Literature DB >> 26684309

Tacrolimus for children with refractory nephrotic syndrome: a one-year prospective, multicenter, and open-label study of Tacrobell®, a generic formula.

Eun Mi Yang1,2, Sang Taek Lee3, Hyun Jin Choi2, Hee Yeon Cho3, Joo Hoon Lee4, Hee Gyung Kang5,6, Young Seo Park4,7, Hae Il Cheong8, Il-Soo Ha2,8.   

Abstract

BACKGROUND: Cyclosporine A and tacrolimus (TAC) are often used as a second-line treatment for children with refractory nephrotic syndrome (NS). This study was undertaken to investigate the efficacy and safety of Tacrobell®, a locally produced generic form of TAC.
METHODS: This study was a one-year prospective, open-label, single-arm, multicenter trial. Fourty-four children with steroid-dependent NS (SDNS) and 33 children with steroid-resistant NS (SRNS) were enrolled. The primary endpoints were defined as the remission rates, whereas the secondary endpoints were recognized as the duration of remission and adverse effects of TAC.
RESULTS: After one-year treatment, 34 (77.3%) of the 44 patients with SDNS were in complete remission, and 6 (13.6%) were in partial remission. Nineteen (43.2%) patients did not relapse during the study; for those who did relapse, the mean duration of remission was 4.6±2.9 months. The number of relapse episodes during the study period (0.90 per patient-year) was significantly lower than that in the preceding year (2.8 per patient-year). After treatment for 3 and 6 months, 12 (36.4%) of the 33 patients with SRNS were in remission, and after treatment for 12 months, the number of patients had increased to 13 (39.4%). The mean time to achieve remission was 4.0±3.2 months. After remission (duration, 3.7±2.7 months), 12 (54.5%) of 22 patients relapsed. The fasting blood glucose and blood pressure levels during the therapy were similar to those at the time of study entry.
CONCLUSIONS: Treatment with Tacrobell® was effective and safe for children with refractory NS. The efficacy of this generic form of TAC was better than that of the original TAC formula.

Entities:  

Keywords:  generic drugs; nephrotic syndrome; tacrolimus

Mesh:

Substances:

Year:  2015        PMID: 26684309     DOI: 10.1007/s12519-015-0062-y

Source DB:  PubMed          Journal:  World J Pediatr            Impact factor:   2.764


  36 in total

1.  Tacrolimus in steroid-resistant and steroid-dependent nephrotic syndrome.

Authors:  T H Westhoff; S Schmidt; W Zidek; J Beige; M van der Giet
Journal:  Clin Nephrol       Date:  2006-06       Impact factor: 0.975

2.  A randomized, open-label, two-period, crossover bioavailability study of two oral formulations of tacrolimus in healthy Korean adults.

Authors:  Kyungsoo Park; Yu Seun Kim; Kwang-Il Kwon; Min Soo Park; Yoon Jung Lee; Kyung Hwan Kim
Journal:  Clin Ther       Date:  2007-01       Impact factor: 3.393

3.  Second-line options for refractory steroid-sensitive and -resistant nephrotic syndrome.

Authors:  Jun Oh; Markus J Kemper
Journal:  Expert Rev Clin Pharmacol       Date:  2010-07       Impact factor: 5.045

4.  Renal function and tubular phosphate handling in long-term cyclosporine- and tacrolimus-based immunosuppression in kidney transplantation.

Authors:  K Falkiewicz; D Kamińska; W Nahaczewska; M Boratyńska; H Owczarek; M Klinger; M Woźniak; D Patrzałek; P Szyber
Journal:  Transplant Proc       Date:  2006 Jan-Feb       Impact factor: 1.066

5.  Primary focal segmental glomerulosclerosis in children: prognostic factors.

Authors:  R Martinelli; A S Okumura; L J Pereira; H Rocha
Journal:  Pediatr Nephrol       Date:  2001-08       Impact factor: 3.714

6.  Management of steroid-resistant focal segmental glomerulosclerosis in children using tacrolimus.

Authors:  Rajendra Bhimma; Miriam Adhikari; Kareshma Asharam; Catherine Connolly
Journal:  Am J Nephrol       Date:  2006-12-07       Impact factor: 3.754

Review 7.  Tacrolimus versus cyclosporin as primary immunosuppression for kidney transplant recipients.

