Literature DB >> 25202099

Sorafenib efficacy in thymic carcinomas seems not to require c-KIT or PDGFR-alpha mutations.

Maria Pagano1, Nuria Maria Asensio Sierra2, Michele Panebianco2, Giulio Rossi3, Roberta Gnoni2, Giancarlo Bisagni2, Corrado Boni2.   

Abstract

PURPOSE: To retrospectively evaluate sorafenib activity and safety in patients with metastatic thymic carcinoma (TC) and to correlate outcome with c-KIT and PDGFR-alpha mutational status. PATIENTS AND METHODS: Patients with metastatic thymic carcinoma treated with sorafenib after at least one prior line of chemotherapy were included. Objective response rate (ORR) and toxicity were evaluated. Analysis of c-KIT and PDGFR-alpha mutational status was performed retrospectively.
RESULTS: From October 2007 to August 2011, 5 patients with metastatic thymic carcinoma were evaluated. A median of 8 cycles of sorafenib (range=3-29) were administered. Two patients (40%) displayed a partial response (PR), two patients presented stable disease (SD), while one patient had progression. The median progression-free (PFS) and overall survival were 28 weeks and 92 weeks, respectively. At mutational analysis, only one patient with PR had c-KIT mutation in exon 17 and was successfully treated with sunitinib for 12 months after progression to sorafenib. No PDGFR-alpha mutations were found.
CONCLUSION: Sorafenib activity seems independent from the c-KIT and PDGFR-alpha mutational status. After progression, sequence treatment with a different tyrosine kinase inhibitor can be considered. These results are promising and need further confirmation on larger, possibly prospective, series of patients. Copyright
© 2014 International Institute of Anticancer Research (Dr. John G. Delinassios), All rights reserved.

Entities:  

Keywords:  PDGFR alpha; Thymic carcinoma; c-KIT; sorafenib; tyrosine kinase

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Year:  2014        PMID: 25202099

Source DB:  PubMed          Journal:  Anticancer Res        ISSN: 0250-7005            Impact factor:   2.480


  4 in total

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Authors:  Fumihiko Hirai; Makoto Edagawa; Shinichiro Shimamatsu; Ryo Toyozawa; Gouji Toyokawa; Kaname Nosaki; Masafumi Yamaguchi; Takashi Seto; Mitsuhiro Twakenoyama; Yukito Ichinose
Journal:  Mol Clin Oncol       Date:  2016-01-28

2.  Sorafenib improves the postoperative effect of early stage renal cell carcinoma.

Authors:  Taiyang Liu; Jie Li; Xiuhua Wen; Zhang Hui; Gui Qi
Journal:  Oncol Lett       Date:  2016-10-12       Impact factor: 2.967

3.  Molecular Profiling of Thymoma and Thymic Carcinoma: Genetic Differences and Potential Novel Therapeutic Targets.

Authors:  Franz Enkner; Bettina Pichlhöfer; Alexandru Teodor Zaharie; Milica Krunic; Tina Maria Holper; Stefan Janik; Bernhard Moser; Karin Schlangen; Barbara Neudert; Karin Walter; Brigitte Migschitz; Leonhard Müllauer
Journal:  Pathol Oncol Res       Date:  2016-11-14       Impact factor: 3.201

4.  Targeted Next-Generation Sequencing of Thymic Epithelial Tumours Revealed Pathogenic Variants in KIT, ERBB2, KRAS, and TP53 in 30% of Thymic Carcinomas.

Authors:  Adam Szpechcinski; Malgorzata Szolkowska; Sebastian Winiarski; Urszula Lechowicz; Piotr Wisniewski; Magdalena Knetki-Wroblewska
Journal:  Cancers (Basel)       Date:  2022-07-12       Impact factor: 6.575

  4 in total

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