Literature DB >> 25218708

Ixabepilone alone or with cetuximab as first-line treatment for advanced/metastatic triple-negative breast cancer.

Olivier Trédan1, Mario Campone2, Jacek Jassem3, Rostislav Vyzula4, Bruno Coudert5, Carmen Pacilio6, Jana Prausova7, Anne-Claire Hardy-Bessard8, Ana Arance9, Pralay Mukhopadhyay10, Alessandra Aloe11, Henri Roché12.   

Abstract

BACKGROUND: Despite high initial sensitivity to chemotherapy, TNBC is associated with a poor prognosis, highlighting the need for novel therapeutic strategies. The aim of this multicenter, randomized, open-label phase II trial was to assess the efficacy of ixabepilone as monotherapy, and the combination of ixabepilone with cetuximab, as first-line treatment in patients with triple-negative locally advanced nonresectable and/or metastatic breast cancer. PATIENTS AND METHODS: Women were randomly assigned to receive either ixabepilone (40 mg/m(2)) every 21 days (n = 40), or ixabepilone (40 mg/m(2)) every 21 days with cetuximab (400 mg/m(2) loading dose, followed by 250 mg/m(2)) once weekly (n = 39). The primary end point of the trial was to estimate the response rates of ixabepilone monotherapy and ixabepilone with cetuximab combination therapy.
RESULTS: Of 79 randomized patients, 77 were treated. Based on an intent-to-treat analysis, an objective response rate of 30% (95% confidence interval [CI], 16.6-46.5) was observed in the monotherapy arm, and 35.9% (95% CI, 21.2-52.8) in the combination arm. Median progression-free survival was 4.1 months in both treatment groups. Safety findings were consistent with the known individual toxicity profiles of ixabepilone and cetuximab. Skin and subcutaneous tissue disorders were more common with combination therapy, as were discontinuations because of adverse events.
CONCLUSION: Ixabepilone monotherapy and the ixabepilone and cetuximab combination demonstrated similar levels of clinical activity in first-line treatment of advanced TNBC, with a predictable safety profile. Further investigation of novel therapies for TNBC is required to improve patient outcomes.
Copyright © 2015 Elsevier Inc. All rights reserved.

Entities:  

Keywords:  Cetuximab; EGFR; Ixabepilone; Metastatic breast cancer; Triple negative

Mesh:

Substances:

Year:  2014        PMID: 25218708     DOI: 10.1016/j.clbc.2014.07.007

Source DB:  PubMed          Journal:  Clin Breast Cancer        ISSN: 1526-8209            Impact factor:   3.225


  27 in total

Review 1.  Clinical implications of molecular heterogeneity in triple negative breast cancer.

Authors:  Brian D Lehmann; Jennifer A Pietenpol
Journal:  Breast       Date:  2015-08-05       Impact factor: 4.380

Review 2.  Systemic treatment approaches in her2-negative advanced breast cancer-guidance on the guidelines.

Authors:  A A Joy; M Ghosh; R Fernandes; M J Clemons
Journal:  Curr Oncol       Date:  2015-03       Impact factor: 3.677

3.  Prognostic Evaluation of Epidermal Growth Factor Receptor (EGFR) Genotype and Phenotype Parameters in Triple-negative Breast Cancers.

Authors:  Sofia Levva; Vassiliki Kotoula; Ioannis Kostopoulos; Kyriaki Manousou; Christos Papadimitriou; Kyriaki Papadopoulou; Sotiris Lakis; Kyriakos Koukoulias; Vasilios Karavasilis; George Pentheroudakis; Eufemia Balassi; Flora Zagouri; Ioannis G Kaklamanos; Dimitrios Pectasides; Evangelia Razis; Gerasimos Aravantinos; Pavlos Papakostas; Dimitrios Bafaloukos; Grigorios Rallis; Helen Gogas; George Fountzilas
Journal:  Cancer Genomics Proteomics       Date:  2017 May-Jun       Impact factor: 4.069

Review 4.  Therapeutic Implications of the Molecular and Immune Landscape of Triple-Negative Breast Cancer.

Authors:  Ana C Gregório; Manuela Lacerda; Paulo Figueiredo; Sérgio Simões; Sérgio Dias; João Nuno Moreira
Journal:  Pathol Oncol Res       Date:  2017-09-14       Impact factor: 3.201

Review 5.  Early clinical development of epidermal growth factor receptor targeted therapy in breast cancer.

Authors:  Naoko Matsuda; Bora Lim; Xiaoping Wang; Naoto T Ueno
Journal:  Expert Opin Investig Drugs       Date:  2017-03-08       Impact factor: 6.206

Review 6.  A perspective on anti-EGFR therapies targeting triple-negative breast cancer.

Authors:  Katsuya Nakai; Mien-Chie Hung; Hirohito Yamaguchi
Journal:  Am J Cancer Res       Date:  2016-08-01       Impact factor: 6.166

7.  Metalloprotease-dependent activation of EGFR modulates CD44+/CD24- populations in triple negative breast cancer cells through the MEK/ERK pathway.

Authors:  Randi Wise; Anna Zolkiewska
Journal:  Breast Cancer Res Treat       Date:  2017-08-08       Impact factor: 4.872

Review 8.  Potentiating Therapeutic Effects of Epidermal Growth Factor Receptor Inhibition in Triple-Negative Breast Cancer.

Authors:  Kyu Sic You; Yong Weon Yi; Jeonghee Cho; Jeong-Soo Park; Yeon-Sun Seong
Journal:  Pharmaceuticals (Basel)       Date:  2021-06-18

9.  SGLT1 is required for the survival of triple-negative breast cancer cells via potentiation of EGFR activity.

Authors:  Huiquan Liu; Ayse Ertay; Ping Peng; Juanjuan Li; Dian Liu; Hua Xiong; Yanmei Zou; Hong Qiu; David Hancock; Xianglin Yuan; Wei-Chien Huang; Rob M Ewing; Julian Downward; Yihua Wang
Journal:  Mol Oncol       Date:  2019-06-14       Impact factor: 6.603

Review 10.  Ixabepilone: Overview of Effectiveness, Safety, and Tolerability in Metastatic Breast Cancer.

Authors:  Nuhad K Ibrahim
Journal:  Front Oncol       Date:  2021-07-06       Impact factor: 6.244

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