Literature DB >> 24888810

Randomized, phase III trial of first-line figitumumab in combination with paclitaxel and carboplatin versus paclitaxel and carboplatin alone in patients with advanced non-small-cell lung cancer.

Corey J Langer1, Silvia Novello2, Keunchil Park2, Maciej Krzakowski2, Daniel D Karp2, Tony Mok2, Rebecca J Benner2, Judith R Scranton2, Anthony J Olszanski2, Jacek Jassem2.   

Abstract

PURPOSE: Figitumumab (CP-751,871), a fully human immunoglobulin G2 monoclonal antibody, inhibits the insulin-like growth factor 1 receptor (IGF-1R). Our multicenter, randomized, phase III study compared figitumumab plus chemotherapy with chemotherapy alone as first-line treatment in patients with advanced non-small-cell lung cancer (NSCLC). PATIENTS AND METHODS: Patients with stage IIIB/IV or recurrent NSCLC disease with nonadenocarcinoma histology received open-label figitumumab (20 mg/kg) plus paclitaxel (200 mg/m(2)) and carboplatin (area under the concentration-time curve, 6 mg · min/mL) or paclitaxel and carboplatin alone once every 3 weeks for up to six cycles. The primary end point was overall survival (OS).
RESULTS: Of 681 randomly assigned patients, 671 received treatment. The study was closed early by an independent Data Safety Monitoring Committee because of futility and an increased incidence of serious adverse events (SAEs) and treatment-related deaths with figitumumab. Median OS was 8.6 months for figitumumab plus chemotherapy and 9.8 months for chemotherapy alone (hazard ratio [HR], 1.18; 95% CI, 0.99 to 1.40; P = .06); median progression-free survival was 4.7 months (95% CI, 4.2 to 5.4) and 4.6 months (95% CI, 4.2 to 5.4), respectively (HR, 1.10; P = .27); the objective response rates were 33% and 35%, respectively. The respective rates of all-causality SAEs were 66% and 51%; P < .01). Treatment-related grade 5 adverse events were also more common with figitumumab (5% v 1%; P < .01).
CONCLUSION: Adding figitumumab to standard chemotherapy failed to increase OS in patients with advanced nonadenocarcinoma NSCLC. Further clinical development of figitumumab is not being pursued.
© 2014 by American Society of Clinical Oncology.

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Year:  2014        PMID: 24888810      PMCID: PMC4067944          DOI: 10.1200/JCO.2013.54.4932

Source DB:  PubMed          Journal:  J Clin Oncol        ISSN: 0732-183X            Impact factor:   44.544


  11 in total

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Authors:  P Therasse; S G Arbuck; E A Eisenhauer; J Wanders; R S Kaplan; L Rubinstein; J Verweij; M Van Glabbeke; A T van Oosterom; M C Christian; S G Gwyther
Journal:  J Natl Cancer Inst       Date:  2000-02-02       Impact factor: 13.506

2.  Expression and function of the insulin-like growth factor I system in human non-small-cell lung cancer and normal lung cell lines.

Authors:  R E Favoni; A de Cupis; F Ravera; C Cantoni; P Pirani; A Ardizzoni; D Noonan; R Biassoni
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3.  Targeting the insulin-like growth factor receptor pathway in lung cancer: problems and pitfalls.

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Review 4.  Targeting insulin and insulin-like growth factor signalling in oncology.

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5.  Expression of insulin-like growth factor receptors I and II in normal human lung and in lung cancer.

Authors:  U Kaiser; C Schardt; D Brandscheidt; E Wollmer; K Havemann
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6.  Phase I, pharmacokinetic and pharmacodynamic study of the anti-insulinlike growth factor type 1 Receptor monoclonal antibody CP-751,871 in patients with multiple myeloma.

Authors:  Martha Q Lacy; Melissa Alsina; Rafael Fonseca; M Luisa Paccagnella; Carrie L Melvin; Donghua Yin; Amarnath Sharma; M Enriquez Sarano; Michael Pollak; Sundar Jagannath; Paul Richardson; Antonio Gualberto
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Review 8.  Emerging role of insulin-like growth factor receptor inhibitors in oncology: early clinical trial results and future directions.

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Journal:  Cancer Chemother Pharmacol       Date:  2012-07-19       Impact factor: 3.333

10.  Figitumumab combined with carboplatin and paclitaxel in treatment-naïve Japanese patients with advanced non-small cell lung cancer.

Authors:  Yasushi Goto; Ikuo Sekine; Maki Tanioka; Takashi Shibata; Chiharu Tanai; Hajime Asahina; Hiroshi Nokihara; Noboru Yamamoto; Hideo Kunitoh; Yuichiro Ohe; Hironori Kikkawa; Emiko Ohki; Tomohide Tamura
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Review 4.  A Review of Monoclonal Antibody-Based Treatments in Non-small Cell Lung Cancer.

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7.  Randomized Phase II Trial of Seribantumab in Combination with Erlotinib in Patients with EGFR Wild-Type Non-Small Cell Lung Cancer.

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Review 8.  Implications of Insulin-like Growth Factor 1 Receptor Activation in Lung Cancer.

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Review 9.  Insulin-like growth factor pathway aberrations and gastric cancer; evaluation of prognostic significance and assessment of therapeutic potentials.

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Review 10.  New advances in targeted gastric cancer treatment.

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