Literature DB >> 25008392

Fulranumab for treatment of diabetic peripheral neuropathic pain: A randomized controlled trial.

Hao Wang1, Gary Romano2, Mary Ellen Frustaci2, Norm Bohidar2, Huizhong Ma2, Panna Sanga2, Seth Ness2, Lucille J Russell2, Margaret Fedgchin2, Kathleen M Kelly2, John Thipphawong2.   

Abstract

OBJECTIVE: To assess efficacy and safety of fulranumab, a fully human monoclonal antibody against nerve growth factor, in patients with diabetic peripheral neuropathic pain (DPNP).
METHODS: In this phase II, double-blind, placebo-controlled trial, patients with moderate to severe DPNP were randomized to treatments with fulranumab (1, 3, or 10 mg) or placebo administered subcutaneously every 4 weeks.
RESULTS: Because of early study termination (clinical hold) by the US Food and Drug Administration, 77 (intent-to-treat) of the planned 200 patients were enrolled. The primary endpoint, the mean reduction of average daily pain at week 12 compared with baseline, showed a positive dose-response relationship (p = 0.014, 1-sided); the pair-wise comparison between the 10-mg group and placebo was significant (unadjusted p = 0.040, 2-sided). An exploratory responder analysis revealed that a greater proportion of patients in the 10-mg group reported ≥30% reduction in the average DPNP intensity compared with placebo at week 12 (p = 0.006). Although not statistically significant, several secondary endpoints showed directionally similar results to the primary efficacy dose-response relationship. During the combined efficacy and safety extension phases, the top 3 treatment-emergent adverse events in the combined fulranumab group were arthralgia (11%), edema peripheral (11%), and diarrhea (9%). No cases of joint replacement or death were reported.
CONCLUSION: Despite early study termination, fulranumab treatment resulted in dose-dependent efficacy and was generally well tolerated. CLASSIFICATION OF EVIDENCE: This study provides Class I evidence that in patients with DPNP, fulranumab 10 mg reduces pain by 1.2 points on an 11-point scale compared with placebo.
© 2014 American Academy of Neurology.

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Year:  2014        PMID: 25008392      PMCID: PMC4141990          DOI: 10.1212/WNL.0000000000000686

Source DB:  PubMed          Journal:  Neurology        ISSN: 0028-3878            Impact factor:   9.910


  33 in total

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  9 in total

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Journal:  Clin J Pain       Date:  2015-11       Impact factor: 3.442

Review 5.  Anti-nerve growth factor in pain management: current evidence.

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Journal:  J Pain Res       Date:  2016-06-08       Impact factor: 3.133

6.  Fulranumab in Patients With Pain Associated With Postherpetic Neuralgia and Postraumatic Neuropathy: Efficacy, Safety, and Tolerability Results From a Randomized, Double-blind, Placebo-controlled, Phase-2 Study.

Authors:  Hao Wang; Gary Romano; Margaret Fedgchin; Lucille Russell; Panna Sanga; Kathleen M Kelly; Mary Ellen Frustaci; John Thipphawong
Journal:  Clin J Pain       Date:  2017-02       Impact factor: 3.442

7.  Fulranumab in patients with interstitial cystitis/bladder pain syndrome: observations from a randomized, double-blind, placebo-controlled study.

Authors:  Hao Wang; Lucille J Russell; Kathleen M Kelly; Steven Wang; John Thipphawong
Journal:  BMC Urol       Date:  2017-01-05       Impact factor: 2.264

Review 8.  Challenges of neuropathic pain: focus on diabetic neuropathy.

Authors:  Daniela C Rosenberger; Vivian Blechschmidt; Hans Timmerman; André Wolff; Rolf-Detlef Treede
Journal:  J Neural Transm (Vienna)       Date:  2020-02-08       Impact factor: 3.575

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Journal:  Mol Pain       Date:  2017 Jan-Dec       Impact factor: 3.395

  9 in total

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