Literature DB >> 25754950

Haematological cancer: BCL-ABL1 resistance mutation--breakthrough with axitinib.

David Killock.   

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Year:  2015        PMID: 25754950     DOI: 10.1038/nrclinonc.2015.42

Source DB:  PubMed          Journal:  Nat Rev Clin Oncol        ISSN: 1759-4774            Impact factor:   66.675


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  1 in total

1.  Axitinib effectively inhibits BCR-ABL1(T315I) with a distinct binding conformation.

Authors:  Tea Pemovska; Eric Johnson; Mika Kontro; Gretchen A Repasky; Jeffrey Chen; Peter Wells; Ciarán N Cronin; Michele McTigue; Olli Kallioniemi; Kimmo Porkka; Brion W Murray; Krister Wennerberg
Journal:  Nature       Date:  2015-02-09       Impact factor: 49.962

  1 in total

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