Literature DB >> 26860632

A Phase II trial of tandutinib (MLN 518) in combination with bevacizumab for patients with recurrent glioblastoma.

Yazmin Odia1, Joohee Sul2, Joanna H Shih3, Teri N Kreisl1, John A Butman4, Fabio M Iwamoto1, Howard A Fine5.   

Abstract

AIM: A Phase II trial of bevacizumab plus tandutinib.
METHODS: We enrolled 41 recurrent, bevacizumab-naive glioblastoma patients for a trial of bevacizumab plus tandutinib. Median age was 55 and 71% were male. Treatment consisted of tandutinib 500 mg two-times a day (b.i.d.) and bevacizumab 10 mg/kg every 2 weeks starting day 15. Of 37 (90%) evaluable, nine (24%) had partial response. RESULTS &
CONCLUSION: Median overall and progression-free survival was 11 and 4.1 months; progression-free survival at 6 months was 23%. All patients suffered treatment-related toxicities; common grade ≥3 toxicities were hypertension (17.1%), muscle weakness (17.1%), lymphopenia (14.6%) and hypophosphatemia (9.8%). Four of six with grade ≥3 tandutinib-related myasthenic-like muscle weakness had electromyography-proven neuromuscular junction pathology. Tandutinib with bevacizumab was as effective but more toxic than bevacizumab monotherapy.

Entities:  

Keywords:  bevacizumab; glioblastoma; tandutinib

Mesh:

Substances:

Year:  2016        PMID: 26860632      PMCID: PMC5514626          DOI: 10.2217/cns-2015-0010

Source DB:  PubMed          Journal:  CNS Oncol        ISSN: 2045-0907


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