Literature DB >> 25748298

Factors influencing the development of cutaneous squamous cell carcinoma in patients on BRAF inhibitor therapy.

Rachael Anforth1, Alexander Menzies2, Karen Byth3, Giuliana Carlos1, Shaun Chou4, Raghwa Sharma5, Richard A Scolyer6, Richard Kefford2, Georgina V Long2, Pablo Fernandez-Peñas7.   

Abstract

BACKGROUND: BRAF inhibitors (BRAFi) cause paradoxical activation of the MAPK pathway in keratinocytes resulting in cutaneous squamous cell carcinoma (cuSCC).
OBJECTIVE: We sought to examine the clinical factors involved in BRAFi-induced cuSCC development.
METHODS: We studied 134 patients with BRAF-mutant metastatic melanoma treated with a BRAFi at Westmead Hospital, Sydney, Australia. Details of cuSCC development and associations with melanoma clinicopathologic features and treatment outcome were examined.
RESULTS: In all, 32 (24%) patients developed 110 cuSCC after commencing treatment. In all, 61 (55%) cuSCC developed within the first 3 months. Age was the only independent risk factor for cuSCC development. After 3 months of therapy 4% of patients younger than 40 years developed cuSCC compared with 33% who were older than 60 years, and the hazard ratio of developing a cuSCC increased by 1.7 (95% confidence interval 1.3-2.3) per decade (P < .001). BRAFi cuSCC occurred more often in sun-protected areas (42%) compared with sporadic cuSCC (21%) (P < .001). cuSCC was not associated with progression-free survival. LIMITATIONS: The study was from a single center and patients were also at risk of sporadic cuSCC.
CONCLUSION: Most BRAFi-induced cuSCC develop within 3 months of BRAFi therapy. The only independent risk factor is increasing age. cuSCC may present in anatomical locations with low ultraviolet exposure such that thorough dermatologic assessment is required.
Copyright © 2015 American Academy of Dermatology, Inc. Published by Elsevier Inc. All rights reserved.

Entities:  

Keywords:  BRAF inhibitors; cutaneous squamous cell carcinoma; dabrafenib; melanoma; vemurafenib

Mesh:

Substances:

Year:  2015        PMID: 25748298     DOI: 10.1016/j.jaad.2015.01.018

Source DB:  PubMed          Journal:  J Am Acad Dermatol        ISSN: 0190-9622            Impact factor:   11.527


  10 in total

1.  Inhibition of oncogenic BRAF activity by indole-3-carbinol disrupts microphthalmia-associated transcription factor expression and arrests melanoma cell proliferation.

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Journal:  Mol Carcinog       Date:  2016-02-15       Impact factor: 4.784

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Journal:  Drug Saf       Date:  2020-05       Impact factor: 5.606

Review 3.  NRAS mutant melanoma: an overview for the clinician for melanoma management.

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Journal:  Melanoma Manag       Date:  2016-02-17

Review 4.  Management of the cutaneous adverse effects of antimelanoma therapy.

Authors:  Rose Congwei Liu; Germana Consuegra; Pablo Fernández-Peñas
Journal:  Melanoma Manag       Date:  2017-11-22

Review 5.  Cutaneous Adverse Events of Anti-PD-1 Therapy and BRAF Inhibitors.

Authors:  Subashini Sharon Gnanendran; Lauren Maree Turner; James Austin Miller; Shelley Ji Eun Hwang; Andrew Charles Miller
Journal:  Curr Treat Options Oncol       Date:  2020-03-19

Review 6.  Drug Combinations as the New Standard for Melanoma Treatment.

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Journal:  Curr Treat Options Oncol       Date:  2016-12

Review 7.  Oh, the Mutations You'll Acquire! A Systematic Overview of Cutaneous Squamous Cell Carcinoma.

Authors:  Stephenie Droll; Xiaomin Bao
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8.  Adverse Effects of Vemurafenib on Skin Integrity: Hyperkeratosis and Skin Cancer Initiation Due to Altered MEK/ERK-Signaling and MMP Activity.

Authors:  Marius Tham; Hans-Jürgen Stark; Anna Jauch; Catherine Harwood; Elizabeth Pavez Lorie; Petra Boukamp
Journal:  Front Oncol       Date:  2022-01-31       Impact factor: 6.244

9.  Phase I, Open-Label, Dose-Escalation/Dose-Expansion Study of Lifirafenib (BGB-283), an RAF Family Kinase Inhibitor, in Patients With Solid Tumors.

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Journal:  J Clin Oncol       Date:  2020-03-17       Impact factor: 44.544

Review 10.  Cutaneous Squamous Cell Carcinoma: From Biology to Therapy.

Authors:  Roberto Corchado-Cobos; Natalia García-Sancha; Rogelio González-Sarmiento; Jesús Pérez-Losada; Javier Cañueto
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  10 in total

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