Literature DB >> 26635918

Phase 1 Dose-Escalation Study with LEC/chTNT-3 and Toceranib Phosphate (Palladia®) in Dogs with Spontaneous Malignancies.

Julie K Jang1, John Chretin2, David Bruyette2, Peisheng Hu1, Alan L Epstein1.   

Abstract

OBJECTIVES: LEC chemokine promotes TH1 responses and recruits immune cells to inflammatory sites. By linking LEC to an antibody targeting tumor necrosis, LEC/chTNT-3 can be used for the immunotherapeutic treatment of tumors. The primary objective of this study was to determine the safety profile of LEC/chTNT-3 and toceranib phosphate (Palladia®) combination therapy in dogs with spontaneous malignancies. Secondary purpose was to determine objective responses to treatment.
METHODS: Twenty-three dogs with cancer were enrolled, covering nine different malignancies. In this dose escalation study, dogs received LEC/chTNT-3 for five days, and toceranib every 48 hours for the remainder of the study. Dogs received physical exams, chemistry panel, urinalysis, and complete blood counts on days 0, 10, 28 of the study, and every 6-8 weeks thereafter.
RESULTS: Lethargy was noted in 13% dogs. There were no statistical differences in the prevalence of anorexia, diarrhea, thrombocytopenia, renal toxicity, or hepatic toxicity before or during the study. There were trends in increases in the prevalence of vomiting, lymphopenia, and neutropenia (all grade 2 or lower, p=0.07) over the initial 28 days of the study. By day 28, 10% of dogs had partial responses, 58% had stable disease, and 32% had progressive disease.
CONCLUSIONS: LEC/chTNT-3 and toceranib were well tolerated. This combination therapy showed some biological activity against a variety of cancers at a low dose and short duration of LEC/chTNT-3 administration.

Entities:  

Keywords:  Canine; Chemokine; Immunocytokine; Immunotherapy; LEC; Safety; TNT antibody; Toceranib

Year:  2015        PMID: 26635918      PMCID: PMC4666026          DOI: 10.4172/1948-5956.1000343

Source DB:  PubMed          Journal:  J Cancer Sci Ther


  38 in total

1.  H60/TNT-3 fusion protein activates NK cells in vitro and improves immunotherapeutic outcome in murine syngeneic tumor models.

Authors:  Meg L Flanagan; Leslie A Khawli; Peisheng Hu; Alan L Epstein
Journal:  J Immunother       Date:  2006 May-Jun       Impact factor: 4.456

2.  Comparison of recombinant derivatives of chimeric TNT-3 antibody for the radioimaging of solid tumors.

Authors:  Leslie A Khawli; Barbara Biela; Peisheng Hu; Alan L Epstein
Journal:  Hybrid Hybridomics       Date:  2003-02

3.  The novel role of tyrosine kinase inhibitor in the reversal of immune suppression and modulation of tumor microenvironment for immune-based cancer therapies.

Authors:  Junko Ozao-Choy; Ge Ma; Johnny Kao; George X Wang; Marcia Meseck; Max Sung; Myron Schwartz; Celia M Divino; Ping-Ying Pan; Shu-Hsia Chen
Journal:  Cancer Res       Date:  2009-03-10       Impact factor: 12.701

4.  Phase I dose-escalating study of SU11654, a small molecule receptor tyrosine kinase inhibitor, in dogs with spontaneous malignancies.

Authors:  Cheryl A London; Alison L Hannah; Regina Zadovoskaya; May B Chien; Cynthia Kollias-Baker; Mona Rosenberg; Sue Downing; Gerald Post; Joseph Boucher; Narmada Shenoy; Dirk B Mendel; Gerald McMahon; Julie M Cherrington
Journal:  Clin Cancer Res       Date:  2003-07       Impact factor: 12.531

5.  131I-chTNT radioimmunotherapy of 43 patients with advanced lung cancer.

Authors:  Like Yu; Dian Wen Ju; Wenping Chen; Tian Li; Zhaoqiang Xu; Changying Jiang; Shaoliang Chen; Qun Tao; Dan Ye; Peisheng Hu; Leslie A Khawli; Clive R Taylor; Alan L Epstein
Journal:  Cancer Biother Radiopharm       Date:  2006-02       Impact factor: 3.099

6.  Chimeric TNT-3/human beta-glucuronidase fusion proteins for antibody-directed enzyme prodrug therapy (ADEPT).

Authors:  Barbara H Biela; Leslie A Khawli; Peisheng Hu; Alan L Epstein
Journal:  Cancer Biother Radiopharm       Date:  2003-06       Impact factor: 3.099

7.  Cytoreductive chemotherapy improves the biodistribution of antibodies directed against tumor necrosis in murine solid tumor models.

Authors:  Julie K Jang; Leslie A Khawli; Ryan Park; Brian W Wu; Zibo Li; David Canter; Peter S Conti; Alan L Epstein
Journal:  Mol Cancer Ther       Date:  2013-10-15       Impact factor: 6.261

8.  Intralesional injection of adenovirus encoding CC chemokine ligand 16 inhibits mammary tumor growth and prevents metastatic-induced death after surgical removal of the treated primary tumor.

Authors:  Cristiana Guiducci; Emma Di Carlo; Mariella Parenza; Mary Hitt; Mirella Giovarelli; Piero Musiani; Mario P Colombo
Journal:  J Immunol       Date:  2004-04-01       Impact factor: 5.422

9.  Pretreatment with a monoclonal antibody/interleukin-2 fusion protein directed against DNA enhances the delivery of therapeutic molecules to solid tumors.

Authors:  J L Hornick; L A Khawli; P Hu; J Sharifi; C Khanna; A L Epstein
Journal:  Clin Cancer Res       Date:  1999-01       Impact factor: 12.531

10.  Identification of myeloid derived suppressor cells in the peripheral blood of tumor bearing dogs.

Authors:  Matthew Sherger; William Kisseberth; Cheryl London; Susan Olivo-Marston; Tracey L Papenfuss
Journal:  BMC Vet Res       Date:  2012-10-31       Impact factor: 2.741

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  1 in total

1.  Updated developments on molecular imaging and therapeutic strategies directed against necrosis.

Authors:  Dongjian Zhang; Meng Gao; Qiaomei Jin; Yicheng Ni; Jian Zhang
Journal:  Acta Pharm Sin B       Date:  2019-02-13       Impact factor: 11.413

  1 in total

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