapse

Mesh:

Substances:

Year:  2016        PMID: 27736689     DOI: 10.1016/j.jad.2016.08.029

Source DB:  PubMed          Journal:  J Affect Disord        ISSN: 0165-0327            Impact factor:   4.839


  9 in total

1.  Attenuation of antidepressant and antisuicidal effects of ketamine by opioid receptor antagonism.

Authors:  Nolan R Williams; Boris D Heifets; Brandon S Bentzley; Christine Blasey; Keith D Sudheimer; Jessica Hawkins; David M Lyons; Alan F Schatzberg
Journal:  Mol Psychiatry       Date:  2019-08-29       Impact factor: 15.992

2.  Opioidergic Agents as Antidepressants: Rationale and Promise.

Authors:  Parnika P Saxena; J Alexander Bodkin
Journal:  CNS Drugs       Date:  2019-01       Impact factor: 5.749

3.  Antidepressant-like effects of BU10119, a novel buprenorphine analogue with mixed κ/μ receptor antagonist properties, in mice.

Authors:  Abdulrahman Almatroudi; Mehrnoosh Ostovar; Christopher P Bailey; Stephen M Husbands; Sarah J Bailey
Journal:  Br J Pharmacol       Date:  2017-11-06       Impact factor: 8.739

4.  Reported Benefits of Low-Dose Naltrexone Appear to Be Independent of the Endogenous Opioid System Involving Proopiomelanocortin Neurons and β-Endorphin.

Authors:  Marissa J Metz; Caitlin M Daimon; Shane T Hentges
Journal:  eNeuro       Date:  2021-06-16

Review 5.  Targeting opioid receptor signaling in depression: do we need selective κ opioid receptor antagonists?

Authors:  Sarah J Bailey; Stephen M Husbands
Journal:  Neuronal Signal       Date:  2018-05-14

6.  Changes in the consumption of antiepileptics and psychotropic medicines after starting low dose naltrexone: A nation-wide register-based controlled before-after study.

Authors:  Guttorm Raknes; Lars Småbrekke
Journal:  Sci Rep       Date:  2019-10-21       Impact factor: 4.379

Review 7.  Augmentative Pharmacological Strategies in Treatment-Resistant Major Depression: A Comprehensive Review.

Authors:  Alice Caldiroli; Enrico Capuzzi; Ilaria Tagliabue; Martina Capellazzi; Matteo Marcatili; Francesco Mucci; Fabrizia Colmegna; Massimo Clerici; Massimiliano Buoli; Antonios Dakanalis
Journal:  Int J Mol Sci       Date:  2021-12-02       Impact factor: 5.923

8.  Depression in Fibromyalgia Patients May Require Low-Dose Naltrexone to Respond: A Case Report.

Authors:  Jagoda Siembida; Brian Johnson
Journal:  Cureus       Date:  2022-02-28

9.  A randomized, double-blind, placebo-controlled, hybrid parallel-arm study of low-dose naltrexone as an adjunctive anti-inflammatory treatment for major depressive disorder.

Authors:  Julia R Plank; Stephanie C Glover; Ben D Moloney; Nicholas R Hoeh; Frederick Sundram; Rachael L Sumner; Suresh Muthukumaraswamy; Joanne C Lin
Journal:  Trials       Date:  2022-09-30       Impact factor: 2.728

  9 in total

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