Literature DB >> 25532017

Epigenetics: novel therapeutics targeting epigenetics.

Stuart J Conway1, Patrick M Woster, Jing-Kang Shen, Gunda Georg, Shaomeng Wang.   

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Year:  2014        PMID: 25532017     DOI: 10.1021/jm501941q

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


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  3 in total

1.  Histone Deacetylase Inhibitory Activity and Antiproliferative Potential of New [6]-Shogaol Derivatives.

Authors:  Chanokbhorn Phaosiri; Chavi Yenjai; Thanaset Senawong; Gulsiri Senawong; Somprasong Saenglee; La-Or Somsakeesit; Pakit Kumboonma
Journal:  Molecules       Date:  2022-05-22       Impact factor: 4.927

2.  Dual NAMPT/HDAC Inhibitors as a New Strategy for Multitargeting Antitumor Drug Discovery.

Authors:  Wei Chen; Guoqiang Dong; Ying Wu; Wannian Zhang; Chaoyu Miao; Chunquan Sheng
Journal:  ACS Med Chem Lett       Date:  2017-12-14       Impact factor: 4.345

3.  Development of a Novel Positron Emission Tomography (PET) Radiotracer Targeting Bromodomain and Extra-Terminal Domain (BET) Family Proteins.

Authors:  Ping Bai; Yu Lan; Hao Wang; Zude Chen; Stephanie Fiedler; Robin Striar; Xiaoxia Lu; Changning Wang
Journal:  Front Mol Biosci       Date:  2020-08-12
  3 in total

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