Literature DB >> 24576030

HER2/neu in Endometrial Cancer: A Promising Therapeutic Target With Diagnostic Challenges.

Natalia Buza1, Dana M Roque, Alessandro D Santin.   

Abstract

CONTEXT: In the era of targeted cancer therapy, there is growing interest in developing novel therapeutic strategies against endometrial carcinoma, especially its most biologically aggressive variant, serous adenocarcinoma. Several publications have demonstrated that a significant proportion of uterine serous carcinomas show HER2 overexpression and/or amplification, suggesting that HER2 may be a promising therapeutic target. Case reports have already shown clinical response to trastuzumab, a humanized monoclonal immunoglobulin (Ig) G1 antibody against HER2, and patients are currently being enrolled in a multi-institutional prospective randomized trial to evaluate the therapeutic efficacy of trastuzumab.
OBJECTIVE: To review current data on HER2 testing and targeted therapy against HER2/neu in endometrial carcinoma. DATA SOURCES: Review of the literature and personal experience of the authors.
CONCLUSIONS: Parallel to the clinical studies, there is a need to develop standardized criteria for HER2 testing in endometrial carcinoma that reflect the unique biological and pathogenetic features of these tumors and correlate with clinical response to therapy. This article presents a comprehensive review of the current state of HER2-based therapy and HER2 testing in endometrial carcinoma.

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Year:  2014        PMID: 24576030     DOI: 10.5858/arpa.2012-0416-RA

Source DB:  PubMed          Journal:  Arch Pathol Lab Med        ISSN: 0003-9985            Impact factor:   5.534


  39 in total

1.  Histopathological features of HER2 overexpression in uterine carcinosarcoma: proposal for requirements in HER2 testing for targeted therapy.

Authors:  Hiroshi Yoshida; Tadaaki Nishikawa; Koji Matsumoto; Masahiko Mori; Yasuyuki Hirashima; Kazuhiro Takehara; Kazuya Ariyoshi; Kosei Hasegawa; Kan Yonemori
Journal:  Virchows Arch       Date:  2021-01-09       Impact factor: 4.064

2.  Human epidermal growth factor 2 (HER2) in early stage uterine serous carcinoma: A multi-institutional cohort study.

Authors:  Britt K Erickson; Omar Najjar; Shari Damast; Adriana Blakaj; Joan Tymon-Rosario; Maryam Shahi; Alessandro Santin; Molly Klein; Michelle Dolan; Ashley Cimino-Mathews; Natalia Buza; J Stuart Ferriss; Rebecca L Stone; Mahmoud Khalifa; Amanda N Fader
Journal:  Gynecol Oncol       Date:  2020-07-21       Impact factor: 5.482

3.  Dual HER2 targeting impedes growth of HER2 gene-amplified uterine serous carcinoma xenografts.

Authors:  Jolijn W Groeneweg; Silvia F Hernandez; Virginia F Byron; Celeste M DiGloria; Hector Lopez; Vanessa Scialabba; Minji Kim; Ling Zhang; Darrell R Borger; Rosemary Tambouret; Rosemary Foster; Bo R Rueda; Whitfield B Growdon
Journal:  Clin Cancer Res       Date:  2014-10-07       Impact factor: 12.531

4.  ΔNp63α is a common inhibitory target in oncogenic PI3K/Ras/Her2-induced cell motility and tumor metastasis.

Authors:  Linshan Hu; Shan Liang; Hu Chen; Tao Lv; Junfeng Wu; Deshi Chen; Min Wu; Shengnan Sun; Haibo Zhang; Han You; Hongbin Ji; Yujun Zhang; Johann Bergholz; Zhi-Xiong Jim Xiao
Journal:  Proc Natl Acad Sci U S A       Date:  2017-05-03       Impact factor: 11.205

5.  HER2 over-expressing high grade endometrial cancer expresses high levels of p95HER2 variant.

Authors:  Whitfield B Growdon; Jolijn Groeneweg; Virginia Byron; Celeste DiGloria; Darrell R Borger; Rosemary Tambouret; Rosemary Foster; Ahmed Chenna; Jeff Sperinde; John Winslow; Bo R Rueda
Journal:  Gynecol Oncol       Date:  2015-01-17       Impact factor: 5.482

6.  Dual HER2/PIK3CA Targeting Overcomes Single-Agent Acquired Resistance in HER2-Amplified Uterine Serous Carcinoma Cell Lines In Vitro and In Vivo.

Authors:  Salvatore Lopez; Emiliano Cocco; Jonathan Black; Stefania Bellone; Elena Bonazzoli; Federica Predolini; Francesca Ferrari; Carlton L Schwab; Diana P English; Elena Ratner; Dan-Arin Silasi; Masoud Azodi; Peter E Schwartz; Corrado Terranova; Roberto Angioli; Alessandro D Santin
Journal:  Mol Cancer Ther       Date:  2015-09-02       Impact factor: 6.261

7.  Immunohistochemical characterisation of molecular subtypes in endometrial cancer.

Authors:  Sylwia M Łapińska-Szumczyk; Anna M Supernat; Hanna I Majewska; Jacek Gulczyński; Wojciech Biernat; Dariusz Wydra; Anna J Żaczek
Journal:  Int J Clin Exp Med       Date:  2015-11-15

8.  HER2-positive endometrial cancer subtype carries poor prognosis.

Authors:  Sylwia Lapińska-Szumczyk; Anna Supernat; Hanna Majewska; Jacek Gulczyński; Agata Luczak; Wojciech Biernat; Dariusz Wydra; Anna J Zaczek
Journal:  Clin Transl Sci       Date:  2014-09-09       Impact factor: 4.689

9.  Detection of ERBB2 amplification in uterine serous carcinoma by next-generation sequencing: an approach highly concordant with standard assays.

Authors:  Carrie L Robinson; Beth T Harrison; Azra H Ligon; Fei Dong; Valeria Maffeis; Ursula Matulonis; Marisa R Nucci; David L Kolin
Journal:  Mod Pathol       Date:  2020-10-19       Impact factor: 7.842

10.  Randomized Phase II Trial of Carboplatin-Paclitaxel Compared with Carboplatin-Paclitaxel-Trastuzumab in Advanced (Stage III-IV) or Recurrent Uterine Serous Carcinomas that Overexpress Her2/Neu (NCT01367002): Updated Overall Survival Analysis.

Authors:  Amanda N Fader; Dana M Roque; Eric Siegel; Natalia Buza; Pei Hui; Osama Abdelghany; Setsuko Chambers; Angeles Alvarez Secord; Laura Havrilesky; David M O'Malley; Floor J Backes; Nicole Nevadunsky; Babak Edraki; Dirk Pikaart; William Lowery; Karim ElSahwi; Paul Celano; Stefania Bellone; Masoud Azodi; Babak Litkouhi; Elena Ratner; Dan-Arin Silasi; Peter E Schwartz; Alessandro D Santin
Journal:  Clin Cancer Res       Date:  2020-06-29       Impact factor: 12.531

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