Literature DB >> 26341927

Anti oxidant potential of Metformin and Pioglitazone in Type 2 Diabetes Mellitus: Beyond their anti glycemic effect.

R K Singh1, B Gupta2, K Tripathi1, S K Singh3.   

Abstract

OBJECTIVE: Insulin sensitizers might influence oxidative stress to improve insulin resistance in diabetes mellitus. The present study was designed with the aim to study the effect of Metformin & Pioglitazone on markers of oxidative stress after 4 weeks of therapy in patients with type 2 diabetes mellitus (Type 2 DM). RESEARCH DESIGN AND METHODS: This was a prospective study with follow up of 4 weeks in patients with Type 2 DM. They were randomized into metformin treated group (N=20) and Pioglitazone treated group (N=20) and healthy age-matched control group (N=20). Data was presented as mean±S.D. Student "t" test, ANOVA and Pearson correlation co-efficient tests were performed to analyze the parametric data in this study.
RESULTS: Baseline clinical characteristics of the two study groups were similar. There is a significant difference for Fasting plasma glucose (FPG) and 2h-Post Prandial Plasma Glucose (PPPG) after 30 days of metformin and pioglitazone treatment. Metformin significantly reduced MDA (p=0.041) and increased SOD (p<0.001). Pioglitazone significantly reduced MDA (p<0.001) but failed to raise SOD level (p=0.132). Mean MDA was 4.57±0.57μM/L in metformin and 2.91±0.66μM/L in pioglitazone treatment with a p-value of <0.001. Further, a similar significant difference was obtained for SOD value by metformin and pioglitazone treatment (7.87±0.72U/ml vs. 6.94±0.53U/ml; p<0.001).
CONCLUSION: Pioglitazone was superior to Metformin to improve oxidative stress as reflected by reduction in MDA but the antioxidant effect i.e. increase in SOD was seen with metformin only. The differing mechanism of actions of the two drugs on oxidative stress favors co prescription of these drugs for better outcome in improving insulin resistance and diabetic complications.
Copyright © 2015 Diabetes India. Published by Elsevier Ltd. All rights reserved.

Entities:  

Keywords:  Malondialdehyde (MDA); Metformin; Pioglitazone; Superoxide Dismutase (SOD); Type 2 Diabetes

Mesh:

Substances:

Year:  2015        PMID: 26341927     DOI: 10.1016/j.dsx.2015.08.016

Source DB:  PubMed          Journal:  Diabetes Metab Syndr        ISSN: 1871-4021


  6 in total

1.  Treatment with Parkinsonia aculeata combats insulin resistance-induced oxidative stress through the increase in PPARγ/CuZn-SOD axis expression in diet-induced obesity mice.

Authors:  Tiago Gomes Araújo; Alexandre Gabarra Oliveira; Juliana Falcato Vecina; Rodrigo Miguel Marin; Eryvelton Souza Franco; Mario J Abdalla Saad; Maria Bernadete de Sousa Maia
Journal:  Mol Cell Biochem       Date:  2016-07-02       Impact factor: 3.396

2.  Effects of Pioglitazone On the Lipid Profile, Serum Antioxidant Capacity, and UCP1 Gene Expression in Mouse Brown Adipose Tissue.

Authors:  Amin Mahmoudi; Keihan Ghatreh Samani; Seyed Asadollah Amini; Esfandiar Heidarian
Journal:  Rep Biochem Mol Biol       Date:  2019-04

3.  Metformin attenuates myocardial ischemia-reperfusion injury via up-regulation of antioxidant enzymes.

Authors:  Xiaoling Wang; Lei Yang; Licheng Kang; Jing Li; Liang Yang; Jincai Zhang; Jie Liu; Mengmeng Zhu; Qiong Zhang; Yanna Shen; Zhi Qi
Journal:  PLoS One       Date:  2017-08-17       Impact factor: 3.240

Review 4.  The Current and Potential Therapeutic Use of Metformin-The Good Old Drug.

Authors:  Józef Drzewoski; Markolf Hanefeld
Journal:  Pharmaceuticals (Basel)       Date:  2021-02-05

5.  A metabolome-wide characterization of the diabetic phenotype in ZDF rats and its reversal by pioglitazone.

Authors:  Thomas J Jönsson; Hans-Ludwig Schäfer; Andreas W Herling; Mark Brönstrup
Journal:  PLoS One       Date:  2018-11-27       Impact factor: 3.240

Review 6.  Heterogeneity of Metabolic Defects in Type 2 Diabetes and Its Relation to Reactive Oxygen Species and Alterations in Beta-Cell Mass.

Authors:  Andris Elksnis; Mats Martinell; Olof Eriksson; Daniel Espes
Journal:  Front Physiol       Date:  2019-02-13       Impact factor: 4.566

  6 in total

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