Literature DB >> 26063741

Safety of oral dofetilide for rhythm control of atrial fibrillation and atrial flutter.

JoEllyn M Abraham1, Walid I Saliba2, Carolyn Vekstein2, David Lawrence2, Mandeep Bhargava2, Mohamed Bassiouny2, David Janiszewski2, Bruce Lindsay2, Michael Militello2, Steven E Nissen2, Stacy Poe2, Christine Tanaka-Esposito2, Kathy Wolski2, Bruce L Wilkoff2.   

Abstract

BACKGROUND: Although dofetilide is widely used in the United States for rhythm control of atrial fibrillation, there is limited postapproval safety data in the atrial fibrillation population despite its known risk of Torsade de pointes (TdP). METHODS AND
RESULTS: We conducted a retrospective chart review of a cohort of 1404 patients initially loaded on dofetilide for atrial fibrillation suppression at the Cleveland Clinic from 2008 to 2012 to evaluate the incidence and risk factors for in-hospital adverse events and the long-term safety of continued use. Of the 17 patients with TdP during loading (1.2%), 10 had a cardiac arrest requiring resuscitation (1 death), 5 had syncope/presyncope, and 2 were asymptomatic. Dofetilide loading was stopped for 105 patients (7.5%) because of QTc prolongation or TdP. Variables correlated with TdP were (1) female sex, 2) 500-μg dose, (3) reduced ejection fraction, and (4) increase in QTc from baseline. One-year all-cause mortality was higher in patients who continued dofetilide compared with those who discontinued use (hazard ratio, 2.48; 95% confidence interval, 1.08-5.71; P=0.03). Those patients who had a TdP event had higher one-year all-cause mortality than those who did not (17.6% versus 3% at 1 year; P<0.001).
CONCLUSIONS: Dofetilide loading has a low but finite risk of TdP and other adverse events that warrant the current Food and Drug Administration-mandated practice of inpatient monitoring during drug loading. In this cohort, all-cause mortality was higher at 1 year in those patients continued on dofetilide and in those patients who experienced TdP while loading.
© 2015 American Heart Association, Inc.

Entities:  

Keywords:  Torsade de pointes; anti-arrhythmic drugs; atrial fibrillation; atrial flutter; dofetilide

Mesh:

Substances:

Year:  2015        PMID: 26063741     DOI: 10.1161/CIRCEP.114.002339

Source DB:  PubMed          Journal:  Circ Arrhythm Electrophysiol        ISSN: 1941-3084


  14 in total

1.  Classification of drug-induced hERG potassium-channel block from electrocardiographic T-wave features using artificial neural networks.

Authors:  Micaela Morettini; Chiara Peroni; Agnese Sbrollini; Ilaria Marcantoni; Laura Burattini
Journal:  Ann Noninvasive Electrocardiol       Date:  2019-07-26       Impact factor: 1.468

2.  Safety of Oral Dofetilide Reloading for Treatment of Atrial Arrhythmias.

Authors:  Jae Hyung Cho; So Jin Youn; JoEllyn C Moore; Roxanne Kyriakakis; Carolyn Vekstein; Michael Militello; Stacy M Poe; Kathy Wolski; Patrick J Tchou; Niraj Varma; Mark J Niebauer; Mandeep Bhargava; Walid I Saliba; Oussama M Wazni; Bruce D Lindsay; Bruce L Wilkoff; Mina K Chung
Journal:  Circ Arrhythm Electrophysiol       Date:  2017-10

Review 3.  Pathophysiological and therapeutic implications in patients with atrial fibrillation and heart failure.

Authors:  Felix Hohendanner; F R Heinzel; F Blaschke; B M Pieske; W Haverkamp; H L Boldt; A S Parwani
Journal:  Heart Fail Rev       Date:  2018-01       Impact factor: 4.214

4.  Short- and long-term clinical predictors of pharmacological cardioversion of persistent atrial fibrillation by dofetilide: A retrospective cohort study of 160 patients.

Authors:  Hafeez Ul Hassan Virk; Waqas T Qureshi; Nayani Makkar; Joseph Bastawrose; Nektarios Souvaliotis; Joshua Aziz; Emad Aziz
Journal:  Clin Cardiol       Date:  2017-03-14       Impact factor: 2.882

5.  Inhibition of the α-Subunit of Phosphoinositide 3-Kinase in Heart Increases Late Sodium Current and Is Arrhythmogenic.

Authors:  Tao Yang; David F Meoli; Javid Moslehi; Dan M Roden
Journal:  J Pharmacol Exp Ther       Date:  2018-03-21       Impact factor: 4.030

6.  Validating the Arrhythmogenic Potential of High-, Intermediate-, and Low-Risk Drugs in a Human-Induced Pluripotent Stem Cell-Derived Cardiac Microphysiological System.

Authors:  Verena Charwat; Bérénice Charrez; Brian A Siemons; Henrik Finsberg; Karoline H Jæger; Andrew G Edwards; Nathaniel Huebsch; Samuel Wall; Evan Miller; Aslak Tveito; Kevin E Healy
Journal:  ACS Pharmacol Transl Sci       Date:  2022-07-29

7.  Predicting critical drug concentrations and torsadogenic risk using a multiscale exposure-response simulator.

Authors:  Francisco Sahli Costabal; Jiang Yao; Anna Sher; Ellen Kuhl
Journal:  Prog Biophys Mol Biol       Date:  2018-10-26       Impact factor: 3.667

8.  Potentially modifiable factors of dofetilide-associated risk of torsades de pointes among hospitalized patients with atrial fibrillation.

Authors:  Niyada Naksuk; Alan M Sugrue; Deepak Padmanabhan; Danesh Kella; Christopher V DeSimone; Suraj Kapa; Samuel J Asirvatham; Hon-Chi Lee; Michael J Ackerman; Peter A Noseworthy
Journal:  J Interv Card Electrophysiol       Date:  2018-10-23       Impact factor: 1.900

Review 9.  Predicting drug-induced QT prolongation and torsades de pointes.

Authors:  Dan M Roden
Journal:  J Physiol       Date:  2016-01-18       Impact factor: 5.182

10.  A Computational Pipeline to Predict Cardiotoxicity: From the Atom to the Rhythm.

Authors:  Pei-Chi Yang; Kevin R DeMarco; Parya Aghasafari; Mao-Tsuen Jeng; John R D Dawson; Slava Bekker; Sergei Y Noskov; Vladimir Yarov-Yarovoy; Igor Vorobyov; Colleen E Clancy
Journal:  Circ Res       Date:  2020-02-24       Impact factor: 17.367

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