Literature DB >> 26310103

Diquafosol sodium ophthalmic solution for the treatment of dry eye: clinical evaluation and biochemical analysis of tear composition.

Chika Shigeyasu1,2,3, Masakazu Yamada4, Yoko Akune5, Kazuo Tsubota6.   

Abstract

PURPOSE: To evaluate the clinical efficacy of 3% diquafosol sodium ophthalmic solution for dry eye, and to analyze the concentration of tear proteins and mucin-like substances after the treatment.
METHODS: Fifty eyes of 25 patients with dry eye syndrome were prospectively enrolled. The patients were treated with diquafosol solution at a dose of 1 drop in each eye 6 times daily for 4 weeks. The parameters of clinical efficacy were tear osmolarity, tear breakup time (BUT), fluorescein staining scores for the cornea and conjunctiva, Schirmer test values, and subjective symptoms evaluated using the ocular surface disease index (OSDI). Tears collected with Schirmer test strips were analyzed by high-performance liquid chromatography, and the concentrations of the total protein and the 4 major tear proteins, namely, secretory IgA, lactoferrin, lipocalin-1, lysozyme, and N-acetyl-neuraminic acid (Neu5Ac), were measured. Neu5Ac is a major sialic acid, a marker of secretory mucins.
RESULTS: The BUT, keratoconjunctival staining scores, and Schirmer test values were improved with statistical significance after the treatment with diquafosol solution, while changes in the other parameters, including tear osmolarity, corneal staining scores, and OSDI scores were not significant. The Neu5Ac concentration was significantly increased, which was not accompanied by changes in tear proteins.
CONCLUSIONS: Topical application of diquafosol significantly improved the clinical parameters of the BUT, keratoconjunctival staining scores, and Schirmer test values and was accompanied by increased sialic acid content in the tears of patients with dry eye.

Entities:  

Keywords:  Diquafosol ophthalmic solution; Dry eye syndrome; Mucins; Sialic acid; Tears

Mesh:

Substances:

Year:  2015        PMID: 26310103     DOI: 10.1007/s10384-015-0408-y

Source DB:  PubMed          Journal:  Jpn J Ophthalmol        ISSN: 0021-5155            Impact factor:   2.447


  30 in total

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Review 2.  Management and therapy of dry eye disease: report of the Management and Therapy Subcommittee of the International Dry Eye WorkShop (2007).

Authors: 
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3.  Facilitation of tear fluid secretion by 3% diquafosol ophthalmic solution in normal human eyes.

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4.  Entrapment of conjunctival goblet cells by desiccation-induced cornification.

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5.  Double-masked, placebo-controlled safety and efficacy trial of diquafosol tetrasodium (INS365) ophthalmic solution for the treatment of dry eye.

Authors:  J Tauber; W F Davitt; J E Bokosky; K K Nichols; B R Yerxa; A E Schaberg; L M LaVange; M C Mills-Wilson; D J Kellerman
Journal:  Cornea       Date:  2004-11       Impact factor: 2.651

Review 6.  Diquafosol tetrasodium: a novel dry eye therapy.

Authors:  Kelly K Nichols; Ben Yerxa; Donald J Kellerman
Journal:  Expert Opin Investig Drugs       Date:  2004-01       Impact factor: 6.206

7.  INS365 suppresses loss of corneal epithelial integrity by secretion of mucin-like glycoprotein in a rabbit short-term dry eye model.

Authors:  Tsutomu Fujihara; Tadahiro Murakami; Takashi Nagano; Masatsugu Nakamura; Katsuhiko Nakata
Journal:  J Ocul Pharmacol Ther       Date:  2002-08       Impact factor: 2.671

8.  Alteration of mucin in human conjunctival epithelia in dry eye.

Authors:  Y Danjo; H Watanabe; A S Tisdale; M George; T Tsumura; M B Abelson; I K Gipson
Journal:  Invest Ophthalmol Vis Sci       Date:  1998-12       Impact factor: 4.799

9.  Sodium hyaluronate eyedrops in the treatment of dry eyes.

Authors:  S Shimmura; M Ono; K Shinozaki; I Toda; E Takamura; Y Mashima; K Tsubota
Journal:  Br J Ophthalmol       Date:  1995-11       Impact factor: 4.638

10.  A randomised, double-masked comparison study of diquafosol versus sodium hyaluronate ophthalmic solutions in dry eye patients.

Authors:  Etsuko Takamura; Kazuo Tsubota; Hitoshi Watanabe; Yuichi Ohashi
Journal:  Br J Ophthalmol       Date:  2012-08-21       Impact factor: 4.638

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2.  The correlation between plasma osmolarity and tear osmolarity.

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Journal:  Int Ophthalmol       Date:  2017-03-02       Impact factor: 2.031

3.  Efficacy of Artificial Tears Based on an Extract of Artemia salina Containing Dinucleotides in a Rabbit Dry Eye Model.

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Review 4.  Current approaches for the regeneration and reconstruction of ocular surface in dry eye.

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