Literature DB >> 25735400

Long-term glycaemic response and tolerability of dapagliflozin versus a sulphonylurea as add-on therapy to metformin in patients with type 2 diabetes: 4-year data.

S Del Prato1, M Nauck2, S Durán-Garcia3, L Maffei4, K Rohwedder5, A Theuerkauf6, S Parikh7.   

Abstract

AIMS: To assess the long-term efficacy and tolerability of dapagliflozin versus glipizide as add-on to metformin in patients with inadequately controlled type 2 diabetes.
METHODS: The present study was an extension of an earlier randomized, double-blind, phase III study of dapagliflozin (n = 406) vs glipizide (n = 408) to 208 weeks (4 years). Patients continued to receive their assigned medication. No statistical treatment-group comparisons were calculated.
RESULTS: At 208 weeks, dapagliflozin compared with glipizide produced sustained reductions in glycated haemoglogin (HbA1c): -0.30% [95% confidence interval (CI), -0.51 to -0.09], in total body weight: -4.38 kg (95% CI -5.31 to -3.46) and in systolic blood pressure (SBP): -3.67 mmHg (95% CI -5.92 to -1.41). The HbA1c coefficient of failure was significantly lower for dapagliflozin than for glipizide: 0.19 (95% CI 0.12-0.25) versus 0.61 (95% CI 0.49-0.72, difference -0.42; p = 0.0001). Dapagliflozin was not associated with glomerular function deterioration, while this occurred more frequently in patients in the glipizide group. Fewer patients reported hypoglycaemia in the dapagliflozin compared with the glipizide group (5.4 vs 51.5%). Genital and urinary tract infections were more common with dapagliflozin than with glipizide, but their incidence decreased with time and all events responded well to antimicrobial treatment.
CONCLUSIONS: In patients completing 4 years of treatment, dapagliflozin was well tolerated and associated with sustained glycaemic efficacy and greater reductions in body weight and SBP versus glipizide.
© 2015 John Wiley & Sons Ltd.

Entities:  

Keywords:  SGLT2 inhibitor; dapagliflozin; durability; efficacy; safety; type 2 diabetes

Mesh:

Substances:

Year:  2015        PMID: 25735400     DOI: 10.1111/dom.12459

Source DB:  PubMed          Journal:  Diabetes Obes Metab        ISSN: 1462-8902            Impact factor:   6.577


  62 in total

Review 1.  Early Combination Therapy with Oral Glucose-Lowering Agents in Type 2 Diabetes.

Authors:  Cristina Bianchi; Giuseppe Daniele; Angela Dardano; Roberto Miccoli; Stefano Del Prato
Journal:  Drugs       Date:  2017-03       Impact factor: 9.546

Review 2.  The actions of SGLT2 inhibitors on metabolism, renal function and blood pressure.

Authors:  Merlin C Thomas; David Z I Cherney
Journal:  Diabetologia       Date:  2018-08-22       Impact factor: 10.122

3.  Impaired Store-Operated Calcium Entry and STIM1 Loss Lead to Reduced Insulin Secretion and Increased Endoplasmic Reticulum Stress in the Diabetic β-Cell.

Authors:  Tatsuyoshi Kono; Xin Tong; Solaema Taleb; Robert N Bone; Hitoshi Iida; Chih-Chun Lee; Paul Sohn; Patrick Gilon; Michael W Roe; Carmella Evans-Molina
Journal:  Diabetes       Date:  2018-08-21       Impact factor: 9.461

Review 4.  Obesity medications in development.

Authors:  Candida J Rebello; Frank L Greenway
Journal:  Expert Opin Investig Drugs       Date:  2019-12-19       Impact factor: 6.206

Review 5.  Renal sodium-glucose cotransporter inhibition in the management of type 2 diabetes mellitus.

Authors:  Muhammad A Abdul-Ghani; Luke Norton; Ralph A DeFronzo
Journal:  Am J Physiol Renal Physiol       Date:  2015-09-09

Review 6.  Saving the sweetness: renal glucose handling in health and disease.

Authors:  Blythe D Shepard; Jennifer L Pluznick
Journal:  Am J Physiol Renal Physiol       Date:  2017-03-29

7.  Management of hyperglycaemia in type 2 diabetes, 2018. A consensus report by the American Diabetes Association (ADA) and the European Association for the Study of Diabetes (EASD).

Authors:  Melanie J Davies; David A D'Alessio; Judith Fradkin; Walter N Kernan; Chantal Mathieu; Geltrude Mingrone; Peter Rossing; Apostolos Tsapas; Deborah J Wexler; John B Buse
Journal:  Diabetologia       Date:  2018-12       Impact factor: 10.122

Review 8.  Renal, metabolic and cardiovascular considerations of SGLT2 inhibition.

Authors:  Ralph A DeFronzo; Luke Norton; Muhammad Abdul-Ghani
Journal:  Nat Rev Nephrol       Date:  2016-12-12       Impact factor: 28.314

9.  Cost-Effectiveness of Dapagliflozin as Add-On to Metformin for the Treatment of Type 2 Diabetes Mellitus in Greece.

Authors:  Charalampos Tzanetakos; Nicholas Tentolouris; Georgia Kourlaba; Nikos Maniadakis
Journal:  Clin Drug Investig       Date:  2016-08       Impact factor: 2.859

10.  Efficacy and Safety Over 2 Years of Exenatide Plus Dapagliflozin in the DURATION-8 Study: A Multicenter, Double-Blind, Phase 3, Randomized Controlled Trial.

Authors:  Serge A Jabbour; Juan P Frías; Azazuddin Ahmed; Elise Hardy; Jasmine Choi; C David Sjöström; Cristian Guja
Journal:  Diabetes Care       Date:  2020-08-18       Impact factor: 19.112

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.