Literature DB >> 27720505

Comparison of the Efficacy and Safety of Fixed-dose S-Amlodipine/Telmisartan and Telmisartan in Hypertensive Patients Inadequately Controlled with Telmisartan: A Randomized, Double-blind, Multicenter Study.

Chang Gyu Park1, Tae Hun Ahn2, Eun Ju Cho3, Won Kim4, Hyung Seob Kim5, Ju Yeong Yang6, Jae Geun Ryu7, Cheol Ho Kim8, Min Soo Hyeon9, Seung Je Tak10, Se Jung Im11, Jong Won Ha11, Wook Beom Pyeon12, Je Geon Jae13, Gyu Rok Han14, Jun Hyung Doh15, Sang Wook Im16, Myeong Muk Lee17.   

Abstract

PURPOSE: The objective of this study was to evaluate the efficacy and safety of the fixed-dose combination S-amlodipine plus telmisartan (S-AM/TEL) compared with TEL monotherapy in patients with hypertension inadequately controlled by TEL monotherapy.
METHODS: this study was a randomized, multicenter, double-blind, parallel group, Phase III, 8-week clinical trial to compare the superiority of the S-AM/TEL 2.5/40-mg and S-AM/TEL 5/40-mg combinations with TEL 80-mg mono-therapy. The primary end point was the change in the mean sitting diastolic blood pressure from baseline (week 0) after 8 weeks of therapy between treatment groups.
FINDINGS: Of 325 patients screened, 183 were randomly assigned to 3 groups (61 in the S-AM/TEL 2.5/40-mg group, 60 in the S-AM/TEL 5/40-mg group, and 62 in the TEL 80-mg group). Mean (SD) age was 53.9 (7.5) years, and male patients comprised 87%. No significant differences were found among the 3 groups in baseline characteristics. The primary end points, the changes of mean (SD) diastolic blood pressure at week 8 from the baseline were -10.56 (7.23) mm Hg in the S-AM/TEL 2.5/40-mg group, -12.32 (9.23) mm Hg in the S-AM/TEL 5/40-mg group, and -2.44 (7.92) mm Hg in the TEL 80-mg group. Both the S-AM/TEL 2.5/40-mg group and the S-AM/TEL 5/40-mg group had a statistically superior hypotensive effect compared with the TEL 80-mg group (P < 0.0001 for both). For evaluation of the safety profile, the frequencies of adverse events (AEs) among the groups were also not significantly different (S-AM/TEL 2.5/40-mg group, 18.6%; S-AM/TEL 5/40-mg group, 20%; and TEL 80-mg group, 22.6%), and the incidences of AEs were not different among the groups. The most common AEs were respiratory disorders, followed by headache, dizziness, and peripheral edema. IMPLICATIONS: Treatment with S-AM/TEL 2.5/40 mg and S-AM/TEL 5/40 mg was superior to increasing the TEL dose in terms of hypotensive effect in patients with hypertension inadequately controlled by TEL monotherapy. S-AM/TEL fixed-dose combinations are an effective and tolerable option for patients inadequately responding to TEL monotherapy and also a good option for improving patients' medication adherence. ClinicalTrials.gov identifier: NCT011426100.
Copyright © 2016. Published by Elsevier Inc.

Entities:  

Keywords:  S-amlodipine; blood pressure; fixed-dose combinations; hypertension; single-pill combination; telmisartan

Mesh:

Substances:

Year:  2016        PMID: 27720505     DOI: 10.1016/j.clinthera.2016.09.006

Source DB:  PubMed          Journal:  Clin Ther        ISSN: 0149-2918            Impact factor:   3.393


  2 in total

Review 1.  S-Amlodipine: An Isomer with Difference-Time to Shift from Racemic Amlodipine.

Authors:  Jamshed Dalal; J C Mohan; S S Iyengar; Jagdish Hiremath; Immaneni Sathyamurthy; Sandeep Bansal; Dhiman Kahali; Arup Dasbiswas
Journal:  Int J Hypertens       Date:  2018-05-20       Impact factor: 2.420

2.  Systematic Review with Network Meta-Analysis: Comparative Efficacy and Safety of Combination Therapy with Angiotensin II Receptor Blockers and Amlodipine in Asian Hypertensive Patients.

Authors:  Dae Wook Lee; Mira Jung; Hye Won Wang; Zainah Khan; Philippe Pinton
Journal:  Int J Hypertens       Date:  2019-11-11       Impact factor: 2.420

  2 in total

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