Literature DB >> 27544669

Enzalutamide as a Fourth- or Fifth-Line Treatment Option for Metastatic Castration-Resistant Prostate Cancer.

Sushil K Badrising1, Vincent van der Noort, Paul Hamberg, Jules L L M Coenen, Maureen J Aarts, Inge M van Oort, Alfons J M van den Eertwegh, Maartje Los, H Pieter van den Berg, Hans Gelderblom, Suzan Vrijaldenhoven, Emile D Kerver, Theo van Voorthuizen, Igle J de Jong, John B Haanen, Andries M Bergman.   

Abstract

OBJECTIVE: To evaluate the efficacy of enzalutamide (Enz) as fourth- or fifth-line treatment in men with metastasized castration-resistant prostate cancer (mCRPC), by analyzing a retrospective cohort of heavily pretreated patients.
METHODS: We evaluated toxicity, overall survival (OS), progression-free survival (PFS) and time to prostate-specific antigen (PSA) progression data from 47 CRPC patients treated with fourth- or fifth-line Enz.
RESULTS: All patients were treated with docetaxel and abiraterone acetate and 42 patients (89%) with cabazitaxel. The median age of the patients was 69 years (IQR, 63-73.5), 79% had bone metastases, 55% had lymph node metastases, and 17% had visceral metastases. The median duration of Enz treatment was 12.0 weeks (IQR, 8.3-20.4), and 11 patients (23%) responded to Enz (maximum PSA decline ≥50%). In general, Enz was well tolerated, with the most frequently reported adverse events being fatigue and nausea. The median OS was 40.1 weeks (95% CI, 25.4-61.4), the median PFS was 12.1 weeks (95% CI, 9.9-14.0) and the median time to PSA progression was 15.7 weeks (95% CI, 14.0-28.7).
CONCLUSIONS: Analysis of this retrospective cohort suggests that Enz is well tolerated and that there is a 23% response rate in heavily pretreated CRPC patients, which is comparable with third-line treatment outcomes.
© 2016 S. Karger AG, Basel.

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Year:  2016        PMID: 27544669     DOI: 10.1159/000448219

Source DB:  PubMed          Journal:  Oncology        ISSN: 0030-2414            Impact factor:   2.935


  6 in total

1.  Activity of cabazitaxel in patients with metastatic castration-resistant prostate cancer after treatment with single or dual regimens of novel androgen receptor-targeting agents.

Authors:  Yukari Bando; Nobuyuki Hinata; Tomoaki Terakawa; Junya Furukawa; Ken-Ichi Harada; Yuzo Nakano; Masato Fujisawa
Journal:  Med Oncol       Date:  2017-08-17       Impact factor: 3.064

2.  Safety and efficacy of cabazitaxel in Japanese patients with castration-resistant prostate cancer.

Authors:  Teppei Yamamoto; Osamu Ishizuka; Hiroshi Oike; Masashi Shiozaki; Tomomi Haba; Tomohiko Oguchi; Kazuyoshi Iijima; Haruaki Kato
Journal:  Prostate Int       Date:  2019-12-02

3.  Osteoblasts derived from mouse mandible enhance tumor growth of prostate cancer more than osteoblasts derived from long bone.

Authors:  Matthew R Eber; Sun H Park; Kelly F Contino; Chirayu M Patel; Fang-Chi Hsu; Yusuke Shiozawa
Journal:  J Bone Oncol       Date:  2020-12-30       Impact factor: 4.072

Review 4.  Progress in Targeted Alpha-Particle-Emitting Radiopharmaceuticals as Treatments for Prostate Cancer Patients with Bone Metastases.

Authors:  Chirayu M Patel; Thaddeus J Wadas; Yusuke Shiozawa
Journal:  Molecules       Date:  2021-04-09       Impact factor: 4.411

Review 5.  Role of the Bone Microenvironment in the Development of Painful Complications of Skeletal Metastases.

Authors:  Sun H Park; Matthew R Eber; D Brooke Widner; Yusuke Shiozawa
Journal:  Cancers (Basel)       Date:  2018-05-10       Impact factor: 6.639

6.  Enzalutamide therapy for advanced prostate cancer: efficacy, resistance and beyond

Authors:  Simon Linder; Henk G van der Poel; Andries M Bergman; Wilbert Zwart; Stefan Prekovic
Journal:  Endocr Relat Cancer       Date:  2018-10-31       Impact factor: 5.678

  6 in total

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