Literature DB >> 27715146

64Cu-PSMA-617 PET/CT Imaging of Prostate Adenocarcinoma: First In-Human Studies.

Bernhard Grubmüller1, Richard P Baum2, Enza Capasso3, Aviral Singh2, Yasaman Ahmadi4, Peter Knoll4, Andreas Floth5, Sergio Righi6, Shahin Zandieh7, Carlo Meleddu3, Shahrokh F Shariat1, Hans Christoph Klingler5, Siroos Mirzaei4.   

Abstract

AIM: The prostate-specific membrane antigen (PSMA) is a cell surface protein, which is overexpressed in nearly all cases of prostate cancer (PCa). PET imaging with 68Ga-PSMA-HBED-CC has recently found widespread application in the diagnosis of recurrent PCa. In this study, the diagnostic potential of 64Cu-labeled PSMA ligand (PSMA-617) PET in patients with PCa has been investigated.
MATERIALS AND METHODS: The study was conducted simultaneously at two nuclear medicine centers, Austria (Vienna, Center 1) and Germany (Bad Berka, Center 2). The patients (n = 29) included in this study were referred for PET (Center 1, 21 patients) or PET/CT (Center 2, 8 patients) imaging with either a high suspicion of recurrent disease or for possible surgical or PSMA radioligand therapy planning. PET images of the whole body were performed at 1 hour p.i. and additional images of the pelvis at 2 hours p.i.
RESULTS: In 23 of 29 patients, at least one focus of pathological tracer uptake suspicious for primary disease in the prostate lobe or recurrent disease was detected. Among healthy organs, the salivary glands, kidneys, and liver showed the highest radiotracer uptake. Lesions suspicious for PCa were detected with excellent contrast as early as 1 hour p.i. with high detection rates even at low prostate-specific antigen (PSA) levels.
CONCLUSION: The preliminary results of this study demonstrate the high potential of 64Cu-PSMA ligand PET/CT imaging in patients with recurrent disease and in the primary staging of selected patients with progressive local disease. The acquired PET images showed an excellent resolution of the detected lesions with very high lesion-to- background contrast. Furthermore, the long half-life of 64Cu allows distribution of the tracer to clinical PET centers that lack radiochemistry facilities for the preparation of 68Ga-PSMA ligand (satellite concept).

Entities:  

Keywords:  64Cu; PET/CT; molecular imaging; prostate cancer; radiopharmaceuticals

Year:  2016        PMID: 27715146     DOI: 10.1089/cbr.2015.1964

Source DB:  PubMed          Journal:  Cancer Biother Radiopharm        ISSN: 1084-9785            Impact factor:   3.099


  17 in total

1.  MUW researcher of the month.

Authors:  Bernhard Grubmüller
Journal:  Wien Klin Wochenschr       Date:  2018-12       Impact factor: 1.704

2.  A PSMA Ligand Labeled with Cobalt-55 for PET Imaging of Prostate Cancer.

Authors:  Johan Hygum Dam; Birgitte Brinkmann Olsen; Christina Baun; Poul Flemming Høilund-Carlsen; Helge Thisgaard
Journal:  Mol Imaging Biol       Date:  2017-12       Impact factor: 3.488

3.  18F-prostate-specific membrane antigen positron emission tomography computed tomography incidental finding in a patient after COVID-19 infection.

Authors:  Siroos Mirzaei; Cherin Farhan; Mario Karolyi
Journal:  World J Nucl Med       Date:  2020-10-02

4.  Soft tissue metastasis of the penis detected by copper-64 labeled prostate-specific membrane antigen positron emission tomography (64Cu-PSMA PET/CT) in a patient with prostate cancer.

Authors:  Cherin Farhan; Siroos Mirzaei
Journal:  Asia Ocean J Nucl Med Biol       Date:  2021

Review 5.  [The role of molecular imaging (PET-CT) in the diagnostic and treatment pf prostate cancer].

Authors:  Siroos Mirzaei; Peter Knoll; Shahin Zandieh
Journal:  Wien Med Wochenschr       Date:  2018-10-22

Review 6.  Current status of theranostics in prostate cancer.

Authors:  Irene Virgolini; Clemens Decristoforo; Alexander Haug; Stefano Fanti; Christian Uprimny
Journal:  Eur J Nucl Med Mol Imaging       Date:  2017-12-28       Impact factor: 9.236

7.  64Cu-PSMA-617: A novel PSMA-targeted radio-tracer for PET imaging in gastric adenocarcinoma xenografted mice model.

Authors:  Xue-Di Han; Chen Liu; Fei Liu; Qing-Hua Xie; Te-Li Liu; Xiao-Yi Guo; Xiao-Xia Xu; Xing Yang; Hua Zhu; Zhi Yang
Journal:  Oncotarget       Date:  2017-05-26

Review 8.  Copper-64: a real theranostic agent.

Authors:  Bianca Gutfilen; Sergio Al Souza; Gianluca Valentini
Journal:  Drug Des Devel Ther       Date:  2018-10-02       Impact factor: 4.162

9.  Establishing Reliable Cu-64 Production Process: From Target Plating to Molecular Specific Tumor Micro-PET Imaging.

Authors:  Qinghua Xie; Hua Zhu; Feng Wang; Xiangxi Meng; Qiushi Ren; Chuanqin Xia; Zhi Yang
Journal:  Molecules       Date:  2017-04-17       Impact factor: 4.411

Review 10.  Nuclear Medicine in Prostate Cancer: A New Era for Radiotracers.

Authors:  Vincenzo Cuccurullo; Giuseppe Danilo Di Stasio; Luigi Mansi
Journal:  World J Nucl Med       Date:  2018 Apr-Jun
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