Literature DB >> 27043419

Novel chemoselective (18)F-radiolabeling of thiol-containing biomolecules under mild aqueous conditions.

Aristeidis Chiotellis1, Filippo Sladojevich, Linjing Mu, Adrienne Müller Herde, Ibai E Valverde, Vladimir Tolmachev, Roger Schibli, Simon M Ametamey, Thomas L Mindt.   

Abstract

We report a novel prosthetic group based on a heterocyclic methylsulfone derivative for the rapid, stable, and chemoselective (18)F-labeling of thiol-containing (bio)molecules under mild aqueous reaction conditions. Compared to established maleimide approaches, the new methodology displays some clear advantages for imaging probe development.

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Year:  2016        PMID： 27043419     DOI： 10.1039/c6cc01982j

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  10 in total

Review 1.  Arylation Chemistry for Bioconjugation.

Authors:  Chi Zhang; Ekaterina V Vinogradova; Alexander M Spokoyny; Stephen L Buchwald; Bradley L Pentelute
Journal:  Angew Chem Int Ed Engl       Date:  2019-02-15       Impact factor: 15.336

Review 2.  18 F-Labeling of Sensitive Biomolecules for Positron Emission Tomography.

Authors:  Hema S Krishnan; Longle Ma; Neil Vasdev; Steven H Liang
Journal:  Chemistry       Date:  2017-09-01       Impact factor: 5.236

3.  Direct 11CN-Labeling of Unprotected Peptides via Palladium-Mediated Sequential Cross-Coupling Reactions.

Authors:  Wenjun Zhao; Hong Geun Lee; Stephen L Buchwald; Jacob M Hooker
Journal:  J Am Chem Soc       Date:  2017-05-17       Impact factor: 15.419

4.  Synthesis of [18 F]Fluoroarenes by Nucleophilic Radiofluorination of N-Arylsydnones.

Authors:  Maruthi Kumar Narayanam; Gaoyuan Ma; Pier Alexandre Champagne; Kendall N Houk; Jennifer M Murphy
Journal:  Angew Chem Int Ed Engl       Date:  2017-09-07       Impact factor: 15.336

5.  Synthesis and Bioconjugation of Thiol-Reactive Reagents for the Creation of Site-Selectively Modified Immunoconjugates.

Authors:  Maria Davydova; Guillaume Dewaele Le Roi; Pierre Adumeau; Brian M Zeglis
Journal:  J Vis Exp       Date:  2019-03-06       Impact factor: 1.355

Review 6.  Click Chemistry and Radiochemistry: The First 10 Years.

Authors:  Jan-Philip Meyer; Pierre Adumeau; Jason S Lewis; Brian M Zeglis
Journal:  Bioconjug Chem       Date:  2016-11-22       Impact factor: 4.774

Review 7.  Affibody Molecules as Targeting Vectors for PET Imaging.

Authors:  Vladimir Tolmachev; Anna Orlova
Journal:  Cancers (Basel)       Date:  2020-03-11       Impact factor: 6.639

8.  18F-Trifluoromethanesulfinate Enables Direct C-H 18F-Trifluoromethylation of Native Aromatic Residues in Peptides.

Authors:  Choon Wee Kee; Osman Tack; Florian Guibbal; Thomas C Wilson; Patrick G Isenegger; Mateusz Imiołek; Stefan Verhoog; Michael Tilby; Giulia Boscutti; Sharon Ashworth; Juliette Chupin; Roxana Kashani; Adeline W J Poh; Jane K Sosabowski; Sven Macholl; Christophe Plisson; Bart Cornelissen; Michael C Willis; Jan Passchier; Benjamin G Davis; Véronique Gouverneur
Journal:  J Am Chem Soc       Date:  2020-01-13       Impact factor: 15.419

Review 9.  Recent Advances in Bioorthogonal Click Chemistry for Efficient Synthesis of Radiotracers and Radiopharmaceuticals.

Authors:  Sajid Mushtaq; Seong-Jae Yun; Jongho Jeon
Journal:  Molecules       Date:  2019-10-02       Impact factor: 4.411

10.  Thiol-Reactive PODS-Bearing Bifunctional Chelators for the Development of EGFR-Targeting [18F]AlF-Affibody Conjugates.

Authors:  Chiara Da Pieve; Ata Makarem; Stephen Turnock; Justyna Maczynska; Graham Smith; Gabriela Kramer-Marek
Journal:  Molecules       Date:  2020-03-29       Impact factor: 4.411
  10 in total

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