Literature DB >> 24641950

Effects of protease activated receptor (PAR)2 blocking peptide on endothelin-1 levels in kidney tissues in endotoxemic rat mode.

Subrina Jesmin1, Nobutake Shimojo2, Naoto Yamaguchi3, Chishimba Nathan Mowa4, Masami Oki5, Sohel Zaedi6, Sayeeda Nusrat Sultana7, Arifur Rahman8, Majedul Islam9, Atsushi Sawamura10, Satoshi Gando11, Satoru Kawano12, Takashi Miyauchi13, Taro Mizutani14.   

Abstract

AIMS: Septic shock, the severe form of sepsis, is associated with development of progressive damage in multiple organs. Kidney can be injured and its functions altered by activation of coagulation, vasoactive-peptide and inflammatory processes in sepsis. Endothelin (ET)-1, a potent vasoconstrictor, is implicated in the pathogenesis of sepsis and its complications. Protease-activated receptors (PARs) are shown to play an important role in the interplay between inflammation and coagulation. We examined the time-dependent alterations of ET-1 and inflammatory cytokine, such as tumor necrosis factor (TNF)-α in kidney tissue in lipopolysaccharide (LPS)-induced septic rat model and the effects of PAR2 blocking peptide on the LPS-induced elevations of renal ET-1 and TNF-α levels. MAIN
METHODS: Male Wistar rats at 8 weeks of age were administered with either saline solution or LPS at different time points (1, 3, 6 and 10h). Additionally, we treated LPS-administered rats with PAR2 blocking peptide for 3h to assess whether blockade of PAR2 has a regulatory role on the ET-1 level in septic kidney. KEY
FINDINGS: An increase in ET-1 peptide level was observed in kidney tissue after LPS administration time-dependently. Levels of renal TNF-α peaked (around 12-fold) at 1h of sepsis. Interestingly, PAR2 blocking peptide normalized the LPS-induced elevations of renal ET-1 and TNF-α levels. SIGNIFICANCE: The present study reveals a distinct chronological expression of ET-1 and TNF-α in LPS-administered renal tissues and that blockade of PAR2 may play a crucial role in treating renal injury, via normalization of inflammation, coagulation and vaso-active peptide.
Copyright © 2014 Elsevier Inc. All rights reserved.

Entities:  

Keywords:  Endothelin-1; Kidney; Lipopolysaccharide; Protease activated receptor 2; Tumor necrosis factor-α

Mesh:

Substances:

Year:  2014        PMID: 24641950     DOI: 10.1016/j.lfs.2014.03.013

Source DB:  PubMed          Journal:  Life Sci        ISSN: 0024-3205            Impact factor:   5.037


  7 in total

1.  Association between Endothelin-1 Levels and Kidney Disease among Blacks.

Authors:  Casey M Rebholz; Jane L Harman; Morgan E Grams; Adolfo Correa; Daichi Shimbo; Josef Coresh; Bessie A Young
Journal:  J Am Soc Nephrol       Date:  2017-07-11       Impact factor: 10.121

Review 2.  Endothelin-1 and the kidney: new perspectives and recent findings.

Authors:  Carmen De Miguel; Joshua S Speed; Malgorzata Kasztan; Eman Y Gohar; David M Pollock
Journal:  Curr Opin Nephrol Hypertens       Date:  2016-01       Impact factor: 2.894

Review 3.  Renal microvascular endothelial cell responses in sepsis-induced acute kidney injury.

Authors:  Grietje Molema; Jan G Zijlstra; Matijs van Meurs; Jan A A M Kamps
Journal:  Nat Rev Nephrol       Date:  2021-10-19       Impact factor: 28.314

Review 4.  The Role of Endothelin and Endothelin Antagonists in Chronic Kidney Disease.

Authors:  Rupesh Raina; Abigail Chauvin; Ronith Chakraborty; Nikhil Nair; Haikoo Shah; Vinod Krishnappa; Kirsten Kusumi
Journal:  Kidney Dis (Basel)       Date:  2019-12-18

5.  Lipopolysaccharide pretreatment increases protease-activated receptor-2 expression and monocyte chemoattractant protein-1 secretion in vascular endothelial cells.

Authors:  Hung-Hsing Chao; Po-Yuan Chen; Wen-Rui Hao; Wei-Ping Chiang; Tzu-Hurng Cheng; Shih-Hurng Loh; Yuk-Man Leung; Ju-Chi Liu; Jin-Jer Chen; Li-Chin Sung
Journal:  J Biomed Sci       Date:  2017-11-15       Impact factor: 8.410

6.  Endothelin receptor-specific control of endoplasmic reticulum stress and apoptosis in the kidney.

Authors:  Carmen De Miguel; William C Hamrick; Janet L Hobbs; David M Pollock; Pamela K Carmines; Jennifer S Pollock
Journal:  Sci Rep       Date:  2017-02-23       Impact factor: 4.379

Review 7.  The role of endothelin-1 and endothelin receptor antagonists in inflammatory response and sepsis.

Authors:  Agata Kowalczyk; Paulina Kleniewska; Michal Kolodziejczyk; Beata Skibska; Anna Goraca
Journal:  Arch Immunol Ther Exp (Warsz)       Date:  2014-10-07       Impact factor: 4.291

  7 in total

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