Literature DB >> 26731724

Temsirolimus in women with platinum-refractory/resistant ovarian cancer or advanced/recurrent endometrial carcinoma. A phase II study of the AGO-study group (AGO-GYN8).

Günter Emons1, Christian Kurzeder2, Barbara Schmalfeldt3, Petra Neuser4, Nikolaus de Gregorio5, Jacobus Pfisterer6, Tjoung-Won Park-Simon7, Sven Mahner8, Willibald Schröder9, Hans-Joachim Lück10, Martin Leonhard Heubner11, Lars Hanker12, Falk Thiel13, Felix Hilpert14.   

Abstract

OBJECTIVES: To evaluate activity and toxicity of mTOR inhibitor temsirolimus in patients with platinum-refractory/resistant ovarian cancer (OC) or advanced/recurrent endometrial carcinoma (EC).
METHODS: Women with epithelial ovarian, fallopian tube or primary peritoneal cancer were eligible, when they had progression during treatment with a platinum based regimen or within 6 months after receiving a platinum based regimen and a previous taxane treatment. Women with advanced/recurrent EC, no longer amenable to curative surgery and/or radiotherapy were eligible when they had no previous or only adjuvant chemotherapy. Preceding endocrine therapy for metastatic/recurrent disease was allowed. Patients received weekly IV infusions of 25mg temsirolimus. Primary endpoint was progression free survival rate after 4 months (OC) or 6 months (EC). A two stage design was applied.
RESULTS: Forty-four patients (OC: n=22; EC: n=22) were enrolled and received temsirolimus treatment. Median age was 56 years (OC) or 63 years (EC). After eight weeks of treatment, 10 of 21 evaluable patients in the OC cohort and 8 of 20 evaluable patients in the EC cohort had progressive disease. Thus efficacy did not meet the predefined levels during the first stage of recruitment and the trial was stopped. Some patients in both cohorts had long lasting PFS (>7 months). Toxicity of temsirolimus was mild.
CONCLUSIONS: Temsirolimus treatment was well tolerated in our patients, but did not meet the predefined efficacy criteria. In our study as in other trials on rapalogs in OC or EC, a few patients had long lasting disease stabilisations.
Copyright © 2015. Published by Elsevier Inc.

Entities:  

Keywords:  Endometrial cancer; Ovarian cancer; Rapalog; Temsirolimus; mTOR inhibitor

Mesh:

Substances:

Year:  2015        PMID: 26731724     DOI: 10.1016/j.ygyno.2015.12.025

Source DB:  PubMed          Journal:  Gynecol Oncol        ISSN: 0090-8258            Impact factor:   5.482


  21 in total

Review 1.  Targeting the PI3K pathway and DNA damage response as a therapeutic strategy in ovarian cancer.

Authors:  Tzu-Ting Huang; Erika J Lampert; Cynthia Coots; Jung-Min Lee
Journal:  Cancer Treat Rev       Date:  2020-04-10       Impact factor: 12.111

2.  ESGO/ESTRO/ESP Guidelines for the management of patients with endometrial carcinoma.

Authors:  Nicole Concin; Carien L Creutzberg; Ignace Vergote; David Cibula; Mansoor Raza Mirza; Simone Marnitz; Jonathan A Ledermann; Tjalling Bosse; Cyrus Chargari; Anna Fagotti; Christina Fotopoulou; Antonio González-Martín; Sigurd F Lax; Domenica Lorusso; Christian Marth; Philippe Morice; Remi A Nout; Dearbhaile E O'Donnell; Denis Querleu; Maria Rosaria Raspollini; Jalid Sehouli; Alina E Sturdza; Alexandra Taylor; Anneke M Westermann; Pauline Wimberger; Nicoletta Colombo; François Planchamp; Xavier Matias-Guiu
Journal:  Virchows Arch       Date:  2021-02       Impact factor: 4.064

