Literature DB >> 25175006

Long term retention of retigabine in a cohort of people with drug resistant epilepsy.

Tim Wehner1, Suganthi Chinnasami2, Jan Novy3, Gail S Bell4, John S Duncan5, Josemir W Sander6.   

Abstract

PURPOSE: To assess the utility of retigabine (RTG) for epilepsy in clinical practice at a single UK tertiary centre.
METHODS: We identified all individuals who were offered RTG from April 2011 to May 2013. We collected demographics, seizure types, previous and current antiepileptic drugs (AEDs), starting and maximum attained daily dose of RTG, clinical benefits, side effects, and reason to discontinue RTG from in- and outpatient encounters until February 28, 2014.
RESULTS: 145 people who had failed a median of 11 AEDs took at least one dose of RTG. One year retention was 32% and decreased following the safety alert by the US Federal Drug Administration (FDA) in April 2013. None became seizure free. 34 people (24%) reported a benefit that was ongoing at last assessment in five (3%). The most relevant benefit was the significant reduction or cessation of drop attacks or seizure-related falls in four women, this persisted at last assessment in two. The presence of simple partial seizures was associated with longer retention, as was a higher attained dose of RTG. Adverse effects were seen in 74% and largely CNS-related or nonspecific and affected the genitourinary system in 13%.
CONCLUSION: Retention of RTG was less favourable compared to data from open label extension studies of the regulatory trials. In comparison with historical data on similar retention audits retention of RTG at one year appears to be less than lamotrigine, topiramate, levetiracetam, pregabalin, zonisamide, and lacosamide, and slightly higher than gabapentin.
Copyright © 2014 The Authors. Published by Elsevier Ltd.. All rights reserved.

Entities:  

Keywords:  Antiepileptic drug; Efficacy; Tolerability

Mesh:

Substances:

Year:  2014        PMID: 25175006     DOI: 10.1016/j.seizure.2014.08.001

Source DB:  PubMed          Journal:  Seizure        ISSN: 1059-1311            Impact factor:   3.184


  4 in total

1.  Variability in expression of the human MDR1 drug efflux transporter and genetic variation of the ABCB1 gene: implications for drug-resistant epilepsy.

Authors:  Anna Heinrich; Xiao-Bo Zhong; Theodore P Rasmussen
Journal:  Curr Opin Toxicol       Date:  2018-12-18

Review 2.  Practical Use of Newer Antiepileptic Drugs as Adjunctive Therapy in Focal Epilepsy.

Authors:  Martin J Brodie
Journal:  CNS Drugs       Date:  2015-11       Impact factor: 5.749

Review 3.  Neuronal and Cardiovascular Potassium Channels as Therapeutic Drug Targets: Promise and Pitfalls.

Authors:  Edward S A Humphries; Caroline Dart
Journal:  J Biomol Screen       Date:  2015-08-24

4.  Efficacy of Retigabine on Acute Limbic Seizures in Adult Rats.

Authors:  L K Friedman; A M Slomko; J P Wongvravit; Z Naseer; S Hu; W Y Wan; S S Ali
Journal:  J Epilepsy Res       Date:  2015-12-31
  4 in total

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