Literature DB >> 27233583

Stability of the Effect of a Standardized Meal on QTc.

Jörg Täubel1, Sara Fernandes1, Georg Ferber2.   

Abstract

BACKGROUND: The assessment of QTc changes after the intake of a standardized meal has been proposed as an alternative approach to prove assay sensitivity when the proarrhythimic potential of a drug is to be excluded in either TQT or intensive Phase I QT studies.
METHODS: In this article, an analysis of the food effect at baseline across periods in two different studies is presented to support the robustness of the method.
RESULTS: The results show that the time-effect attributed to food is stable over different study periods demonstrating consistency of the physiological response triggered by food.
CONCLUSIONS: Stability and reproducibility of the effect is comparable with moxifloxacin.
© 2016 Wiley Periodicals, Inc.

Entities:  

Keywords:  QTc; assay sensitivity; food effect; interval

Mesh:

Substances:

Year:  2016        PMID: 27233583      PMCID: PMC6931674          DOI: 10.1111/anec.12371

Source DB:  PubMed          Journal:  Ann Noninvasive Electrocardiol        ISSN: 1082-720X            Impact factor:   1.468


  11 in total

1.  Shortening of the QT interval after food can be used to demonstrate assay sensitivity in thorough QT studies.

Authors:  Jorg Taubel; Alex H Wong; Asif Naseem; Georg Ferber; A John Camm
Journal:  J Clin Pharmacol       Date:  2011-11-08       Impact factor: 3.126

2.  Insulin at normal physiological levels does not prolong QT(c) interval in thorough QT studies performed in healthy volunteers.

Authors:  Jorg Taubel; Ulrike Lorch; Georg Ferber; Jatinder Singh; Velislav N Batchvarov; Irina Savelieva; A John Camm
Journal:  Br J Clin Pharmacol       Date:  2013-02       Impact factor: 4.335

Review 3.  The IQ-CSRC prospective clinical Phase 1 study: "Can early QT assessment using exposure response analysis replace the thorough QT study?".

Authors:  Borje Darpo; Nenad Sarapa; Christine Garnett; Charles Benson; Corina Dota; Georg Ferber; Venkateswar Jarugula; Lars Johannesen; James Keirns; Kevin Krudys; Catherine Ortemann-Renon; Steve Riley; Danise Rogers-Subramaniam; Norman Stockbridge
Journal:  Ann Noninvasive Electrocardiol       Date:  2013-12-30       Impact factor: 1.468

4.  QTc interval (cardiac repolarization): lengthening after meals.

Authors:  D Nagy; R DeMeersman; D Gallagher; A Pietrobelli; A S Zion; D Daly; S B Heymsfield
Journal:  Obes Res       Date:  1997-11

5.  Reproducibility of QTc interval changes after meal intake.

Authors:  Katerina Hnatkova; Donna Kowalski; James J Keirns; E Marcel van Gelderen; Marek Malik
Journal:  J Electrocardiol       Date:  2015-01-08       Impact factor: 1.438

6.  Establishing assay sensitivity in QT studies: experience with the use of moxifloxacin in an early phase clinical pharmacology study and comparison with its effect in a thorough QT study.

Authors:  Rashmi R Shah; Pierre Maison-Blanche; Thierry Duvauchelle; Philippe Robert; Emmanuel Denis
Journal:  Eur J Clin Pharmacol       Date:  2015-10-01       Impact factor: 2.953

7.  Thorough QT study of the effect of oral moxifloxacin on QTc interval in the fed and fasted state in healthy Japanese and Caucasian subjects.

Authors:  Jorg Taubel; Georg Ferber; Ulrike Lorch; Velislav Batchvarov; Irina Savelieva; A John Camm
Journal:  Br J Clin Pharmacol       Date:  2014-01       Impact factor: 4.335

8.  Acute hyperglycaemia disturbs cardiac repolarization in Type 1 diabetes.

Authors:  D Gordin; C Forsblom; M Rönnback; P-H Groop
Journal:  Diabet Med       Date:  2008-01       Impact factor: 4.359

9.  Single Doses up to 800 mg of E-52862 Do Not Prolong the QTc Interval--A Retrospective Validation by Pharmacokinetic-Pharmacodynamic Modelling of Electrocardiography Data Utilising the Effects of a Meal on QTc to Demonstrate ECG Assay Sensitivity.

Authors:  Jörg Täubel; Georg Ferber; Ulrike Lorch; Duolao Wang; Mariano Sust; A John Camm
Journal:  PLoS One       Date:  2015-08-20       Impact factor: 3.240

10.  QTc changes after meal intake: sex differences and correlates.

Authors:  Katerina Hnatkova; Donna Kowalski; James J Keirns; E Marcel van Gelderen; Marek Malik
Journal:  J Electrocardiol       Date:  2014-08-02       Impact factor: 1.438

View more
  4 in total

Review 1.  Scientific white paper on concentration-QTc modeling.

Authors:  Christine Garnett; Peter L Bonate; Qianyu Dang; Georg Ferber; Dalong Huang; Jiang Liu; Devan Mehrotra; Steve Riley; Philip Sager; Christoffer Tornoe; Yaning Wang
Journal:  J Pharmacokinet Pharmacodyn       Date:  2017-12-05       Impact factor: 2.745

2.  Estimation of the Power of the Food Effect on QTc to Show Assay Sensitivity.

Authors:  Georg Ferber; Sara Fernandes; Jörg Täubel
Journal:  J Clin Pharmacol       Date:  2017-08-17       Impact factor: 3.126

3.  The Cardiovascular Effects of a Meal: J-Tpeak and Tpeak -Tend Assessment and Further Insights Into the Physiological Effects.

Authors:  Jörg Täubel; Georg Ferber; Leen Van Langenhoven; Teresa Del Bianco; Sara Fernandes; Dilshat Djumanov; Jørgen K Kanters; Claus Graff; A John Camm
Journal:  J Clin Pharmacol       Date:  2019-01-11       Impact factor: 3.126

4.  A Phase 1 Study to Investigate the Effects of Cortexolone 17α-Propionate, Also Known as Clascoterone, on the QT Interval Using the Meal Effect to Demonstrate ECG Assay Sensitivity.

Authors:  Jörg Täubel; Alessandro Mazzetti; Georg Ferber; William Burch; Sara Fernandes; Avani Patel; Christopher S Spencer; Anne Freier; Claus Graff; Jørgen K Kanters; John Camm
Journal:  Clin Pharmacol Drug Dev       Date:  2021-05-03
  4 in total

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