Literature DB >> 26795290

Tracer Kinetic Analysis of (S)-¹⁸F-THK5117 as a PET Tracer for Assessing Tau Pathology.

My Jonasson1, Anders Wall2, Konstantinos Chiotis3, Laure Saint-Aubert3, Helena Wilking4, Margareta Sprycha4, Beatrice Borg4, Alf Thibblin4, Jonas Eriksson5, Jens Sörensen2, Gunnar Antoni5, Agneta Nordberg6, Mark Lubberink1.   

Abstract

UNLABELLED: Because a correlation between tau pathology and the clinical symptoms of Alzheimer disease (AD) has been hypothesized, there is increasing interest in developing PET tracers that bind specifically to tau protein. The aim of this study was to evaluate tracer kinetic models for quantitative analysis and generation of parametric images for the novel tau ligand (S)-(18)F-THK5117.
METHODS: Nine subjects (5 with AD, 4 with mild cognitive impairment) received a 90-min dynamic (S)-(18)F-THK5117 PET scan. Arterial blood was sampled for measurement of blood radioactivity and metabolite analysis. Volume-of-interest (VOI)-based analysis was performed using plasma-input models; single-tissue and 2-tissue (2TCM) compartment models and plasma-input Logan and reference tissue models; and simplified reference tissue model (SRTM), reference Logan, and SUV ratio (SUVr). Cerebellum gray matter was used as the reference region. Voxel-level analysis was performed using basis function implementations of SRTM, reference Logan, and SUVr. Regionally averaged voxel values were compared with VOI-based values from the optimal reference tissue model, and simulations were made to assess accuracy and precision. In addition to 90 min, initial 40- and 60-min data were analyzed.
RESULTS: Plasma-input Logan distribution volume ratio (DVR)-1 values agreed well with 2TCM DVR-1 values (R(2)= 0.99, slope = 0.96). SRTM binding potential (BP(ND)) and reference Logan DVR-1 values were highly correlated with plasma-input Logan DVR-1 (R(2)= 1.00, slope ≈ 1.00) whereas SUVr(70-90)-1 values correlated less well and overestimated binding. Agreement between parametric methods and SRTM was best for reference Logan (R(2)= 0.99, slope = 1.03). SUVr(70-90)-1 values were almost 3 times higher than BP(ND) values in white matter and 1.5 times higher in gray matter. Simulations showed poorer accuracy and precision for SUVr(70-90)-1 values than for the other reference methods. SRTM BP(ND) and reference Logan DVR-1 values were not affected by a shorter scan duration of 60 min.
CONCLUSION: SRTM BP(ND) and reference Logan DVR-1 values were highly correlated with plasma-input Logan DVR-1 values. VOI-based data analyses indicated robust results for scan durations of 60 min. Reference Logan generated quantitative (S)-(18)F-THK5117 DVR-1 parametric images with the greatest accuracy and precision and with a much lower white-matter signal than seen with SUVr(70-90)-1 images.
© 2016 by the Society of Nuclear Medicine and Molecular Imaging, Inc.

Entities:  

Keywords:  Alzheimer’s disease; kinetic modeling; parametric images; positron emission tomography; tau

Mesh:

Substances:

Year:  2016        PMID: 26795290     DOI: 10.2967/jnumed.115.158519

Source DB:  PubMed          Journal:  J Nucl Med        ISSN: 0161-5505            Impact factor:   10.057


  25 in total

1.  Characterization of the radiolabeled metabolite of tau PET tracer 18F-THK5351.

Authors:  Ryuichi Harada; Shozo Furumoto; Tetsuro Tago; Katsutoshi Furukawa; Aiko Ishiki; Naoki Tomita; Ren Iwata; Manabu Tashiro; Hiroyuki Arai; Kazuhiko Yanai; Yukitsuka Kudo; Nobuyuki Okamura
Journal:  Eur J Nucl Med Mol Imaging       Date:  2016-07-19       Impact factor: 9.236

Review 2.  Future Directions in Imaging Neurodegeneration.

Authors:  Joseph C Masdeu
Journal:  Curr Neurol Neurosci Rep       Date:  2017-01       Impact factor: 5.081

3.  Evaluation of 18F-RO-948 PET for Quantitative Assessment of Tau Accumulation in the Human Brain.

Authors:  Hiroto Kuwabara; Robert A Comley; Edilio Borroni; Michael Honer; Kelly Kitmiller; Joshua Roberts; Lorena Gapasin; Anil Mathur; Gregory Klein; Dean F Wong
Journal:  J Nucl Med       Date:  2018-08-10       Impact factor: 10.057

4.  Comparability of [18F]THK5317 and [11C]PIB blood flow proxy images with [18F]FDG positron emission tomography in Alzheimer's disease.

Authors:  Elena Rodriguez-Vieitez; Antoine Leuzy; Konstantinos Chiotis; Laure Saint-Aubert; Anders Wall; Agneta Nordberg
Journal:  J Cereb Blood Flow Metab       Date:  2016-07-20       Impact factor: 6.200

5.  In Vivo Comparison of Tau Radioligands 18F-THK-5351 and 18F-THK-5317.

Authors:  Tobey J Betthauser; Patrick J Lao; Dhanabalan Murali; Todd E Barnhart; Shozo Furumoto; Nobuyuki Okamura; Charles K Stone; Sterling C Johnson; Bradley T Christian
Journal:  J Nucl Med       Date:  2016-11-10       Impact factor: 10.057

6.  The cerebellum shrinks faster than normal ageing in Alzheimer's disease but not in mild cognitive impairment.

Authors:  Hossein Tabatabaei-Jafari; Erin Walsh; Marnie E Shaw; Nicolas Cherbuin
Journal:  Hum Brain Mapp       Date:  2017-03-21       Impact factor: 5.038

7.  Spatially constrained kinetic modeling with dual reference tissues improves 18F-flortaucipir PET in studies of Alzheimer disease.

Authors:  Yun Zhou; Shaney Flores; Syahir Mansor; Russ C Hornbeck; Zhude Tu; Joel S Perlmutter; Beau Ances; John C Morris; Robert J Gropler; Tammie L S Benzinger
Journal:  Eur J Nucl Med Mol Imaging       Date:  2021-02-18       Impact factor: 9.236

8.  Cerebrospinal Fluid Clearance in Alzheimer Disease Measured with Dynamic PET.

Authors:  Mony J de Leon; Yi Li; Nobuyuki Okamura; Wai H Tsui; Les A Saint-Louis; Lidia Glodzik; Ricardo S Osorio; Juan Fortea; Tracy Butler; Elizabeth Pirraglia; Silvia Fossati; Hee-Jin Kim; Roxana O Carare; Maiken Nedergaard; Helene Benveniste; Henry Rusinek
Journal:  J Nucl Med       Date:  2017-03-16       Impact factor: 10.057

9.  In Vivo Characterization and Quantification of Neurofibrillary Tau PET Radioligand 18F-MK-6240 in Humans from Alzheimer Disease Dementia to Young Controls.

Authors:  Tobey J Betthauser; Karly A Cody; Matthew D Zammit; Dhanabalan Murali; Alexander K Converse; Todd E Barnhart; Charles K Stone; Howard A Rowley; Sterling C Johnson; Bradley T Christian
Journal:  J Nucl Med       Date:  2018-05-18       Impact factor: 10.057

Review 10.  An Update on the State of Tau Radiotracer Development: a Brief Review.

Authors:  Grant Rigney; Cyrus Ayubcha; Thomas J Werner; Abass Alavi
Journal:  Mol Imaging Biol       Date:  2021-05-13       Impact factor: 3.488

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