Literature DB >> 26389758

Trastuzumab Emtansine (T-DM1) in Patients With HER2-Positive Metastatic Breast Cancer Previously Treated With Chemotherapy and 2 or More HER2-Targeted Agents: Results From the T-PAS Expanded Access Study.

Denise A Yardley1, Ian E Krop, Patricia M LoRusso, Musa Mayer, Brian Barnett, Bongin Yoo, Edith A Perez.   

Abstract

PURPOSE: The antibody-drug conjugate trastuzumab emtansine (T-DM1) has improved outcomes in patients with human epidermal growth factor receptor 2 (HER2)-positive metastatic breast cancer (MBC), as demonstrated in phase III studies. Few data approximating its use in routine clinical practice are available.
METHODS: The T-DM1 Patient Access Study was an expanded-access, multicenter study of T-DM1 in US patients with pretreated HER2-positive locally advanced breast cancer or MBC. The primary endpoint was safety. The secondary endpoint was investigator-assessed objective response rate among patients with measurable disease at baseline. Data are presented for the first 215 enrolled patients.
RESULTS: The median number of prior systemic MBC agents was 8 (range, 3-23). At baseline, median left ventricular ejection fraction was 60%, and 52.6% of patients had nonclinically significant cardiovascular disease. Median T-DM1 treatment duration was 5.0 months (range, 0-29 months; median follow-up, 5.9 months), with 18.6% having received more than 18 cycles. The most common any-grade adverse events were fatigue (50.7%) and nausea (38.1%). Adverse events of grade 3 or greater were reported in 46.5%, most commonly thrombocytopenia and platelet count decrease (10.2%). Bleeding of grade 3 or greater was reported in 4 patients (1.9%). Cardiac dysfunction (primarily asymptomatic left ventricular ejection fraction decreases) was reported in 14 patients (6.5%). Among those with measurable disease at baseline (n = 172), objective response rate was 25.6% (95% confidence interval, 19.2%-32.8%). DISCUSSION: The safety profile of T-DM1 in this real-world setting of heterogeneous, HER2-positive, pretreated, locally advanced breast cancer or MBC was comparable with that reported in phases II and III studies of similar patient populations. T-DM1 was efficacious with no new safety signals.

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Year:  2015        PMID: 26389758     DOI: 10.1097/PPO.0000000000000144

Source DB:  PubMed          Journal:  Cancer J        ISSN: 1528-9117            Impact factor:   3.360


  13 in total

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6.  A retrospective multicentric observational study of trastuzumab emtansine in HER2 positive metastatic breast cancer: a real-world experience.

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Review 7.  Targeted therapeutic options and future perspectives for HER2-positive breast cancer.

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8.  Tissue cross-reactivity studies of CPGJ701 in humans, cynomolgus monkeys and Sprague-Dawley rats and correlation analysis with in vivo toxicity.

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Journal:  Ann Transl Med       Date:  2020-03

9.  Assessment of racial differences in the incidence of thrombocytopenia induced by trastuzumab emtansine: a systematic review and meta-analysis.

Authors:  Jingyi Zhang; Yaning Yang; Ru Chen; Shanshan Chen; Jiayu Wang; Yang Luo; Fei Ma; Binghe Xu; Ying Fan
Journal:  Ann Transl Med       Date:  2021-07

10.  Practical consensus recommendations regarding the management of HER2 neu positive metastatic breast cancer.

Authors:  M Basade; M Singhal; A K Rathi; M Nandi; S Minhas; C Goswami; S Shinde; P M Parikh; S Aggarwal
Journal:  South Asian J Cancer       Date:  2018 Apr-Jun
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