Literature DB >> 26213885

Targeting Adenosine Monophosphate-Activated Protein Kinase by Metformin Adjusts Post-Ischemic Hyperemia and Extracellular Neuronal Discharge in Transient Global Cerebral Ischemia.

Yaghoob Farbood1,2, Alireza Sarkaki1,2, Leila Khalaj3, Fariba Khodagholi4,5, Mohammad Badavi1,2, Ghorbangol Ashabi1,2.   

Abstract

OBJECTIVE: I/R and its subsequent reactive hyperemia results in different adverse effects such as brain edema and BBB disruption. AMPK activation has been perceived as one of the target factors for I/R treatment. We investigated the effect of Met (an AMPK activator) on some physiological parameters including vascular responses, hyperemia, BBB disruption, and electrophysiological activity following tGCI.
METHODS: Rats were pretreated with Met for two weeks and CC was administered half an hour before tGCI. Brain vascular responses, hyperemia, BBB disruption, and electrophysiological activity were evaluated following the ischemia.
RESULTS: Met attenuated BBB disruption and reactive hyperemia in tGCI rats compared with the untreated I/R rats (p < 0.001). Met administration along with CC in the ischemic rats reversed the beneficial effects of Met on BBB disruption and reactive hyperemia (p < 0.001). Electrophysiological records indicated that Met increased spike rates in the ischemic rats comparing with I/R rats (p < 0.001), whereas, CC administration blocked the beneficial effects of Met on the neuronal discharges (p < 0.05).
CONCLUSION: We established a regulatory role for AMPK in vascular and electrophysiological responses to tGCI. Studies are ongoing to determine if activation of AMPK in the reperfusion period would offer similar protection.
© 2015 John Wiley & Sons Ltd.

Entities:  

Keywords:  adenosine monophosphate-activated protein kinase; blood-brain barrier permeability; cerebral blood flow; global cerebral ischemia; metformin; single-unit recording

Mesh:

Substances:

Year:  2015        PMID: 26213885     DOI: 10.1111/micc.12224

Source DB:  PubMed          Journal:  Microcirculation        ISSN: 1073-9688            Impact factor:   2.628


  8 in total

1.  The Antidiabetic Drug Metformin Stimulates Glycolytic Lactate Production in Cultured Primary Rat Astrocytes.

Authors:  Adrian Westhaus; Eva Maria Blumrich; Ralf Dringen
Journal:  Neurochem Res       Date:  2015-10-03       Impact factor: 3.996

2.  Vanillic acid attenuates cerebral hyperemia, blood-brain barrier disruption and anxiety-like behaviors in rats following transient bilateral common carotid occlusion and reperfusion.

Authors:  Seyed Esmaeil Khoshnam; Yaghoob Farbood; Hadi Fathi Moghaddam; Alireza Sarkaki; Mohammad Badavi; Layasadat Khorsandi
Journal:  Metab Brain Dis       Date:  2018-01-22       Impact factor: 3.584

3.  Neuroprotective effects of metformin on traumatic brain injury in rats is associated with the AMP-activated protein kinase signaling pathway.

Authors:  Siavash Rahimi; Ahmadreza Ferdowsi; Ali Siahposht-Khachaki
Journal:  Metab Brain Dis       Date:  2020-07-03       Impact factor: 3.584

Review 4.  Repurposing metformin to treat age-related neurodegenerative disorders and ischemic stroke.

Authors:  Sejal Sharma; Saeideh Nozohouri; Bhuvaneshwar Vaidya; Thomas Abbruscato
Journal:  Life Sci       Date:  2021-03-11       Impact factor: 6.780

Review 5.  To Use or Not to Use Metformin in Cerebral Ischemia: A Review of the Application of Metformin in Stroke Rodents.

Authors:  Isaac Arbeláez-Quintero; Mauricio Palacios
Journal:  Stroke Res Treat       Date:  2017-05-28

Review 6.  The stress polarity pathway: AMPK 'GIV'-es protection against metabolic insults.

Authors:  Pradipta Ghosh
Journal:  Aging (Albany NY)       Date:  2017-02-15       Impact factor: 5.682

7.  The evidence of metabolic-improving effect of metformin in Ay/a mice with genetically-induced melanocortin obesity and the contribution of hypothalamic mechanisms to this effect.

Authors:  Kira Derkach; Irina Zakharova; Inna Zorina; Andrey Bakhtyukov; Irina Romanova; Liubov Bayunova; Alexander Shpakov
Journal:  PLoS One       Date:  2019-03-14       Impact factor: 3.240

Review 8.  Reciprocal Association between the Apical Junctional Complex and AMPK: A Promising Therapeutic Target for Epithelial/Endothelial Barrier Function?

Authors:  Kazuto Tsukita; Tomoki Yano; Atsushi Tamura; Sachiko Tsukita
Journal:  Int J Mol Sci       Date:  2019-11-29       Impact factor: 5.923

  8 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.