3.  Role of YAP1 as a Marker of Sensitivity to Dual AKT and P70S6K Inhibition in Ovarian and Uterine Malignancies.

Authors:  Rebecca A Previs; Guillermo N Armaiz-Pena; Cristina Ivan; Heather J Dalton; Rajesha Rupaimoole; Jean M Hansen; Yasmin Lyons; Jie Huang; Monika Haemmerle; Michael J Wagner; Kshipra M Gharpure; Archana S Nagaraja; Justyna Filant; Michael H McGuire; Kyunghee Noh; Piotr L Dorniak; Sarah L Linesch; Lingegowda S Mangala; Sunila Pradeep; Sherry Y Wu; Anil K Sood
Journal:  J Natl Cancer Inst       Date:  2017-07-01       Impact factor: 13.506

4.  Phase II, 2-stage, 2-arm, PIK3CA mutation stratified trial of MK-2206 in recurrent endometrial cancer.

Authors:  Andrea P Myers; Panagiotis A Konstantinopoulos; William T Barry; Weixiu Luo; Russell R Broaddus; Vicky Makker; Ronny Drapkin; Joyce Liu; Austin Doyle; Neil S Horowitz; Funda Meric-Bernstam; Michael Birrer; Carol Aghajanian; Robert L Coleman; Gordon B Mills; Lewis C Cantley; Ursula A Matulonis; Shannon N Westin
Journal:  Int J Cancer       Date:  2019-12-13       Impact factor: 7.396

5.  Targeting BET Proteins BRD2 and BRD3 in Combination with PI3K-AKT Inhibition as a Therapeutic Strategy for Ovarian Clear Cell Carcinoma.

Authors:  Shogo Shigeta; Goldie Y L Lui; Reid Shaw; Russell Moser; Kay E Gurley; Grace Durenberger; Rachele Rosati; Robert L Diaz; Tan A Ince; Elizabeth M Swisher; Carla Grandori; Christopher J Kemp
Journal:  Mol Cancer Ther       Date:  2021-01-28       Impact factor: 6.009

Review 6.  Molecular Characterization of Epithelial Ovarian Cancer: Implications for Diagnosis and Treatment.

Authors:  Veronica Rojas; Kim M Hirshfield; Shridar Ganesan; Lorna Rodriguez-Rodriguez
Journal:  Int J Mol Sci       Date:  2016-12-15       Impact factor: 5.923

7.  PI3K/AKT/mTOR Pathway in Ovarian Cancer Treatment: Are We on the Right Track?

Authors:  Maria Luisa Gasparri; Erlisa Bardhi; Ilary Ruscito; Andrea Papadia; Ammad Ahmad Farooqi; Claudia Marchetti; Giorgio Bogani; Irene Ceccacci; Michael D Mueller; Pierluigi Benedetti Panici
Journal:  Geburtshilfe Frauenheilkd       Date:  2017-10-26       Impact factor: 2.915

8.  PaccMann: a web service for interpretable anticancer compound sensitivity prediction.

Authors:  Joris Cadow; Jannis Born; Matteo Manica; Ali Oskooei; María Rodríguez Martínez
Journal:  Nucleic Acids Res       Date:  2020-07-02       Impact factor: 16.971

Review 9.  A Review of mTOR Pathway Inhibitors in Gynecologic Cancer.

Authors:  Andréia Cristina de Melo; Eduardo Paulino; Álvaro Henrique Ingles Garces
Journal:  Oxid Med Cell Longev       Date:  2017-02-13       Impact factor: 6.543

10.  Therapeutic efficacy of liposomal Grb2 antisense oligodeoxynucleotide (L-Grb2) in preclinical models of ovarian and uterine cancer.

Authors:  Olivia D Lara; Emine Bayraktar; Paola Amero; Shaolin Ma; Cristina Ivan; Wei Hu; Ying Wang; Lingegowda S Mangala; Prasanta Dutta; Pratip Bhattacharya; Ana Tari Ashizawa; Gabriel Lopez-Berestein; Cristian Rodriguez-Aguayo; Anil K Sood
Journal:  Oncotarget       Date:  2020-07-21
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