Literature DB >> 25146938

Epidermal growth factor receptor (EGFR) exon 20 mutations in non-small-cell lung cancer and resistance to EGFR-tyrosine kinase inhibitors.

Hyun Sun Woo1, Hee Kyung Ahn, Ha Yeon Lee, Inkeun Park, Young Saing Kim, Junshik Hong, Sun Jin Sym, Jinny Park, Jae Hoon Lee, Dong Bok Shin, Eun Kyung Cho.   

Abstract

INTRODUCTION: In patients with non-small cell lung cancer (NSCLC), the predictive value of rare epidermal growth factor receptor (EGFR) exon 20 mutations in determining a patient's response to EGFR tyrosine kinase inhibitor (TKI) treatment is unclear. PATIENTS AND METHODS: We reviewed data for NSCLC patients harboring EGFR exon 20 mutations from two hospitals in Korea. EGFR mutations were analyzed using directional sequencing.
RESULTS: We identified eight patients carrying EGFR exon 20 mutations, seven of whom had insertional mutations. Three patients carried previously unreported insertional mutations. Among six patients who were treated with EGFR TKI, one showed stable disease and three showed primary resistance. Response evaluations were not performed for the other two patients because of their clinical deterioration.
CONCLUSIONS: EGFR exon 20 insertional mutations, including three that were previously unreported, were associated with the poor response of patients to TKI treatment.

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Year:  2014        PMID: 25146938     DOI: 10.1007/s10637-014-0146-x

Source DB:  PubMed          Journal:  Invest New Drugs        ISSN: 0167-6997            Impact factor:   3.850


  21 in total

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2.  Erlotinib versus standard chemotherapy as first-line treatment for European patients with advanced EGFR mutation-positive non-small-cell lung cancer (EURTAC): a multicentre, open-label, randomised phase 3 trial.

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Review 3.  Pathology of lung cancer.

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Journal:  Clin Chest Med       Date:  2011-12       Impact factor: 2.878

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Journal:  Clin Cancer Res       Date:  2004-12-15       Impact factor: 12.531

8.  Natural history and molecular characteristics of lung cancers harboring EGFR exon 20 insertions.

Authors:  Geoffrey R Oxnard; Peter C Lo; Mizuki Nishino; Suzanne E Dahlberg; Neal I Lindeman; Mohit Butaney; David M Jackman; Bruce E Johnson; Pasi A Jänne
Journal:  J Thorac Oncol       Date:  2013-02       Impact factor: 15.609

9.  Phase III study of afatinib or cisplatin plus pemetrexed in patients with metastatic lung adenocarcinoma with EGFR mutations.

Authors:  Lecia V Sequist; James Chih-Hsin Yang; Nobuyuki Yamamoto; Kenneth O'Byrne; Vera Hirsh; Tony Mok; Sarayut Lucien Geater; Sergey Orlov; Chun-Ming Tsai; Michael Boyer; Wu-Chou Su; Jaafar Bennouna; Terufumi Kato; Vera Gorbunova; Ki Hyeong Lee; Riyaz Shah; Dan Massey; Victoria Zazulina; Mehdi Shahidi; Martin Schuler
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10.  EGFR exon 20 insertion mutation in Japanese lung cancer.

Authors:  Hidefumi Sasaki; Katsuhiko Endo; Minoru Takada; Masaaki Kawahara; Naoto Kitahara; Hisaichi Tanaka; Meinoshin Okumura; Akihide Matsumura; Keiji Iuchi; Tomoya Kawaguchi; Osamu Kawano; Haruhiro Yukiue; Tomoki Yokoyama; Motoki Yano; Yoshitaka Fujii
Journal:  Lung Cancer       Date:  2007-08-07       Impact factor: 5.705

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  13 in total

1.  Uncommon EGFR mutations in lung carcinoma: features and treatment outcomes in a retrospective French cohort.

Authors:  Pierre Tankere; Romain Boidot; Philippe Bonniaud; Ayoube Zouak; Pascal Foucher; Alice Milliere; Aurélie Bertaut; Laure Favier; Aurélie Lagrange; François Ghiringhelli; Courèche Guillaume Kaderbhai; Cléa Fraisse
Journal:  J Thorac Dis       Date:  2022-06       Impact factor: 3.005

2.  Valproic acid, an inhibitor of class I histone deacetylases, reverses acquired Erlotinib-resistance of lung adenocarcinoma cells: a Connectivity Mapping analysis and an experimental study.

