Literature DB >> 26553698

Efficacy of ex vivo autologous and in vivo platelet transfusion in the reversal of P2Y12 inhibition by clopidogrel, prasugrel, and ticagrelor: the APTITUDE study.

Stephen A O'Connor1, Julien Amour1, Anne Mercadier1, Réjane Martin1, Mathieu Kerneis1, Jérémie Abtan1, Delphine Brugier1, Johanne Silvain1, Olivier Barthélémy1, Pascal Leprince1, Gilles Montalescot2, Jean-Philippe Collet1.   

Abstract

BACKGROUND: Allogenic platelet transfusions (PT) are administered to treat excessive bleeding in patients on P2Y12 receptor inhibitors (RI). We assessed the effect of ex vivo and in vivo PT on platelet activation and aggregation in patients on dual antiplatelet therapy. METHODS AND
RESULTS: In the Antagonize P2Y12 Treatment Inhibitors by Transfusion of Platelets in an Urgent or Delayed Timing After Acute Coronary Syndrome or Percutaneous Coronary Intervention Presentation-Acute Coronary Syndrome (APTITUDE-ACS) study, patients presenting with acute coronary syndrome or for elective percutaneous coronary intervention, receiving loading doses of clopidogrel (600 mg, n=13 or 900 mg, n=12), prasugrel 60 mg (n=10), or ticagrelor 180 mg (n=10) were included. PT was performed ex vivo by mixing platelet-rich plasma from blood sampling performed at baseline in increasing proportions with platelet-rich plasma sampled 4 hours after loading dose. The percentage restoration of residual platelet aggregation achieved with 80% proportion PT (residual platelet aggregation 80% PT mix/residual platelet aggregation baseline×100) significantly decreased with increasing potency of P2Y12 RI (83.9±11%, 73±14%, 66.3±15%, 40.9±19% for clopidogrel 600 mg, clopidogrel 900 mg, prasugrel, and ticagrelor, respectively; P for trend <0.0001). In the APTITUDE-Coronary Artery Bypass Graft (APTITUDE-CABG) study, vasodilator-stimulated phosphoprotein-platelet reactivity index, a specific marker of the P2Y12 RI drug-effect, was assessed before and after in vivo PT administered for excessive bleeding in patients undergoing cardiac surgery while on a maintenance dose of aspirin and clopidogrel (n=45), prasugrel (n=6), or ticagrelor (n=3). When compared with baseline, there was a significant relative increase of 23.1% in platelet activation after PT transfusion (42.2±23.6% versus 56.6±18.2%; P=0.0008).
CONCLUSIONS: PT restores platelet reactivity in patients with acute coronary syndrome/percutaneous coronary intervention and in patients undergoing cardiac surgery on P2Y12 RI while bleeding with a less effect with increasing potency of P2Y12 inhibition. CLINICAL TRIAL REGISTRATION: URL: http://www.recherche-biomedicale.sante.gouv.fr/pro/comites/coordonnees.htm and http://www.cnil.fr/. Unique identifiers: No. 301111 and No. 1547216v0.
© 2015 American Heart Association, Inc.

Entities:  

Keywords:  hemorrhage; percutaneous coronary intervention; platelet activation; platelet function tests; platelet transfusion

Mesh:

Substances:

Year:  2015        PMID: 26553698     DOI: 10.1161/CIRCINTERVENTIONS.115.002786

Source DB:  PubMed          Journal:  Circ Cardiovasc Interv        ISSN: 1941-7640            Impact factor:   6.546


  9 in total

Review 1.  Non-cardiac surgery in patients with coronary artery disease: risk evaluation and periprocedural management.

Authors:  Davide Cao; Rishi Chandiramani; Davide Capodanno; Jeffrey S Berger; Matthew A Levin; Mary T Hawn; Dominick J Angiolillo; Roxana Mehran
Journal:  Nat Rev Cardiol       Date:  2020-08-05       Impact factor: 32.419

2.  Reversal of the platelet inhibitory effect of the P2Y12 inhibitors clopidogrel, prasugrel, and ticagrelor in vitro: a new approach to an old issue.

Authors:  Lisa Schoener; Stefanie Jellinghaus; Bernhardt Richter; Christian Pfluecke; Georg Ende; Marian Christoph; Silvio Quick; Tobias Loehn; Uwe Speiser; David M Poitz; Johannes Mierke; Ruth H Strasser; Karim Ibrahim
Journal:  Clin Res Cardiol       Date:  2017-06-26       Impact factor: 5.460

3.  The European guideline on management of major bleeding and coagulopathy following trauma: fifth edition.

Authors:  Donat R Spahn; Bertil Bouillon; Vladimir Cerny; Jacques Duranteau; Daniela Filipescu; Beverley J Hunt; Radko Komadina; Marc Maegele; Giuseppe Nardi; Louis Riddez; Charles-Marc Samama; Jean-Louis Vincent; Rolf Rossaint
Journal:  Crit Care       Date:  2019-03-27       Impact factor: 9.097

4.  Impact of Timing on the Functional Recovery Achieved With Platelet Supplementation After Treatment With Ticagrelor.

Authors:  M Urooj Zafar; Donald A Smith; Usman Baber; Samantha Sartori; Kevin Chen; David W Lam; Carlos A Linares-Koloffon; Juan Rey-Mendoza; Gustavo Jimenez Britez; Gines Escolar; Valentin Fuster; Juan J Badimon
Journal:  Circ Cardiovasc Interv       Date:  2017-08       Impact factor: 6.546

Review 5.  Organ transplantation and drug eluting stents: Perioperative challenges.

Authors:  Aparna Dalal
Journal:  World J Transplant       Date:  2016-12-24

6.  Bleeding risk of ticagrelor compared to clopidogrel in intensive care unit patients with acute coronary syndrome: A propensity-score matching analysis.

Authors:  Thibault Charpentier; Cyril Ferdynus; Thomas Lair; Charlotte Cordier; Caroline Brulliard; Dorothée Valance; Malo Emery; Margot Caron; Nicolas Allou; Jérôme Allyn
Journal:  PLoS One       Date:  2020-05-04       Impact factor: 3.240

Review 7.  Platelet transfusion for patients with platelet dysfunction: effectiveness, mechanisms, and unanswered questions.

Authors:  Robert H Lee; Raj S Kasthuri; Wolfgang Bergmeier
Journal:  Curr Opin Hematol       Date:  2020-11       Impact factor: 3.218

8.  Adrenaline enhances in vitro platelet activation and aggregation in blood samples from ticagrelor-treated patients.

Authors:  Sukhi Singh; Carl Johan Malm; Sofia Ramström; Camilla Hesse; Anders Jeppsson
Journal:  Res Pract Thromb Haemost       Date:  2018-09-30

9.  Reversal of Antithrombotic Therapy: Is it Necessary and Sufficient?

Authors:  Richard C Becker
Journal:  JACC Basic Transl Sci       Date:  2017-04-24
  9 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.