Literature DB >> 25376458

Inhibitor of apoptosis proteins (IAPs) may be effective therapeutic targets for treating endometriosis.

Takashi Uegaki1, Fuminori Taniguchi2, Kazuomi Nakamura3, Mitsuhiko Osaki4, Futoshi Okada4, Osamu Yamamoto5, Tasuku Harada1.   

Abstract

STUDY QUESTION: What is the role of the inhibitor of apoptosis proteins (IAPs) in human endometriotic tissues and a mouse model of endometriosis? SUMMARY ANSWER: Four IAP proteins were expressed in endometriotic tissue indicating IAPs may be a key factor in the pathogenesis and progression of endometriosis. WHAT IS KNOWN ALREADY: Overexpression of IAPs protects against a number of proapoptotic stimuli. IAPs (c-IAP1, c-IAP2, XIAP and Survivin) are expressed in human ectopic endometrial stromal cells (ESCs) from ovarian endometriomas. STUDY DESIGN, SIZE, DURATION: Forty-eight women with or without ovarian endometrioma are included in this study. BALB/c mice (n = 24) were used for the mouse endometriosis model. Mice with surgically induced endometriosis were treated with an IAP antagonist (BV6) for 4 weeks. PARTICIPANTS/MATERIALS, SETTING,
METHODS: Human ectopic endometrial tissues from chocolate cysts and eutopic endometrial tissue were collected. ESCs were enzymatically isolated from these tissues. ESC proliferation was examined by 5-bromo-2'-deoxyuridine-enzyme-linked immunosorbent assay. IAPs expression in tissue derived from eutopic endometria and chocolate cysts was evaluated using real-time RT-PCR and immunohistochemistry. A homologous mouse endometriosis model was established by transplanting donor mouse uterine tissue into the abdominal cavities of recipient mice. After treating the mice with BV6 (i.p. 10 mg/ml), the extent of endometriosis-like lesions in mice was measured and proliferative activity assessed by Ki67 staining. All experiments were repeated a minimum of three times. MAIN RESULTS AND THE ROLE OF CHANCE: IAP (c-IAP1, c-IAP2, XIAP and Survivin) mRNA and protein in human ectopic endometrial tissues were expressed at higher levels than in eutopic endometrial tissues (P < 0.05). All four IAPs proteins were expressed in mouse endometriosis-like implants. BV6 inhibited BrdU incorporation of human ESCs (P < 0.05 versus control). BV6 also decreased the total number, weight, surface area and Ki67 positive cells in the endometriosis-like lesions in the mice (P < 0.05 versus control). LIMITATIONS, REASONS FOR CAUTION: Endometriotic lesions were surgically induced in mice by transplanting mouse uterine tissue only, not human pathological endometriotic tissue. Furthermore, the effects of BV6 on human ESCs and mouse endometriosis-like lesions may differ between the species. WIDER IMPLICATIONS OF THE
FINDINGS: Our data support the hypothesis that IAPs are involved in the development of endometriosis, and therefore an inhibitor of IAPs has potential as a novel treatment for endometriosis. STUDY FUNDING/COMPETING INTERESTS: This work was supported by KAKENHI (Japan Society for the Promotion of Science, Grant-in-Aid: to F.T.; 21592098 and to T.H.; 24659731) and Yamaguchi Endocrine Research Foundation. The authors have no conflicts of interest to disclose.
© The Author 2014. Published by Oxford University Press on behalf of the European Society of Human Reproduction and Embryology. All rights reserved. For Permissions, please email: journals.permissions@oup.com.

Entities:  

Keywords:  BV6; endometrial stromal cells; inhibitor of apoptosis proteins family; mouse endometriosis model

Mesh:

Substances:

Year:  2014        PMID: 25376458      PMCID: PMC4262468          DOI: 10.1093/humrep/deu288

Source DB:  PubMed          Journal:  Hum Reprod        ISSN: 0268-1161            Impact factor:   6.918


  33 in total

1.  Apoptosis in endometrial glandular and stromal cells in women with and without endometriosis.

Authors:  W P Dmowski; J Ding; J Shen; N Rana; B B Fernandez; D P Braun
Journal:  Hum Reprod       Date:  2001-09       Impact factor: 6.918

2.  Cellular inhibitors of apoptosis are global regulators of NF-κB and MAPK activation by members of the TNF family of receptors.

