Literature DB >> 24865132

Safety and efficacy of the dipeptidyl peptidase-4 inhibitor linagliptin in elderly patients with type 2 diabetes: a comprehensive analysis of data from 1331 individuals aged ≥ 65 years.

G Schernthaner1, A H Barnett, S Patel, U Hehnke, M von Eynatten, H-J Woerle.   

Abstract

AIMS: To investigate individual patient data from a comprehensive trials programme to evaluate the safety and efficacy of the dipeptidyl peptidase-4 (DPP-4) inhibitor linagliptin across a range of glucose-lowering regimens in a large elderly population with type 2 diabetes mellitus (T2DM).
METHODS: Data were pooled from individuals aged ≥ 65 years, who participated in seven phase III, placebo-controlled clinical trials of linagliptin (24-52 weeks). Safety was assessed by incidence and severity of adverse events (AEs) with a focus on hypoglycaemia. The primary efficacy endpoint was change in glycated haemoglobin (HbA1c).
RESULTS: In total, 841 subjects received linagliptin 5 mg once a day and 490 received placebo. At baseline, the population had a mean ± s.d. age of 71.0 ± 4.6 years and a mean HbA1c concentration of 8.0 ± 0.8%; 63.5% of subjects received ≥ 2 antidiabetes drugs. Overall AEs and drug-related AEs were experienced by similar proportions of patients (linagliptin 71.3, placebo 73.3; linagliptin 18.1, placebo 19.8%, respectively). The incidence of investigator-reported hypoglycaemia was 21.4% with linagliptin and 25.7% with placebo. Severe hypoglycaemic events were rare and there were fewer in the linagliptin group (1.0 vs. 1.8%). At week 24, the placebo-corrected adjusted mean ± s.e. reduction in HbA1c with linagliptin was -0.62 ± 0.06% (95% CI: -0.73, -0.51).
CONCLUSIONS: Data from this large cohort show that linagliptin is a well-tolerated and efficacious therapy for elderly patients with T2DM. Treatment with linagliptin may support individualized treatment goals, while effectively managing the risk of hypoglycaemia or drug-related side effects.
© 2014 John Wiley & Sons Ltd.

Entities:  

Keywords:  DPP-IV inhibitor; diabetes mellitus

Mesh:

Substances:

Year:  2014        PMID: 24865132     DOI: 10.1111/dom.12321

Source DB:  PubMed          Journal:  Diabetes Obes Metab        ISSN: 1462-8902            Impact factor:   6.577


  7 in total

1.  A Randomized Controlled Study Comparing a DPP4 Inhibitor (Linagliptin) and Basal Insulin (Glargine) in Patients With Type 2 Diabetes in Long-term Care and Skilled Nursing Facilities: Linagliptin-LTC Trial.

Authors:  Guillermo E Umpierrez; Saumeth Cardona; David Chachkhiani; Maya Fayfman; Sahebi Saiyed; Heqiong Wang; Priyathama Vellanki; J Sonya Haw; Darin E Olson; Francisco J Pasquel; Theodore M Johnson
Journal:  J Am Med Dir Assoc       Date:  2017-12-27       Impact factor: 4.669

Review 2.  Linagliptin: an update of its use in patients with type 2 diabetes mellitus.

Authors:  Kate McKeage
Journal:  Drugs       Date:  2014-10       Impact factor: 9.546

3.  Cardiovascular and kidney outcomes of linagliptin treatment in older people with type 2 diabetes and established cardiovascular disease and/or kidney disease: A prespecified subgroup analysis of the randomized, placebo-controlled CARMELINA® trial.

Authors:  Mark E Cooper; Julio Rosenstock; Takashi Kadowaki; Yutaka Seino; Christoph Wanner; Sven Schnaidt; Douglas Clark; Odd Erik Johansen
Journal:  Diabetes Obes Metab       Date:  2020-02-27       Impact factor: 6.577

4.  Long-Term Efficacy and Safety of Linagliptin in a Japanese Population with Type 2 Diabetes Aged ≥ 60 Years Treated with Basal Insulin: A Randomised Trial.

Authors:  Eiichi Araki; Yuriko Unno; Yuko Tanaka; Wataru Sakamoto; Yuki Miyamoto
Journal:  Adv Ther       Date:  2019-09-03       Impact factor: 3.845

Review 5.  Glucose-lowering therapy in type 2 diabetes. New hope after the EMPA-REG outcome trial.

Authors:  G Schernthaner; G-H Schernthaner
Journal:  Herz       Date:  2016-05       Impact factor: 1.443

6.  Incretin-Based Therapy and Risk of Pancreatic Cancer in Patients with Type 2 Diabetes Mellitus: A Meta-analysis of Randomized Controlled Trials.

Authors:  Han Chen; Xiaoying Zhou; Tao Chen; Bingtuan Liu; Wujuan Jin; Huiyuan Gu; Tianyuan Hong; Guoxin Zhang
Journal:  Diabetes Ther       Date:  2016-09-21       Impact factor: 2.945

7.  Real-World Glycemic Lowering Effectiveness of Linagliptin Among Adults with Type 2 Diabetes by Age, Renal Function, and Race.

Authors:  Byron J Hoogwerf; Michele MacKenzie; Whitney Sealls; Jeanine Cordova; Pranav Gandhi
Journal:  Diabetes Ther       Date:  2020-05-27       Impact factor: 2.945

  7 in total

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