Literature DB >> 24616015

Ruthenium-catalyzed C7 amidation of indoline C-H bonds with sulfonyl azides.

Changduo Pan1, Ablimit Abdukader, Jie Han, Yixiang Cheng, Chengjian Zhu.   

Abstract

A ruthenium-catalyzed direct C7 amidation of indoline C-H bonds with sulfonyl azides was developed. This procedure allows the synthesis of a variety of 7-amino-substituted indolines, which are useful in pharmaceutical. The good functional tolerances, as well as the mild conditions, are prominent feature of this method.
© 2014 WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim.

Entities:  

Keywords:  CH activation; amidation; indolines; ruthenium; sulfonyl azides

Mesh：

Substances：

Year:  2014        PMID： 24616015     DOI： 10.1002/chem.201304236

Source DB:  PubMed          Journal:  Chemistry        ISSN： 0947-6539            Impact factor:   5.236


  6 in total

1.  Concise Total Syntheses of (+)-Haplocidine and (+)-Haplocine via Late-Stage Oxidation of (+)-Fendleridine Derivatives.

Authors:  Kolby L White; Mohammad Movassaghi
Journal:  J Am Chem Soc       Date:  2016-08-26       Impact factor: 15.419

2.  Rhodium-Catalyzed C(sp2)-H Alkoxycarbonylation/Acylation of Indolines with Anhydrides as a Carbonyl Source.

Authors:  Hirotsugu Suzuki; Fumito Sasamori; Takanori Matsuda
Journal:  Org Lett       Date:  2022-01-31       Impact factor: 6.005

3.  Iridium-catalyzed regioselective C-H sulfonamidation of 1,2,4-thiadiazoles with sulfonyl azides in water.

Authors:  Xian-Ting Cao; Su-Ning Wei; Hao-Tian Sun; Meng Li; Zuo-Ling Zheng; Guannan Wang
Journal:  RSC Adv       Date:  2021-06-22       Impact factor: 4.036

Review 4.  Direct sulfonamidation of (hetero)aromatic C-H bonds with sulfonyl azides: a novel and efficient route to N-(hetero)aryl sulfonamides.

Authors:  Zhi Liu; Abdolghaffar Ebadi; Mohsen Toughani; Nihat Mert; Esmail Vessally
Journal:  RSC Adv       Date:  2020-10-08       Impact factor: 4.036

5.  Rh(iii)-catalyzed C-7 arylation of indolines with arylsilanes via C-H activation.

Authors:  Haiqing Luo; Qi Xie; Kai Sun; Jianbo Deng; Lin Xu; Kejun Wang; Xuzhong Luo
Journal:  RSC Adv       Date:  2019-06-10       Impact factor: 4.036

6.  Indoline-6-Sulfonamide Inhibitors of the Bacterial Enzyme DapE.

Authors:  Cory T Reidl; Tahirah K Heath; Iman Darwish; Rachel M Torrez; Maxwell Moore; Elliot Gild; Boguslaw P Nocek; Anna Starus; Richard C Holz; Daniel P Becker
Journal:  Antibiotics (Basel)       Date:  2020-09-11
  6 in total

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