Literature DB >> 26336809

Effects of Recombinant Human Leptin (Metreleptin) on Nocturnal Luteinizing Hormone Secretion in Lipodystrophy Patients.

Brent S Abel1, Ranganath Muniyappa, Pamela Stratton, Monica C Skarulis, Phillip Gorden, Rebecca J Brown.   

Abstract

BACKGROUND: Leptin replacement in patients with leptin gene mutations improves hypogonadotropic hypogonadism. The effects of leptin replacement on luteinizing hormone (LH) secretion in patients with lipodystrophy are unknown. AIM: We examined nocturnal LH secretory dynamics on and off exogenous leptin therapy using a 2-period, nonrandomized study that included leptin-naïve and leptin-treated subjects with lipodystrophy.
METHODS: In period 1 (5 days) the leptin-treated group (n = 4) continued leptin; leptin was then withdrawn for the next 14 days (period 2). Leptin-naïve subjects (n = 8) were studied without leptin in period 1 and with leptin replacement in period 2. LH secretory dynamics were assessed (23:00-07:00 h, sampling every 10 min, analyzed by multiparameter deconvolution algorithm) at the end of each period.
RESULTS: Mean (on vs. off: 5.0 ± 3.1 vs. 3.2 ± 1.3 IU/l, p = 0.04) and integrated LH concentrations (2,403 ± 1,495 vs. 1,534 ± 642 IU × l-1 × min-1, p = 0.04) were higher on leptin therapy. Leptin treatment increased burst mass (9.7± 15.4 vs. 7.0 ± 11.2 IU/l, p = 0.03) and tended to nonsignificantly increase LH burst frequency (0.77 ± 0.26 vs. 0.67 ± 0.24 h-1, p = 0.08). Consequently, leptin therapy increased the pulsatile production rate (64 ± 101 vs. 57 ± 73 IU × l-1 × 8 h-1, p = 0.01). On leptin, testosterone (507 ± 286 vs. 360 ± 174 ng/dl, p = 0.09) and estradiol levels (74 ± 36 vs. 29 ± 24 pg/ml, p = 0.01) were higher in males and females, respectively.
CONCLUSIONS: Leptin increases spontaneous nocturnal LH secretion in patients with lipodystrophy. This is consistent with rodent and in vitro studies showing a direct stimulatory effect (hypothalamic, pituitary or both) of leptin on LH secretion. These novel findings may explicate some of the salutary effects of leptin therapy on the hypothalamic-pituitary-gonadal axis in lipodystrophy.
© 2015 S. Karger AG, Basel.

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Year:  2015        PMID: 26336809      PMCID: PMC7269156          DOI: 10.1159/000439432

Source DB:  PubMed          Journal:  Neuroendocrinology        ISSN: 0028-3835            Impact factor:   4.914


  24 in total

1.  Effects of recombinant leptin therapy in a child with congenital leptin deficiency.

Authors:  I S Farooqi; S A Jebb; G Langmack; E Lawrence; C H Cheetham; A M Prentice; I A Hughes; M A McCamish; S O'Rahilly
Journal:  N Engl J Med       Date:  1999-09-16       Impact factor: 91.245

2.  Congenital leptin deficiency is associated with severe early-onset obesity in humans.

Authors:  C T Montague; I S Farooqi; J P Whitehead; M A Soos; H Rau; N J Wareham; C P Sewter; J E Digby; S N Mohammed; J A Hurst; C H Cheetham; A R Earley; A H Barnett; J B Prins; S O'Rahilly
Journal:  Nature       Date:  1997-06-26       Impact factor: 49.962

3.  Characterization of the physiological pattern of episodic gonadotropin secretion throughout the human menstrual cycle.

Authors:  M Filicori; N Santoro; G R Merriam; W F Crowley
Journal:  J Clin Endocrinol Metab       Date:  1986-06       Impact factor: 5.958

4.  Leptin substitution results in the induction of menstrual cycles in an adolescent with leptin deficiency and hypogonadotropic hypogonadism.

Authors:  J von Schnurbein; A Moss; S A Nagel; H Muehleder; K M Debatin; I S Farooqi; M Wabitsch
Journal:  Horm Res Paediatr       Date:  2012-02-14       Impact factor: 2.852

5.  Phenotypic effects of leptin replacement on morbid obesity, diabetes mellitus, hypogonadism, and behavior in leptin-deficient adults.

