Literature DB >> 25108579

Enzalutamide Antitumour Activity Against Metastatic Castration-resistant Prostate Cancer Previously Treated with Docetaxel and Abiraterone: A Multicentre Analysis.

Klaus Brasso1, Frederik B Thomsen2, Andres J Schrader3, Sebastian C Schmid4, David Lorente5, Margitta Retz4, Axel S Merseburger6, Christoph A von Klot6, Martin Boegemann7, Johann de Bono5.   

Abstract

BACKGROUND: The degree of antitumour activity of enzalutamide following disease progression on docetaxel and abiraterone remains controversial.
OBJECTIVE: To examine the effect of enzalutamide in patients progressing following taxane-based chemotherapy and abiraterone. DESIGN, SETTING, AND PARTICIPANTS: Metastatic castration-resistant prostate cancer patients entering one of four European compassionate use programmes of enzalutamide. OUTCOME MEASUREMENTS AND STATISTICAL ANALYSIS: The primary end point was overall survival (OS). Secondary end points were association between OS and posttreatment prostate-specific antigen (PSA) kinetics, patient characteristics, and progression-free survival, respectively. Kaplan-Meier survival analysis and Cox proportional hazard analysis were performed. RESULTS AND LIMITATIONS: We identified 137 patients who prior to enzalutamide had progressed following a median of eight cycles of docetaxel and seven courses of abiraterone. The median time on enzalutamide was 3.2 mo; median OS from the time patients started enzalutamide was 8.3 mo (95% confidence interval, 6.8-9.8). Only 45 (38%) and 22 (18%) patients had PSA declines (unconfirmed) >30% and 50%, respectively. Patients who had more than 30% or 50% falls in PSA had improved survival compared with patients who had no such PSA fall (11.4 mo vs 7.1 mo; p=0.001 and 12.6 vs 7.4 mo; p=0.007, respectively). Poor performance status and low haemoglobin was negatively associated with OS.
CONCLUSIONS: Median OS on enzalutamide following disease progression on taxane-based chemotherapy and abiraterone was modest, but patients who experience a PSA decline >30% or 50%, respectively, with enzalutamide in this setting had longer survival. PATIENT
SUMMARY: Enzalutamide produces modest prostate-specific antigen (PSA) responses in patients progressing following chemotherapy and abiraterone. Despite a modest PSA response, survival may still be improved.
Copyright © 2014 European Association of Urology. Published by Elsevier B.V. All rights reserved.

Entities:  

Keywords:  Abiraterone; Castration-resistant prostate cancer; Docetaxel; Enzalutamide; PSA; Survival

Mesh:

Substances:

Year:  2014        PMID: 25108579     DOI: 10.1016/j.eururo.2014.07.028

Source DB:  PubMed          Journal:  Eur Urol        ISSN: 0302-2838            Impact factor:   20.096


  31 in total

Review 1.  What do we know about treatment sequencing of abiraterone, enzalutamide, and chemotherapy in metastatic castration-resistant prostate cancer?

Authors:  Souhil Lebdai; Victor Basset; Julien Branchereau; Alexandre de La Taille; Vincent Flamand; Thierry Lebret; Thibaut Murez; Yann Neuzillet; Guillaume Ploussard; François Audenet
Journal:  World J Urol       Date:  2015-09-15       Impact factor: 4.226

Review 2.  An update on enzalutamide in the treatment of prostate cancer.

Authors:  Axel S Merseburger; Gabriel P Haas; Christoph-A von Klot
Journal:  Ther Adv Urol       Date:  2015-02

3.  Prostate cancer: Enzalutamide AFFIRMs its benefits.

Authors:  Robert Phillips
Journal:  Nat Rev Urol       Date:  2014-08-26       Impact factor: 14.432

4.  177Lu-PSMA-617 radioligand therapy and outcome in patients with metastasized castration-resistant prostate cancer.

Authors:  Axel Bräuer; Lena Sophie Grubert; Wolfgang Roll; Andres Jan Schrader; Michael Schäfers; Martin Bögemann; Kambiz Rahbar
Journal:  Eur J Nucl Med Mol Imaging       Date:  2017-06-17       Impact factor: 9.236

Review 5.  Sequencing Treatment for Castration-Resistant Prostate Cancer.

Authors:  Catherine E Handy; Emmanuel S Antonarakis
Journal:  Curr Treat Options Oncol       Date:  2016-12

Review 6.  [Systemic treatment of advanced prostate cancer].

Authors:  Alexander Kretschmer; Tilman Todenhöfer
Journal:  Urologe A       Date:  2020-12       Impact factor: 0.639

Review 7.  Managing Metastatic Castration-Resistant Prostate Cancer in the Pre-chemotherapy Setting: A Changing Approach in the Era of New Targeted Agents.

Authors:  Zafeiris Zafeiriou; Anuradha Jayaram; Adam Sharp; Johann S de Bono
Journal:  Drugs       Date:  2016-03       Impact factor: 9.546

8.  Synaptophysin expression on circulating tumor cells in patients with castration resistant prostate cancer undergoing treatment with abiraterone acetate or enzalutamide.

Authors:  Sumanta K Pal; Miaoling He; Lin Chen; Lixin Yang; Raju Pillai; Przemyslaw Twardowski; JoAnn Hsu; Marcin Kortylewski; Jeremy O Jones
Journal:  Urol Oncol       Date:  2017-12-27       Impact factor: 3.498

9.  Steroid sidestep: evading androgen ablation by abiraterone.

Authors:  Nima Sharifi
Journal:  Clin Cancer Res       Date:  2014-11-28       Impact factor: 12.531

Review 10.  Current treatment strategies for advanced prostate cancer.

Authors:  Kazumasa Komura; Christopher J Sweeney; Teruo Inamoto; Naokazu Ibuki; Haruhito Azuma; Philip W Kantoff
Journal:  Int J Urol       Date:  2017-12-20       Impact factor: 3.369

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