Literature DB >> 24672092

Effects of cimetidine, a histamine type 2 receptor antagonist, on microcirculatory disturbance of the stomach induced by full-thickness burn injuries as a model for surgical stress in rats.

Hideki Ishikawa1, Masashi Yoshida2, Go Wakabayashi2, Yoshihide Otani2, Motohide Shimazu2, Tetsuro Kubota2, Koichiro Kumai2, Naoki Aikawa1, Masaki Kitajima2.   

Abstract

BACKGROUND: We have reported the preventive effect of cimetidine, a histamine type 2 receptor antagonist, on decreased gastric mucosal blood flow induced by burn injury, a model of surgical stress.
OBJECTIVE: The present study was performed to assess the effects of cimetidine on gastric microcirculatory disturbance induced by surgical stress.
METHODS: Twelve male Wistar rats were anesthetized and a 30% full-thickness dorsal scald burn was inflicted. The total lengths of gastric erosions were measured using stereoscopic microscopy. Microvascular images in the basal region of the gastric mucosa were observed using an intravital microscope, and the diameters of venules and collecting venules were measured. Rolling leukocytes inside and along the venules, an indication of endothelial damage to the microcirculation, were observed. The rats were assigned to the cimetidine group or the control group (both, n = 6). Cimetidine 100 mg/kg was administered 30 minutes before and 2.5 hours after infliction of the burn injury. Animals in the control group were given only isotonic saline. Values are expressed as mean (SD).
RESULTS: Contraction of venules was easily observed in all rats in the control group. However, venular contraction was rarely observed in the cimetidine group. The total length of gastric erosions was significantly decreased in the cimetidine group compared with the control group (0.93 [0.58] μm vs 5.98 [5.18] μm, respectively; P < 0.05). The percentages of rolling leukocytes that passed the confluence of a prevenule and a venule were also significantly decreased in the cimetidine group compared with the control group (4.7% [7.3%] vs 22.6% [5.7%]; P < 0.01). The diameters of the venules and collecting venules were significantly larger in the cimetidine group (57.3 [6.8] μm and 75.9 [3.6] μm, respectively) than in the control group (30.9 [9.2] μm and 46.8 [8.0] μm, respectively) (both, P < 0.01).
CONCLUSIONS: The present study suggests that cimetidine may have a protective effect against gastric microcirculatory disturbances induced by burn injury, a model of surgical stress.

Entities:  

Keywords:  cimetidine; endothelial damage; gastric microcirculation; gastric mucosal lesion; histamine type 2 receptor antagonist; thermal injury

Year:  2004        PMID: 24672092      PMCID: PMC3964572          DOI: 10.1016/j.curtheres.2004.07.001

Source DB:  PubMed          Journal:  Curr Ther Res Clin Exp        ISSN: 0011-393X


  26 in total

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Authors:  M Kitajima; S Otsuka; A Shimizu; M Nakajima; T Kiuchi; Y Ikeda; A Oshima
Journal:  J Clin Gastroenterol       Date:  1988       Impact factor: 3.062

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Authors:  A Rosenberg; P H Guth
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3.  Radioautographic characterization of H1 and H2 receptor antagonists. Binding sites in rat gastric mucosal microcirculatory system.

Authors:  M Nakamura; M Oda; K Kaneko; K Honda; H Komatsu; M Tsuchiya
Journal:  Adv Exp Med Biol       Date:  1988       Impact factor: 2.622

4.  A protease inhibitor attenuates gastric erosions and microcirculatory disturbance in the early period after thermal injury in rats.

Authors:  M Yoshida; G Wakabayashi; H Ishikawa; Y Otani; M Shimazu; T Kubota; K Kumal; I Kurose; S Miura; H Ishii; M Kitajima
Journal:  J Gastroenterol Hepatol       Date:  1998-01       Impact factor: 4.029

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Journal:  Surgery       Date:  1979-10       Impact factor: 3.982

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Journal:  Gastroenterology       Date:  1982-09       Impact factor: 22.682

7.  Gastric microcirculatory disturbance and behaviour of leucocytes after thermal injury: intravital observation of arteriovenous shunting channels in the gastric submucosal layer.

Authors:  M Yoshida; D Fukumura; G Wakabayashi; Y Otani; A Oshima; M Shimazu; T Kubota; K Kumai; I Kurose; S Miura
Journal:  J Gastroenterol Hepatol       Date:  1995 Jul-Aug       Impact factor: 4.029

8.  Sialyl Lewis X analog attenuates gastric microcirculatory disturbance and gastric mucosal erosion induced by thermal injury in rats.

Authors:  Hideki Ishikawa; Masashi Yoshida; Go Wakabayashi; Masahiko Nakamura; Motohide Shimazu; Masaki Kitajima
Journal:  J Gastroenterol Hepatol       Date:  2003-01       Impact factor: 4.029

9.  Role of neutrophil-mediated inflammation in aspirin-induced gastric mucosal injury.

Authors:  N Yoshida; T Yoshikawa; Y Nakamura; M Arai; K Matsuyama; S Iinuma; N Yagi; Y Naito; M Miyasaka; M Kondo
Journal:  Dig Dis Sci       Date:  1995-11       Impact factor: 3.199

10.  H2-receptor antagonists are scavengers of oxygen radicals.

Authors:  D Lapenna; S De Gioia; A Mezzetti; L Grossi; D Festi; L Marzio; F Cuccurullo
Journal:  Eur J Clin Invest       Date:  1994-07       Impact factor: 4.686

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