Literature DB >> 26293127

GLP-1 receptor agonists in type 1 diabetes: a proof-of-concept approach.

Isabella Crisci1, Michele Aragona1, Konstantina Savvina Politi1, Giuseppe Daniele1, Stefano Del Prato2.   

Abstract

AIMS: To test potential efficacy of liraglutide, a GLP-1 receptor agonist, in subjects with type 1 diabetes (T1DM).
METHODS: We have recruited nine T1DM patients (age 40.1 ± 6.4 years, duration of diabetes 19.2 ± 8.8 years, BMI 24.3 ± 3.5 kg/m(2), HbA1c 8.2 ± 1.0 %-66 ± 11 mmol/mol, daily insulin dose: 0.6 ± 0.1 IU/kg) on continuous subcutaneous insulin therapy with undetectable C-peptide. In addition to existing treatment was administered in single-blind (a) therapy subcutaneously with 0.1 ml of saline solution for 3 days and (b) 0.1 ml of liraglutide (0.6 mg/day) for a further 3 days with daily glucose excursions recorded by continuous glucose monitoring.
RESULTS: Adding liraglutide resulted in a significant reduction in mean blood glucose (138 ± 29 vs. 163 ± 29 mg/dl, p < 0.0001) and standard deviation (42 ± 9 vs. 60 ± 15 mg/dl, p < 0.0001). The area under the curve (AUC) for blood glucose >140 mg/dl was also significantly reduced (22.2 ± 16.4 vs. 41.1 ± 19.7 mg/dl h, p < 0.05) with no difference in AUC for blood glucose <70 mg/dl (liraglutide 0.7 ± 0.9 mg/dl h; placebo: 0.8 ± 1.4 mg/dl h, p = NS). Finally, adding liraglutide reduced daily insulin requirement (37.5 ± 17.2 vs. 42.9 ± 22.4 UI/day, p < 0.01).
CONCLUSIONS: Short-term treatment with liraglutide, in T1DM, reduces average blood glucose, blood glucose variability and daily insulin requirement without increasing risk of hypoglycemia.

Entities:  

Keywords:  Continuous glucose monitoring; Glycemic variability; Insulin pump therapy; Liraglutide; Type 1 diabetes

Mesh:

Substances:

Year:  2015        PMID: 26293127     DOI: 10.1007/s00592-015-0800-6

Source DB:  PubMed          Journal:  Acta Diabetol        ISSN: 0940-5429            Impact factor:   4.280


  2 in total

1.  The GLP-1 receptor agonists exenatide and liraglutide activate Glucose transport by an AMPK-dependent mechanism.

Authors:  Francesco Andreozzi; Gregory Alexander Raciti; Cecilia Nigro; Gaia Chiara Mannino; Teresa Procopio; Alberto M Davalli; Francesco Beguinot; Giorgio Sesti; Claudia Miele; Franco Folli
Journal:  J Transl Med       Date:  2016-07-30       Impact factor: 5.531

Review 2.  Differentiation of Diabetes by Pathophysiology, Natural History, and Prognosis.

Authors:  Jay S Skyler; George L Bakris; Ezio Bonifacio; Tamara Darsow; Robert H Eckel; Leif Groop; Per-Henrik Groop; Yehuda Handelsman; Richard A Insel; Chantal Mathieu; Allison T McElvaine; Jerry P Palmer; Alberto Pugliese; Desmond A Schatz; Jay M Sosenko; John P H Wilding; Robert E Ratner
Journal:  Diabetes       Date:  2016-12-15       Impact factor: 9.461

  2 in total

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