Literature DB >> 27092721

Celecoxib and Pioglitazone as Potential Therapeutics for Regulating TGF-β-Induced Hyaluronan in Dysthyroid Myopathy.

Anny M S Cheng1, Han Y Yin2, Angus Chen3, Ya-Wen Liu4, Mei-Chun Chuang4, Hua He1, Sean Tighe1, Hosam Sheha1, Shu-Lang Liao5.   

Abstract

PURPOSE: To investigate the role of extraocular muscles (EOM) myoblasts in Graves ophthalmopathy (GO) pathology and the effect of a cyclooxygenase (COX)-2 inhibitor and a peroxisome proliferator-activated receptor (PPAR)-γ agonist in its treatment.
METHODS: Myoblasts were isolated and cultured from EOM of 10 patients with GO and 4 without (non-GO). The cultured myoblasts were treated with IFN-γ, insulin-like growth factor (IGF)-1, IL-1β, and TNF-α, and the effect on PPAR-γ, COX-2, TGF-β, and thyroid stimulating hormone receptor (TSH-R) expressions were assessed using real-time (RT)-PCR, ELISA, and Western blot. The effect of a COX-2 inhibitor and a PPAR-γ agonist on the expression of TGF-β, hyaluronan synthases (HAS)-1, -2, and -3, and hyaluronan (HA) were further evaluated.
RESULTS: Real-time PCR showed significant upregulation in PPAR-γ, COX-2, TGF-β, and TSH-R mRNA expression in GO myoblasts when treated with TNF-α but not in the non-GO. While IFN-γ and IGF-1 had no significant effect, IL-1β did upregulate COX-2 expression. These results were further confirmed by ELISA and Western blotting. Tumor necrosis factor α-induced TGF-β in turn significantly increased HA expression and HAS3 level, but not HAS1 and HAS2. The cyclooxygenase 2 inhibitor and PPAR-γ agonist substantially diminished this TNF-α-induced TGF-β, HA, and HAS3 expression.
CONCLUSIONS: These results demonstrate the role of EOM myoblasts in the pathogenesis of GO. The cyclooxygenase 2 inhibitor and PPAR-γ agonist in this study are potential treatments for GO due to their ability to suppress TNF-α-induced TGF-β, HAS, and HA upregulation.

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Year:  2016        PMID: 27092721     DOI: 10.1167/iovs.15-18018

Source DB:  PubMed          Journal:  Invest Ophthalmol Vis Sci        ISSN: 0146-0404            Impact factor:   4.799


  6 in total

1.  Sphingosine-1-phosphate is involved in inflammatory reactions in patients with Graves' orbitopathy.

Authors:  Yuri Seo; Min Kyung Chae; Sol Ah Han; Eun Jig Lee; Joon H Lee; Jin Sook Yoon
Journal:  Inflamm Res       Date:  2017-03-31       Impact factor: 4.575

Review 2.  The role of transforming growth factor beta in thyroid autoimmunity: current knowledge and future perspectives.

Authors:  Efstratios Kardalas; Evangelos Sakkas; Marek Ruchala; Djuro Macut; George Mastorakos
Journal:  Rev Endocr Metab Disord       Date:  2021-09-16       Impact factor: 6.514

Review 3.  Thinking inside the box: Current insights into targeting orbital tissue remodeling and inflammation in thyroid eye disease.

Authors:  Vardaan Gupta; Christine L Hammond; Elisa Roztocil; Mithra O Gonzalez; Steven E Feldon; Collynn F Woeller
Journal:  Surv Ophthalmol       Date:  2021-09-04       Impact factor: 6.197

Review 4.  TGF-β Physiology as a Novel Therapeutic Target Regarding Autoimmune Thyroid Diseases: Where Do We Stand and What to Expect.

Authors:  Efstratios Kardalas; Spyridoula Maraka; Maria Papagianni; George Paltoglou; Charalampos Siristatidis; George Mastorakos
Journal:  Medicina (Kaunas)       Date:  2021-06-14       Impact factor: 2.430

Review 5.  The roles of PPARγ and its agonists in autoimmune diseases: A comprehensive review.

Authors:  Yu Liu; Jiayu Wang; Shuangyan Luo; Yi Zhan; Qianjin Lu
Journal:  J Autoimmun       Date:  2020-07-01       Impact factor: 7.094

6.  The Effect of Prostaglandin Analogue Bimatoprost on Thyroid-Associated Orbitopathy.

Authors:  Catherine J Choi; Wensi Tao; Ravi Doddapaneni; Zenith Acosta-Torres; Nathan W Blessing; Bradford W Lee; Daniel Pelaez; Sara T Wester
Journal:  Invest Ophthalmol Vis Sci       Date:  2018-12-03       Impact factor: 4.799

  6 in total

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