Literature DB >> 24596143

Efficacy of nelfinavir as monotherapy in refractory adenoid cystic carcinoma: Results of a phase II clinical trial.

Andrew C Hoover1, Mohammed M Milhem, Carryn M Anderson, Wenqing Sun, Brian J Smith, Henry T Hoffman, John M Buatti.   

Abstract

BACKGROUND: Adenoid cystic carcinomas (ACCs) are malignant salivary gland tumors noteworthy for high rates of late failure with limited salvage therapy options. We have previously shown increased Akt signaling is common in ACC and the human immunodeficiency virus (HIV) protease inhibitor nelfinavir (NFV) inhibits in vitro tumor growth by suppressing Akt signaling. This phase II trial was conducted to determine progression-free survival in response to NFV in patients with recurrent/endstage ACC who have failed standard therapies.
METHODS: Eligible patients had recurrent or end-stage ACC and measureable disease per Response Evaluation Criteria in Solid Tumors (RECIST) criteria. NFV was provided at 1250 mg twice daily.
RESULTS: Among 15 trial participants, median progression-free survival was 5.5 months (lower 95% bound 4.4 months). No patient achieved a RECIST partial or complete response to therapy.
CONCLUSION: NFV monotherapy does not result in a meaningful improvement in clinical outcomes among patients with recurrent ACC.
© 2014 Wiley Periodicals, Inc.

Entities:  

Keywords:  Akt; adenoid cystic carcinoma; head and neck cancer; nelfinavir; salivary gland cancer

Mesh:

Substances:

Year:  2014        PMID: 24596143      PMCID: PMC4285572          DOI: 10.1002/hed.23664

Source DB:  PubMed          Journal:  Head Neck        ISSN: 1043-3074            Impact factor:   3.147


  23 in total

Review 1.  Adenoid cystic carcinoma: a retrospective clinical review.

Authors:  A J Khan; M P DiGiovanna; D A Ross; C T Sasaki; D Carter; Y H Son; B G Haffty
Journal:  Int J Cancer       Date:  2001-06-20       Impact factor: 7.396

2.  Nelfinavir induces liposarcoma apoptosis through inhibition of regulated intramembrane proteolysis of SREBP-1 and ATF6.

Authors:  Min Guan; Kristen Fousek; Chunling Jiang; Song Guo; Tim Synold; Bixin Xi; Chu-Chih Shih; Warren A Chow
Journal:  Clin Cancer Res       Date:  2011-02-25       Impact factor: 12.531

3.  PIK3CA mutations in patients with advanced cancers treated with PI3K/AKT/mTOR axis inhibitors.

Authors:  Filip Janku; Apostolia M Tsimberidou; Ignacio Garrido-Laguna; Xuemei Wang; Rajyalakshmi Luthra; David S Hong; Aung Naing; Gerald S Falchook; John W Moroney; Sarina A Piha-Paul; Jennifer J Wheler; Stacy L Moulder; Siqing Fu; Razelle Kurzrock
Journal:  Mol Cancer Ther       Date:  2011-01-07       Impact factor: 6.261

Review 4.  Targeting phosphatidylinositol 3 kinase (PI3K)-Akt beyond rapalogs.

Authors:  Shin Ogita; Patricia Lorusso
Journal:  Target Oncol       Date:  2011-05-06       Impact factor: 4.493

5.  Long-term (120-Week) antiviral efficacy and tolerability of fosamprenavir/ritonavir once daily in therapy-naive patients with HIV-1 infection: an uncontrolled, open-label, single-arm follow-on study.

Authors:  Joseph C Gathe; Robin Wood; Ian Sanne; Edwin DeJesus; Dirk Schürmann; Andrzej Gladysz; Cindy Garris; Naomi Givens; Robert Elston; Jane Yeo
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6.  Tamoxifen enhances the cytotoxic effects of nelfinavir in breast cancer cells.

Authors:  Ansgar Brüning; Klaus Friese; Alexander Burges; Ioannis Mylonas
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7.  Phase I trial of the human immunodeficiency virus protease inhibitor nelfinavir and chemoradiation for locally advanced pancreatic cancer.