Authors:  Eugene Varfolomeev; Tatiana Goncharov; Heather Maecker; Kerry Zobel; László G Kömüves; Kurt Deshayes; Domagoj Vucic
Journal:  Sci Signal       Date:  2012-03-20       Impact factor: 8.192

3.  Role of estrogen receptor signaling required for endometriosis-like lesion establishment in a mouse model.

Authors:  Katherine A Burns; Karina F Rodriguez; Sylvia C Hewitt; Kyathanahalli S Janardhan; Steven L Young; Kenneth S Korach
Journal:  Endocrinology       Date:  2012-06-14       Impact factor: 4.736

4.  The cellular inhibitor of apoptosis protein-2 is a possible target of novel treatment for endometriosis.

Authors:  Fuminori Taniguchi; Hiroko Higaki; Masao Izawa; Yukihiro Azuma; Eriko Hirakawa; Imari Deura; Tomio Iwabe; Kohkichi Hata; Tasuku Harada
Journal:  Am J Reprod Immunol       Date:  2014-01-02       Impact factor: 3.886

5.  Bcl-2 and Fas expression in eutopic and ectopic human endometrium during the menstrual cycle in relation to endometrial cell apoptosis.

Authors:  H Watanabe; H Kanzaki; S Narukawa; T Inoue; H Katsuragawa; Y Kaneko; T Mori
Journal:  Am J Obstet Gynecol       Date:  1997-02       Impact factor: 8.661

6.  Tumor necrosis factor-alpha-induced interleukin-8 (IL-8) expression in endometriotic stromal cells, probably through nuclear factor-kappa B activation: gonadotropin-releasing hormone agonist treatment reduced IL-8 expression.

Authors:  Yasuko Sakamoto; Tasuku Harada; Sayako Horie; Yumiko Iba; Fuminori Taniguchi; Souichi Yoshida; Tomio Iwabe; Naoki Terakawa
Journal:  J Clin Endocrinol Metab       Date:  2003-02       Impact factor: 5.958

Review 7.  Targeting IAP (inhibitor of apoptosis) proteins for therapeutic intervention in tumors.

Authors:  Domagoj Vucic
Journal:  Curr Cancer Drug Targets       Date:  2008-03       Impact factor: 3.428

8.  X chromosome-linked inhibitor of apoptosis regulates cell death induction by proapoptotic receptor agonists.

Authors:  Eugene Varfolomeev; Bruno Alicke; J Michael Elliott; Kerry Zobel; Kristina West; Harvey Wong; Justin M Scheer; Avi Ashkenazi; Stephen E Gould; Wayne J Fairbrother; Domagoj Vucic
Journal:  J Biol Chem       Date:  2009-10-23       Impact factor: 5.157

Review 9.  Evaluation and management of women with endometriosis.

Authors:  Craig A Winkel
Journal:  Obstet Gynecol       Date:  2003-08       Impact factor: 7.661

10.  Creation of immortalised epithelial cells from ovarian endometrioma.

Authors:  Y Bono; S Kyo; M Takakura; Y Maida; Y Mizumoto; M Nakamura; K Nomura; T Kiyono; M Inoue
Journal:  Br J Cancer       Date:  2012-02-21       Impact factor: 7.640

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  3 in total

1.  Identification of key genes and pathways in endometriosis by integrated expression profiles analysis.

Authors:  Ding Cui; Yang Liu; Junyan Ma; Kaiqing Lin; Kaihong Xu; Jun Lin
Journal:  PeerJ       Date:  2020-12-07       Impact factor: 2.984

Review 2.  Endometriosis in the Mouse: Challenges and Progress Toward a 'Best Fit' Murine Model.

Authors:  Katherine A Burns; Amelia M Pearson; Jessica L Slack; Elaine D Por; Alicia N Scribner; Nazmin A Eti; Richard O Burney
Journal:  Front Physiol       Date:  2022-01-13       Impact factor: 4.566

3.  Interleukin-1/-33 Signaling Pathways as Therapeutic Targets for Endometriosis.

Authors:  Toru Kato; Koubun Yasuda; Kazufumi Matsushita; Ken J Ishii; Seiichi Hirota; Tomohiro Yoshimoto; Hiroaki Shibahara
Journal:  Front Immunol       Date:  2019-08-22       Impact factor: 7.561

  3 in total

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