Literature DB >> 25916088

Early effects of oral administration of esomeprazole and omeprazole on the intragastric pH.

Hiroshi Iida, Masahiko Inamori, Kotone Okuno, Yusuke Sekino, Eiji Sakai, Hidenori Okubo, Takuma Higurashi, Hiroki Endo, Kunihiro Hosono, Masato Yoneda, Tomoko Koide, Hirokazu Takahashi, Ayumu Goto, Kensuke Kubota, Satoru Saito, Shin Maeda, Atsushi Nakajima, Eiji Gotoh.   

Abstract

BACKGROUND/AIMS: The aim of our study was to investigate the inhibitory effects on gastric acid secretion of a single oral dose of a proton pump inhibitor, esomeprazole 20 mg and omeprazole 20 mg.
METHODOLOGY: A total of 14 Helicobacter pylori-negative male subjects participated in this study. Intragastric pH was monitored continuously for 6 hours after a single oral dose of omeprazole 20 mg and a single oral dose of esomeprazole 20 mg. Each administration was separated by a 7-day washout period.
RESULTS: During the 6-hour study period, the average pH after administration of esomeprazole was higher than that after the administration of omeprazole. Also during the 6-hour study period, each of pH > 2, 3, 3.5, 4, and 5 was maintained for a longer duration after administration of esomeprazole 20 mg than after administration of omeprazole 20 mg (median: 75.4% vs. 53.8%, p = 0.0138; 52.1% vs. 33.4%, p = 0.0188; 45.8% vs. 28.2%, p = 0.0262; 42.5% vs. 20.7%, p = 0.0414; 35.8% vs. 11.6%, p = 0.0262; respectively).
CONCLUSIONS: In Helicobacter pylori-negative healthy male subjects, single oral administration of esomeprazole 20 mg increased the intragastric pH more rapidly than single oral administration of omeprazole 20 mg.

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Year:  2015        PMID: 25916088

Source DB:  PubMed          Journal:  Hepatogastroenterology        ISSN: 0172-6390


  2 in total

1.  Pharmacokinetics and Acid Suppressant Efficacy of Esomeprazole after Intravenous, Oral, and Subcutaneous Administration to Healthy Beagle Dogs.

Authors:  J-H Hwang; J-W Jeong; G-H Song; T-S Koo; K-W Seo
Journal:  J Vet Intern Med       Date:  2017-04-13       Impact factor: 3.333

2.  Pharmacokinetics and pharmacodynamics of intravenous esomeprazole at 2 different dosages in dogs.

Authors:  Do-Hyun Seo; Jong-Bok Lee; Ji-Hye Hwang; Jong-Woo Jeong; Gun-Ho Song; Tae-Sung Koo; Kyoung-Won Seo
Journal:  J Vet Intern Med       Date:  2018-12-13       Impact factor: 3.333

  2 in total

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