Authors:  A Webster; R C Woodroffe; R S Taylor; J R Chapman; J C Craig
Journal:  Cochrane Database Syst Rev       Date:  2005-10-19

8.  Tacrolimus therapy in pediatric patients with treatment-resistant nephrotic syndrome.

Authors:  Kim Loeffler; Manjula Gowrishankar; Verna Yiu
Journal:  Pediatr Nephrol       Date:  2004-02-03       Impact factor: 3.714

Review 9.  Corticosteroid therapy for nephrotic syndrome in children.

Authors:  E M Hodson; N S Willis; J C Craig
Journal:  Cochrane Database Syst Rev       Date:  2007-10-17

10.  Second-line immunosuppressive treatment of childhood nephrotic syndrome: a single-center experience.

Authors:  J Kim; N Patnaik; N Chorny; R Frank; L Infante; C Sethna
Journal:  Nephron Extra       Date:  2014-01-04
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  9 in total

1.  CYP3A5 and CYP3A7 genetic polymorphisms affect tacrolimus concentration in pediatric patients with nephrotic range proteinuria.

Authors:  Hongxia Liu; Qinxia Xu; Wenyan Huang; Qi Zhao; Zhihu Jiang; Xinyu Kuang; Zhiling Li; Huajun Sun; Xiaoyan Qiu
Journal:  Eur J Clin Pharmacol       Date:  2019-08-10       Impact factor: 2.953

Review 2.  Calcineurin inhibitors and nephrotoxicity in children.

Authors:  Fei Liu; Jian-Hua Mao
Journal:  World J Pediatr       Date:  2018-03-12       Impact factor: 2.764

Review 3.  Off-label use of tacrolimus in children with glomerular disease: Effectiveness, safety and pharmacokinetics.

Authors:  Guo-Xiang Hao; Lin-Lin Song; Dong-Feng Zhang; Le-Qun Su; Evelyne Jacqz-Aigrain; Wei Zhao
Journal:  Br J Clin Pharmacol       Date:  2020-01-14       Impact factor: 4.335

4.  Efficacy of Rituximab vs Tacrolimus in Pediatric Corticosteroid-Dependent Nephrotic Syndrome: A Randomized Clinical Trial.

Authors:  Biswanath Basu; Anja Sander; Birendranath Roy; Stella Preussler; Shilpita Barua; T K S Mahapatra; Franz Schaefer
Journal:  JAMA Pediatr       Date:  2018-08-01       Impact factor: 16.193

5.  Associations Between Cessation of Second-Line Therapies and Relapse Rates of Childhood Refractory Minimal-Change Nephrotic Syndrome: A Single-Center, Retrospective Chart Review.

Authors:  Jing Jin; Yufeng Li; Yaju Zhu; Jiajia Ni
Journal:  Curr Ther Res Clin Exp       Date:  2022-04-12

Review 6.  Second and Third Generational Advances in Therapies of the Immune-Mediated Kidney Diseases in Children and Adolescents.

Authors:  Ryszard Grenda; Łukasz Obrycki
Journal:  Children (Basel)       Date:  2022-04-11

7.  Risk factors and clinical characteristics of tacrolimus-induced acute nephrotoxicity in children with nephrotic syndrome: a retrospective case-control study.

Authors:  Ping Gao; Xin-Lei Guan; Rui Huang; Xiao-Fang Shang-Guan; Jiang-Wei Luan; Mao-Chang Liu; Hua Xu; Xiao-Wen Wang
Journal:  Eur J Clin Pharmacol       Date:  2019-11-19       Impact factor: 2.953

8.  Diltiazem on tacrolimus exposure and dose sparing in Chinese pediatric primary nephrotic syndrome: impact of CYP3A4, CYP3A5, ABCB1, and SLCO1B3 polymorphisms.

Authors:  Junyan Wang; Lingfei Huang; Peng Gao; Yan Hu; Yinghua Ni; Zhengyi Zhu; Liwen Zhang; Jufei Yang; Huifen Zhang; Luo Fang
Journal:  Eur J Clin Pharmacol       Date:  2020-08-15       Impact factor: 2.953

9.  Population pharmacokinetics of tacrolimus in children with nephrotic syndrome.

Authors:  Guo-Xiang Hao; Xin Huang; Dong-Feng Zhang; Yi Zheng; Hai-Yan Shi; Yan Li; Evelyne Jacqz-Aigrain; Wei Zhao
Journal:  Br J Clin Pharmacol       Date:  2018-05-22       Impact factor: 4.335

  9 in total

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