Authors:  Wenlei Zhuo; Liang Zhang; Yi Zhu; Qichao Xie; Bo Zhu; Zhengtang Chen
Journal:  Am J Cancer Res       Date:  2015-06-15       Impact factor: 6.166

3.  Screening for major driver oncogene alterations in adenosquamous lung carcinoma using PCR coupled with next-generation and Sanger sequencing methods.

Authors:  Xiaohua Shi; Huanwen Wu; Junliang Lu; Huanli Duan; Xuguang Liu; Zhiyong Liang
Journal:  Sci Rep       Date:  2016-02-29       Impact factor: 4.379

Review 4.  Not all epidermal growth factor receptor mutations in lung cancer are created equal: Perspectives for individualized treatment strategy.

Authors:  Yoshihisa Kobayashi; Tetsuya Mitsudomi
Journal:  Cancer Sci       Date:  2016-08-09       Impact factor: 6.716

5.  Non-classic EGFR mutations in a cohort of Dutch EGFR-mutated NSCLC patients and outcomes following EGFR-TKI treatment.

Authors:  J L Kuiper; S M S Hashemi; E Thunnissen; P J F Snijders; K Grünberg; E Bloemena; D Sie; P E Postmus; D A M Heideman; E F Smit
Journal:  Br J Cancer       Date:  2016-11-22       Impact factor: 7.640

6.  Epidermal growth factor receptor exon 20 mutation in lung cancer: types, incidence, clinical features and impact on treatment.

Authors:  Vanita Noronha; Anuradha Choughule; Vijay M Patil; Amit Joshi; Rajiv Kumar; Deepa Susan Joy Philip; Shripad Banavali; Amit Dutt; Kumar Prabhash
Journal:  Onco Targets Ther       Date:  2017-06-09       Impact factor: 4.147

7.  Clinical features and treatment outcome of non-small cell lung cancer (NSCLC) patients with uncommon or complex epidermal growth factor receptor (EGFR) mutations.

Authors:  Stefano Frega; Martina Lorenzi; Matteo Fassan; Stefano Indraccolo; Fiorella Calabrese; Adolfo Favaretto; Laura Bonanno; Valentina Polo; Giulia Zago; Francesca Lunardi; Ilaria Attili; Alberto Pavan; Massimo Rugge; Valentina Guarneri; PierFranco Conte; Giulia Pasello
Journal:  Oncotarget       Date:  2017-05-16

8.  Combination effects of ellagic acid with erlotinib in a Ba/F3 cell line expressing EGFR H773_V774 insH mutation.

Authors:  Chuanqi Xie; Jindong Kong; Fujun Miao; Xuanjun Wang; Jun Sheng
Journal:  Thorac Cancer       Date:  2020-06-11       Impact factor: 3.500

9.  [Clinical Features of EGFR Double Mutation in Non-small Cell Lung Cancer].

Authors:  Mengyao Wang; Dunqiang Ren; Caihong Guo; Xiaoqian Ding; Hongmei Wang
Journal:  Zhongguo Fei Ai Za Zhi       Date:  2018-08-20

Review 10.  Mechanisms of resistance to EGFR tyrosine kinase inhibitors.

Authors:  Lihua Huang; Liwu Fu
Journal:  Acta Pharm Sin B       Date:  2015-07-26       Impact factor: 11.413

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