Literature DB >> 26148596

Sensitization to oxaliplatin in HCT116 and HT29 cell lines by metformin and ribavirin and differences in response to mitochondrial glutaminase inhibition.

Silvina M Richard, Veronica L Martinez Marignac1.   

Abstract

AIM OF STUDY: In the present study, we evaluated the effect of ribavirin and metformin on the sensitivity of oxaliplatin and 5-fluorouracil (5-FU) on colon cancer.
MATERIALS AND METHODS: Cell viability of two commercially available colon cancer cell lines (HT29 and HCT116) were analyzed by sulforhodamine B (SRB) assay.
RESULTS: A clinically achievable and nontoxic concentration of ribavirin and metformin showed a significant synergistic effect on oxaliplatin in HT29 and HCT116 cell lines. Ribavirin showed a synergistic effect on oxaliplatin in HT29 (R = 2.93, P < 0.001) and HCT116 (R = 1.71, P < 0.001), while only in HT29 metformin synergized with oxaliplatin by 2.66 (± 0.28, P < 0.01). In addition, both cell lines showed significant differences in response to Compound 968, inhibitor of mitochondrial glutaminase activity.
CONCLUSION: The data suggested that these cell lines not only turn to metabolic different sustainability process after oxaliplatin treatment but that they also have different basal metabolic requirements of glutamine in vitro which can be exploits in the future for colorectal cancer (CRC) treatment and further studies are required.

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Year:  2015        PMID: 26148596     DOI: 10.4103/0973-1482.157317

Source DB:  PubMed          Journal:  J Cancer Res Ther        ISSN: 1998-4138            Impact factor:   1.805


  15 in total

1.  AGR2 silencing contributes to metformin-dependent sensitization of colorectal cancer cells to chemotherapy.

Authors:  Andrea Martisova; Lucia Sommerova; Katarina Kuricova; Jan Podhorec; Borivoj Vojtesek; Katerina Kankova; Roman Hrstka
Journal:  Oncol Lett       Date:  2019-09-04       Impact factor: 2.967

2.  Glutaminase sustains cell survival via the regulation of glycolysis and glutaminolysis in colorectal cancer.

Authors:  Zhou Song; Bo Wei; Canrong Lu; Peiyu Li; Lin Chen
Journal:  Oncol Lett       Date:  2017-07-07       Impact factor: 2.967

3.  Use of an anti-viral drug, Ribavirin, as an anti-glioblastoma therapeutic.

Authors:  F Volpin; J Casaos; J Sesen; A Mangraviti; J Choi; N Gorelick; J Frikeche; T Lott; R Felder; S J Scotland; T S K Eisinger-Mathason; H Brem; B Tyler; N Skuli
Journal:  Oncogene       Date:  2016-12-12       Impact factor: 9.867

4.  Impact of Metformin Use and Diabetic Status During Adjuvant Fluoropyrimidine-Oxaliplatin Chemotherapy on the Outcome of Patients with Resected Colon Cancer: A TOSCA Study Subanalysis.

Authors:  Claudio Vernieri; Fabio Galli; Laura Ferrari; Paolo Marchetti; Sara Lonardi; Evaristo Maiello; Rosario V Iaffaioli; Maria G Zampino; Alberto Zaniboni; Sabino De Placido; Maria Banzi; Azzurra Damiani; Daris Ferrari; Gerardo Rosati; Roberto F Labianca; Paolo Bidoli; Giovanni L Frassineti; Mario Nicolini; Lorenzo Pavesi; Maria C Tronconi; Angela Buonadonna; Sabrina Ferrario; Giovanni Lo Re; Vincenzo Adamo; Emiliano Tamburini; Mario Clerico; Paolo Giordani; Francesco Leonardi; Sandro Barni; Andrea Ciarlo; Luigi Cavanna; Stefania Gori; Saverio Cinieri; Marina Faedi; Massimo Aglietta; Maria Antista; Katia F Dotti; Francesca Galli; Maria Di Bartolomeo
Journal:  Oncologist       Date:  2019-01-03

5.  Cytotoxic effects of the newly-developed chemotherapeutic agents 17-AAG in combination with oxaliplatin and capecitabine in colorectal cancer cell lines.

Authors:  Mahshid Mohammadian; Shima Zeynali; Anahita Fathi Azarbaijani; Mohammad Hassan Khadem Ansari; Fatemeh Kheradmand
Journal:  Res Pharm Sci       Date:  2017-12

6.  Cytotoxic Compounds from Wrightia pubescens (R.Br.).

Authors:  Mariquit M De Los Reyes; Glenn G Oyong; Vincent Antonio S Ng; Chien-Chang Shen; Consolacion Y Ragasa
Journal:  Pharmacognosy Res       Date:  2018 Jan-Mar

Review 7.  Strategy to targeting the immune resistance and novel therapy in colorectal cancer.

Authors:  Wang Gang; Jun-Jie Wang; Rui Guan; Sun Yan; Feng Shi; Jia-Yan Zhang; Zi-Meng Li; Jing Gao; Xing-Li Fu
Journal:  Cancer Med       Date:  2018-04-15       Impact factor: 4.452

8.  Metformin suppressed the proliferation of LoVo cells and induced a time-dependent metabolic and transcriptional alteration.

Authors:  Jiaojiao He; Ke Wang; Ningning Zheng; Yunping Qiu; Guoxiang Xie; Mingming Su; Wei Jia; Houkai Li
Journal:  Sci Rep       Date:  2015-11-30       Impact factor: 4.379

9.  Ribavirin as a potential therapeutic for atypical teratoid/rhabdoid tumors.

Authors:  Betty Tyler; Nicolas Skuli; Joshua Casaos; Sakibul Huq; Tarik Lott; Raphael Felder; John Choi; Noah Gorelick; Michael Peters; Yuanxuan Xia; Russell Maxwell; Tianna Zhao; Chenchen Ji; Thomas Simon; Julie Sesen; Sarah J Scotland; Richard E Kast; Jeffrey Rubens; Eric Raabe; Charles G Eberhart; Eric M Jackson; Henry Brem
Journal:  Oncotarget       Date:  2018-01-03

10.  Combined blockade of EGFR and glutamine metabolism in preclinical models of colorectal cancer.

Authors:  Allison S Cohen; Ling Geng; Ping Zhao; Allie Fu; Michael L Schulte; Ramona Graves-Deal; M Kay Washington; Jordan Berlin; Robert J Coffey; H Charles Manning
Journal:  Transl Oncol       Date:  2020-07-08       Impact factor: 4.243

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