Literature DB >> 25819462

Treatment of spontaneous preterm labour with retosiban: a phase 2 proof-of-concept study.

Steven Thornton1, Hugh Miller2, Guillermo Valenzuela3, Jerry Snidow4, Brendt Stier5, Michael J Fossler5, Timothy H Montague5, Marcy Powell4, Kathleen J Beach5.   

Abstract

AIM: The aim was to investigate the efficacy and safety of intravenous retosiban in women with spontaneous preterm labour.
METHODS: This was a randomized, double-blind, placebo-controlled, phase 2 trial. Retosiban was administered intravenously for 48 h to women in spontaneous preterm labour between 30(0/7) and 35(6/7)  weeks' gestation with an uncomplicated singleton pregnancy in an in-patient obstetric unit. Outcome measures were uterine quiescence (primary endpoint), days to delivery, preterm delivery and safety.
RESULTS: Uterine quiescence was achieved in 62% of women who received retosiban (n = 30) compared with 41% who received placebo (n = 34). The relative risk (RR) was 1.53 (95% credible interval [CrI] 0.98, 2.48; NS). Retosiban resulted in a significant increase in time to delivery compared with placebo (mean difference 8.2 days, 95% CrI 2.7, 13.74). This difference was consistent across all gestational ages. The proportion of preterm births in the retosiban and placebo groups was 18.7% (95% CrI 7.4%, 33.7%) and 47.2% (95% CrI 31.4%, 63.4%), respectively. The RR of preterm birth in women treated with retosiban was 0.38 (95% CrI 0.15, 0.81). There were no deliveries within 7 days in the retosiban group, but there were six (17.6%) births in the placebo group. The maternal, fetal and neonatal adverse events were comparable in the retosiban and placebo groups.
CONCLUSIONS: Intravenous administration of retosiban in women with spontaneous preterm labour was associated with a greater than 1 week increase in time to delivery compared with placebo, a significant reduction in preterm deliveries, a non-significant increase in uterine quiescence and a favourable safety profile.
© 2015 The British Pharmacological Society.

Entities:  

Keywords:  preterm birth; preterm labour; proof-of-concept study; retosiban; uterine quiescence

Mesh:

Substances:

Year:  2015        PMID: 25819462      PMCID: PMC4594710          DOI: 10.1111/bcp.12646

Source DB:  PubMed          Journal:  Br J Clin Pharmacol        ISSN: 0306-5251            Impact factor:   4.335


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