Literature DB >> 25223403

Concise synthesis of 2,4-disubstituted thiazoles from β-azido disulfides and carboxylic acids or anhydrides: asymmetric synthesis of cystothiazole C.

Yi Liu1, Xue Sun, Xing Zhang, Jun Liu, Yuguo Du.   

Abstract

A novel and efficient method for the one-pot synthesis of 2,4-disubstituted thiazoles from carboxylic acids or anhydrides is presented. Based on this new method, the total synthesis of the bis-2,4-disubstituted bis(thiazoles) natural product cystothiazole C is also presented.

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Year:  2014        PMID： 25223403     DOI： 10.1039/c4ob01460j

Source DB:  PubMed          Journal:  Org Biomol Chem        ISSN： 1477-0520            Impact factor:   3.876


  3 in total

1.  Cysteine Isocyanide in Multicomponent Reaction: Synthesis of Peptido-Mimetic 1,3-Azoles.

Authors:  Thimmalapura M Vishwanatha; Katarzyna Kurpiewska; Justyna Kalinowska-Tłuścik; Alexander Dömling
Journal:  J Org Chem       Date:  2017-08-25       Impact factor: 4.354

Review 2.  Thiazoles and Thiazolidinones as COX/LOX Inhibitors.

Authors:  Konstantinos Liaras; Maria Fesatidou; Athina Geronikaki
Journal:  Molecules       Date:  2018-03-18       Impact factor: 4.411

3.  Catalyst-free reductive cyclization of bis(2-aminophenyl) disulfide with CO2 in the presence of BH3NH3 to synthesize 2-unsubstituted benzothiazole derivatives.

Authors:  Xiao Li; Zhenbao Liu; Hailong Hong; Limin Han; Ning Zhu
Journal:  RSC Adv       Date:  2022-06-20       Impact factor: 4.036
  3 in total

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