Authors:  Julio Licinio; Sinan Caglayan; Metin Ozata; Bulent O Yildiz; Patricia B de Miranda; Fiona O'Kirwan; Robert Whitby; Liyin Liang; Pinchas Cohen; Shalender Bhasin; Ronald M Krauss; Johannes D Veldhuis; Anthony J Wagner; Alex M DePaoli; Samuel M McCann; Ma-Li Wong
Journal:  Proc Natl Acad Sci U S A       Date:  2004-03-09       Impact factor: 11.205

6.  Effect of leptin replacement on pituitary hormone regulation in patients with severe lipodystrophy.

Authors:  Elif Arioglu Oral; Elaine Ruiz; Alexa Andewelt; Nancy Sebring; Anthony J Wagner; Alex M Depaoli; Phillip Gorden
Journal:  J Clin Endocrinol Metab       Date:  2002-07       Impact factor: 5.958

7.  The role of falling leptin levels in the neuroendocrine and metabolic adaptation to short-term starvation in healthy men.

Authors:  Jean L Chan; Kathleen Heist; Alex M DePaoli; Johannes D Veldhuis; Christos S Mantzoros
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8.  Positional cloning of the mouse obese gene and its human homologue.

Authors:  Y Zhang; R Proenca; M Maffei; M Barone; L Leopold; J M Friedman
Journal:  Nature       Date:  1994-12-01       Impact factor: 49.962

9.  Leptin levels and luteinizing hormone pulsatility in normal cycling women and their relationship to daily changes in metabolic rate.

Authors:  Rebecca M Fenichel; Jennifer E Dominguez; Laurel Mayer; B Timothy Walsh; Carol Boozer; Michelle P Warren
Journal:  Fertil Steril       Date:  2008-03-04       Impact factor: 7.329

10.  A mutation in the human leptin receptor gene causes obesity and pituitary dysfunction.

Authors:  K Clément; C Vaisse; N Lahlou; S Cabrol; V Pelloux; D Cassuto; M Gourmelen; C Dina; J Chambaz; J M Lacorte; A Basdevant; P Bougnères; Y Lebouc; P Froguel; B Guy-Grand
Journal:  Nature       Date:  1998-03-26       Impact factor: 49.962

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  5 in total

Review 1.  The Head-to-Toe Hormone: Leptin as an Extensive Modulator of Physiologic Systems.

Authors:  Monica Misch; Prasanth Puthanveetil
Journal:  Int J Mol Sci       Date:  2022-05-13       Impact factor: 6.208

2.  Metreleptin-mediated improvements in insulin sensitivity are independent of food intake in humans with lipodystrophy.

Authors:  Rebecca J Brown; Areli Valencia; Megan Startzell; Elaine Cochran; Peter J Walter; H Martin Garraffo; Hongyi Cai; Ahmed M Gharib; Ronald Ouwerkerk; Amber B Courville; Shanna Bernstein; Robert J Brychta; Kong Y Chen; Mary Walter; Sungyoung Auh; Phillip Gorden
Journal:  J Clin Invest       Date:  2018-07-16       Impact factor: 14.808

Review 3.  Update on Therapeutic Options in Lipodystrophy.

Authors:  Baris Akinci; Rasimcan Meral; Elif Arioglu Oral
Journal:  Curr Diab Rep       Date:  2018-10-29       Impact factor: 4.810

Review 4.  The Diagnosis and Management of Lipodystrophy Syndromes: A Multi-Society Practice Guideline.

Authors:  Rebecca J Brown; David Araujo-Vilar; Pik To Cheung; David Dunger; Abhimanyu Garg; Michelle Jack; Lucy Mungai; Elif A Oral; Nivedita Patni; Kristina I Rother; Julia von Schnurbein; Ekaterina Sorkina; Takara Stanley; Corinne Vigouroux; Martin Wabitsch; Rachel Williams; Tohru Yorifuji
Journal:  J Clin Endocrinol Metab       Date:  2016-10-06       Impact factor: 5.958

Review 5.  Polycystic ovary syndrome in familial partial lipodystrophy type 2 (FPLD2): basic and clinical aspects.

Authors:  Alessandra Gambineri; Laura Zanotti
Journal:  Nucleus       Date:  2018       Impact factor: 4.197

  5 in total

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