Literature DB >> 26898835

Enhancing the selectivity of kinase inhibitors in oncology: a chemical biology perspective.

Sean Maddox1, David Hecht2, Jeffrey L Gustafson1.   

Abstract

Keywords:  chemical probe; drug discovery; kinase inhibition; oncology; target selectivity

Mesh:

Substances:

Year:  2016        PMID: 26898835     DOI: 10.4155/fmc.15.193

Source DB:  PubMed          Journal:  Future Med Chem        ISSN: 1756-8919            Impact factor:   3.808


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  1 in total

1.  Effects of rigidity on the selectivity of protein kinase inhibitors.

Authors:  Amir Assadieskandar; Caiqun Yu; Pierre Maisonneuve; Xu Liu; Ying-Chu Chen; G K Surya Prakash; Igor Kurinov; Frank Sicheri; Chao Zhang
Journal:  Eur J Med Chem       Date:  2018-01-31       Impact factor: 6.514

  1 in total

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