Literature DB >> 26826439

Perspectives on the amorphisation/milling relationship in pharmaceutical materials.

M Descamps1, J F Willart2.   

Abstract

This paper presents an overview of recent advances in understanding the role of the amorphous state in the physical and chemical transformations of pharmaceutical materials induced by mechanical milling. The following points are addressed: (1) Is milling really able to amorphise crystals?, (2) Conditions for obtaining an amorphisation, (3) Milling of hydrates, (4) Producing amorphous state without changing the chemical nature, (5) Milling induced crystal to crystal transformations: mediation by an amorphous state, (6) Nature of the amorphous state obtained by milling, (7) Milling of amorphous compounds: accelerated aging or rejuvenation, (8) Specific recrystallisation behaviour, and (9) Toward a rationalisation and conceptual framework.
Copyright © 2016 Elsevier B.V. All rights reserved.

Keywords:  Amorphous; Milling; Pharmaceuticals; Phase transitions; Polymorphism

Mesh：

Year:  2016        PMID： 26826439     DOI： 10.1016/j.addr.2016.01.011

Source DB:  PubMed          Journal:  Adv Drug Deliv Rev        ISSN： 0169-409X            Impact factor:   15.470


  8 in total

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2.  An Enthalpy-Balance Model for Timewise Evolution of Temperature during Wet Stirred Media Milling of Drug Suspensions.

Authors:  Gulenay Guner; Sherif Elashri; Mirsad Mehaj; Natasha Seetharaman; Helen F Yao; Donald J Clancy; Ecevit Bilgili
Journal:  Pharm Res       Date:  2022-08-02       Impact factor: 4.580

3.  Challenges of Mechanochemistry: Is In Situ Real-Time Quantitative Phase Analysis Always Reliable? A Case Study of Organic Salt Formation.

Authors:  Adam A L Michalchuk; Ivan A Tumanov; Sumit Konar; Simon A J Kimber; Colin R Pulham; Elena V Boldyreva
Journal:  Adv Sci (Weinh)       Date:  2017-05-08       Impact factor: 16.806

4.  Physicochemical characterization, the Hirshfeld surface, and biological evaluation of two meloxicam compounding pharmacy samples.

Authors:  Luciana F A Romani; Maria I Yoshida; Elionai C L Gomes; Renes R Machado; Felipe F Rodrigues; Márcio M Coelho; Marcelo A Oliveira; Maria B Freitas-Marques; Rosane A S San Gil; Wagner N Mussel
Journal:  J Pharm Anal       Date:  2017-12-19

5.  Preparation of curcumin self-micelle solid dispersion with enhanced bioavailability and cytotoxic activity by mechanochemistry.

Authors:  Qihong Zhang; Nikolay E Polyakov; Yulia S Chistyachenko; Mikhail V Khvostov; Tatjana S Frolova; Tatjana G Tolstikova; Alexandr V Dushkin; Weike Su
Journal:  Drug Deliv       Date:  2018-11       Impact factor: 6.419

6.  Understanding Concomitant Physical and Chemical Transformations of Simvastatin During Dry Ball Milling.

Authors:  Dattatray Modhave; Isha Saraf; Anjali Karn; Amrit Paudel
Journal:  AAPS PharmSciTech       Date:  2020-05-21       Impact factor: 3.246

7.  Mechanochemical preparation of triptolide-loaded self-micelle solid dispersion with enhanced oral bioavailability and improved anti-tumor activity.

Authors:  Dabu Zhu; Qiuqin Zhang; Yifang Chen; Minghua Xie; Jianbo Li; Shen Yao; Ming Li; Zhao Lou; Yue Cai; Xuanrong Sun
Journal:  Drug Deliv       Date:  2022-12       Impact factor: 6.819

8.  Stoichiometrically Governed Curcumin Solid Dispersion and Its Cytotoxic Evaluation on Colorectal Adenocarcinoma Cells.

Authors:  Jamal Moideen Muthu Mohamed; Ali Alqahtani; Fazil Ahmad; V Krishnaraju; K Kalpana
Journal:  Drug Des Devel Ther       Date:  2020-11-02       Impact factor: 4.162
  8 in total

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