Literature DB >> 27730680

A Highly Efficient Copper-Mediated Radioiodination Approach Using Aryl Boronic Acids.

Pu Zhang1, Rongqiang Zhuang1, Zhide Guo1, Xinhui Su2, Xiaoyuan Chen3, Xianzhong Zhang1.   

Abstract

A convenient and quantitative radioiodination method by copper-mediated cross-coupling of aryl boronic acids was developed. The mild labeling conditions, ready availability of the boronic acid substrate, simple operation, broad functional group tolerance and excellent radiochemical yield (RCY) make this a practical strategy for radioiodine labeling without further purification.
© 2016 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim.

Entities:  

Keywords:  copper catalysts; molecular imaging; radiochemistry; radioiodination; radiopharmaceuticals

Year:  2016        PMID： 27730680     DOI： 10.1002/chem.201604105

Source DB:  PubMed          Journal:  Chemistry        ISSN： 0947-6539            Impact factor:   5.236


  12 in total

1.  Radioiodinated Small-Molecule Tyrosine Kinase Inhibitor for HER2-Selective SPECT Imaging.

Authors:  Longguang Tang; Chenyu Peng; Bowen Tang; Zijing Li; Xiangyu Wang; Jindian Li; Fei Gao; Lumei Huang; Duo Xu; Pu Zhang; Rongqiang Zhuang; Xinhui Su; Xiaoyuan Chen; Xianzhong Zhang
Journal:  J Nucl Med       Date:  2018-04-13       Impact factor: 10.057

2.  [11C]Cyanation of arylboronic acids in aqueous solutions.

Authors:  Longle Ma; Michael S Placzek; Jacob M Hooker; Neil Vasdev; Steven H Liang
Journal:  Chem Commun (Camb)       Date:  2017-06-05       Impact factor: 6.222

3.  Rapid Cu-Catalyzed [211At]Astatination and [125I]Iodination of Boronic Esters at Room Temperature.

Authors:  Sean W Reilly; Mehran Makvandi; Kuiying Xu; Robert H Mach
Journal:  Org Lett       Date:  2018-03-21       Impact factor: 6.005

4.  Exploration of alcohol-enhanced Cu-mediated radiofluorination toward practical labeling.

Authors:  Dong Zhou; Wenhua Chu; John A Katzenellenbogen
Journal:  J Labelled Comp Radiopharm       Date:  2021-10-19       Impact factor: 1.921

5.  Copper-Mediated Nucleophilic Radiobromination of Aryl Boron Precursors: Convenient Preparation of a Radiobrominated PARP-1 Inhibitor.

Authors:  Dong Zhou; Wenhua Chu; Thomas Voller; John A Katzenellenbogen
Journal:  Tetrahedron Lett       Date:  2018-04-11       Impact factor: 2.415

6.  ImmunoPET: Concept, Design, and Applications.

Authors:  Weijun Wei; Zachary T Rosenkrans; Jianjun Liu; Gang Huang; Quan-Yong Luo; Weibo Cai
Journal:  Chem Rev       Date:  2020-03-23       Impact factor: 60.622

7.  Bifunctional aryliodonium salts for highly efficient radioiodination and astatination of antibodies.

Authors:  F Guérard; L Navarro; Y-S Lee; A Roumesy; C Alliot; M Chérel; M W Brechbiel; J-F Gestin
Journal:  Bioorg Med Chem       Date:  2017-09-19       Impact factor: 3.641

8.  Copper-Mediated Late-stage Radiofluorination: Five Years of Impact on Pre-clinical and Clinical PET Imaging.

Authors:  Jay S Wright; Tanpreet Kaur; Sean Preshlock; Sean S Tanzey; Wade P Winton; Liam S Sharninghausen; Nicholas Wiesner; Allen F Brooks; Melanie S Sanford; Peter J H Scott
Journal:  Clin Transl Imaging       Date:  2020-05-26

9.  Investigation on the reactivity of nucleophilic radiohalogens with arylboronic acids in water: access to an efficient single-step method for the radioiodination and astatination of antibodies.

Authors:  Marion Berdal; Sébastien Gouard; Romain Eychenne; Séverine Marionneau-Lambot; Mikaël Croyal; Alain Faivre-Chauvet; Michel Chérel; Joëlle Gaschet; Jean-François Gestin; François Guérard
Journal:  Chem Sci       Date:  2020-11-23       Impact factor: 9.825

10.  Rapid Iododeboronation with and without Gold Catalysis: Application to Radiolabelling of Arenes.

Authors:  Stacey Webster; Kerry M O'Rourke; Conor Fletcher; Sally L Pimlott; Andrew Sutherland; Ai-Lan Lee
Journal:  Chemistry       Date:  2017-12-14       Impact factor: 5.236
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