Authors:  Thomas B Brunner; Matthias Geiger; Gerhard G Grabenbauer; Marga Lang-Welzenbach; Tine S Mantoni; Alexander Cavallaro; Rolf Sauer; Werner Hohenberger; W Gillies McKenna
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8.  Radiation response in two HPV-infected head-and-neck cancer cell lines in comparison to a non-HPV-infected cell line and relationship to signaling through AKT.

Authors:  Anjali K Gupta; John H Lee; Werner W Wilke; Harry Quon; Gareth Smith; Amit Maity; John M Buatti; Douglas R Spitz
Journal:  Int J Radiat Oncol Biol Phys       Date:  2009-07-01       Impact factor: 7.038

9.  The impact of nelfinavir exposure on cancer development among a large cohort of HIV-infected patients.

Authors:  Nancy F Crum-Cianflone; Katherine Huppler Hullsiek; Vincent Marconi; Amy Weintrob; Anuradha Ganesan; R Vincent Barthel; Susan Fraser; Mollie Poehlman Roediger; Brian Agan; Scott Wegner
Journal:  J Acquir Immune Defic Syndr       Date:  2009-07-01       Impact factor: 3.731

10.  Signaling pathways in adenoid cystic cancers: implications for treatment.

Authors:  Anjali K Gupta; Werner W Wilke; Erin N Taylor; Kellie L Bodeker; Henry T Hoffman; Mohammed M Milhem; John M Buatti; Robert A Robinson
Journal:  Cancer Biol Ther       Date:  2009-10-22       Impact factor: 4.742

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  8 in total

Review 1.  Systemic therapies for salivary gland adenoid cystic carcinoma.

Authors:  Sosuke Sahara; Alexandra E Herzog; Jacques E Nör
Journal:  Am J Cancer Res       Date:  2021-09-15       Impact factor: 5.942

Review 2.  Nelfinavir and other protease inhibitors in cancer: mechanisms involved in anticancer activity.

Authors:  Tomas Koltai
Journal:  F1000Res       Date:  2015-01-12

Review 3.  Redox Homeostasis and Cellular Antioxidant Systems: Crucial Players in Cancer Growth and Therapy.

Authors:  Barbara Marengo; Mariapaola Nitti; Anna Lisa Furfaro; Renata Colla; Chiara De Ciucis; Umberto Maria Marinari; Maria Adelaide Pronzato; Nicola Traverso; Cinzia Domenicotti
Journal:  Oxid Med Cell Longev       Date:  2016-06-21       Impact factor: 6.543

Review 4.  Adenoid cystic carcinoma: current therapy and potential therapeutic advances based on genomic profiling.

Authors:  Young Kwang Chae; Su Yun Chung; Andrew A Davis; Benedito A Carneiro; Sunandana Chandra; Jason Kaplan; Aparna Kalyan; Francis J Giles
Journal:  Oncotarget       Date:  2015-11-10

Review 5.  The Impact of Matrix Metalloproteinase-9 on the Sequential Steps of the Metastatic Process.

Authors:  Giovanni Barillari
Journal:  Int J Mol Sci       Date:  2020-06-25       Impact factor: 5.923

Review 6.  The Anti-Angiogenic Effects of Anti-Human Immunodeficiency Virus Drugs.

Authors:  Giovanni Barillari
Journal:  Front Oncol       Date:  2020-05-21       Impact factor: 6.244

Review 7.  Marketed nonsteroidal anti-inflammatory agents, antihypertensives, and human immunodeficiency virus protease inhibitors: as-yet-unused weapons of the oncologists' arsenal.

Authors:  Panagiota Papanagnou; Panagiotis Baltopoulos; Maria Tsironi
Journal:  Ther Clin Risk Manag       Date:  2015-05-18       Impact factor: 2.423

Review 8.  Adenoid cystic carcinoma: A review of recent advances, molecular targets, and clinical trials.

Authors:  Patrick M Dillon; Samhita Chakraborty; Christopher A Moskaluk; Prashant J Joshi; Christopher Y Thomas
Journal:  Head Neck       Date:  2015-06-16       Impact factor: 3.147

  8 in total

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