Literature DB >> 24549816

In vitro cell integrated impactor deposition methodology for the study of aerodynamically relevant size fractions from commercial pressurised metered dose inhalers.

Mehra Haghi1, Daniela Traini, Paul Young.   

Abstract

PURPOSE: The purpose of this study was to present a modified Andersen cascade impactor (ACI) as a platform to evaluate the deposition and subsequent transport of aerosol micropaticles across airway epithelial cells.
METHODS: The impaction plate of an ACI was modified to accommodate up to eight Snapwells. Aerodynamic particle size distribution of the modified ACI was investigated with two commercially available formulations of Ventolin® (salbutamol sulphate) and QVAR® (beclomethasone dipropionate). Deposition and transport of these drug microparticles across sub-bronchial epithelial Calu-3 cells were also studied.
RESULTS: The modified ACI demonstrated reproducible deposition patterns of the commercially available pressurised metered dose inhalers compared to the standard ACI. Furthermore, the Calu-3 cells could be placed in different stages of the modified ACI. No significant effect was observed among the transport rate of different particle sizes deposited on Calu-3 cells within the range of 3.3 to 0.4 μm.
CONCLUSIONS: The use of the cell compatible ACI to assess the fate of microparticles after deposition on the respiratory epithelia may allow for better understanding of deposited microparticles in vivo.

Entities:  

Mesh:

Substances:

Year:  2014        PMID: 24549816     DOI: 10.1007/s11095-013-1282-2

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  27 in total

1.  Large porous particle impingement on lung epithelial cell monolayers--toward improved particle characterization in the lung.

Authors:  Jennifer Fiegel; Carsten Ehrhardt; Ulrich Friedrich Schaefer; Claus-Michael Lehr; Justin Hanes
Journal:  Pharm Res       Date:  2003-05       Impact factor: 4.200

Review 2.  Analysis of cascade impactor mass distributions.

Authors:  Craig Dunbar; Jolyon Mitchell
Journal:  J Aerosol Med       Date:  2005

Review 3.  Pulmonary cell culture models to study the safety and efficacy of innovative aerosol medicines.

Authors:  Michael Bur; Claus-Michael Lehr
Journal:  Expert Opin Drug Deliv       Date:  2008-06       Impact factor: 6.648

4.  Drug transport across pulmonary epithelial cell monolayers: effects of particle size, apical liquid volume, and deposition technique.

Authors:  Michael Bur; Hanno Huwer; Leon Muys; Claus-Michael Lehr
Journal:  J Aerosol Med Pulm Drug Deliv       Date:  2010-06       Impact factor: 2.849

5.  A novel cell compatible impingement system to study in vitro drug absorption from dry powder aerosol formulations.

Authors:  Michael Bur; Barbara Rothen-Rutishauser; Hanno Huwer; Claus-Michael Lehr
Journal:  Eur J Pharm Biopharm       Date:  2008-08-17       Impact factor: 5.571

6.  A novel method for assessing dissolution of aerosol inhaler products.

Authors:  Neal M Davies; Majid R Feddah
Journal:  Int J Pharm       Date:  2003-04-14       Impact factor: 5.875

7.  Size analysis of a pressurized metered dose inhaler-delivered solution formulation by an Aerosizer-LD time-of-flight aerosol particle size spectrometer.

Authors:  Mark W Nagel; Kimberly J Wiersema; Sara Lou Bates; Jolyon P Mitchell
Journal:  J Aerosol Med       Date:  2002

8.  Fluticasone uptake across Calu-3 cells is mediated by salmeterol when deposited as a combination powder inhaler.

Authors:  Mehra Haghi; Daniela Traini; Dirkje S Postma; Mary Bebawy; Paul M Young
Journal:  Respirology       Date:  2013-11       Impact factor: 6.424

9.  Critical characteristics for corticosteroid solution metered dose inhaler bioequivalence.

Authors:  C I Grainger; M Saunders; F Buttini; R Telford; L L Merolla; G P Martin; S A Jones; B Forbes
Journal:  Mol Pharm       Date:  2012-02-10       Impact factor: 4.939

10.  The permeability of large molecular weight solutes following particle delivery to air-interfaced cells that model the respiratory mucosa.

Authors:  C I Grainger; L L Greenwell; G P Martin; B Forbes
Journal:  Eur J Pharm Biopharm       Date:  2008-09-25       Impact factor: 5.571

View more
  8 in total

1.  Absorption and Clearance of Pharmaceutical Aerosols in the Human Nose: Effects of Nasal Spray Suspension Particle Size and Properties.

Authors:  Alex Rygg; Michael Hindle; P Worth Longest
Journal:  Pharm Res       Date:  2015-12-21       Impact factor: 4.200

2.  Delivery of pDNA Polyplexes to Bronchial and Alveolar Epithelial Cells Using a Mesh Nebulizer.

Authors:  Larissa Gomes Dos Reis; Maree Svolos; Lyn M Moir; Rima Jaber; Norbert Windhab; Paul M Young; Daniela Traini
Journal:  Pharm Res       Date:  2018-11-15       Impact factor: 4.200

3.  Sweetening Inhaled Antibiotic Treatment for Eradication of Chronic Respiratory Biofilm Infection.

Authors:  Ching-Yee Loo; Wing-Hin Lee; Gianluca Lauretani; Santo Scalia; David Cipolla; Daniela Traini; Paul Young; Hui Xin Ong
Journal:  Pharm Res       Date:  2018-02-07       Impact factor: 4.200

4.  Immunomodulatory effects of a low-dose clarithromycin-based macrolide solution pressurised metered dose inhaler.

Authors:  Mehra Haghi; Alessandro Saadat; Bing Zhu; Gaia Colombo; Gregory King; Paul M Young; Daniela Traini
Journal:  Pharm Res       Date:  2014-12-24       Impact factor: 4.200

5.  Inhalable Clarithromycin Microparticles for Treatment of Respiratory Infections.

Authors:  Frantiescoli Dimer; Cristiane de Souza Carvalho-Wodarz; Jörg Haupenthal; Rolf Hartmann; Claus-Michael Lehr
Journal:  Pharm Res       Date:  2015-06-26       Impact factor: 4.200

Review 6.  Nanoparticle Delivery Platforms for RNAi Therapeutics Targeting COVID-19 Disease in the Respiratory Tract.

Authors:  Yuan Zhang; Juhura G Almazi; Hui Xin Ong; Matt D Johansen; Scott Ledger; Daniela Traini; Philip M Hansbro; Anthony D Kelleher; Chantelle L Ahlenstiel
Journal:  Int J Mol Sci       Date:  2022-02-22       Impact factor: 5.923

7.  Deposition and transport of linezolid mediated by a synthetic surfactant Synsurf® within a pressurized metered dose inhaler: a Calu-3 model.

Authors:  Lyné van Rensburg; Johann M van Zyl; Johan Smith
Journal:  Drug Des Devel Ther       Date:  2018-05-04       Impact factor: 4.162

Review 8.  Modifying and Integrating in vitro and ex vivo Respiratory Models for Inhalation Drug Screening.

Authors:  Aylin Cidem; Peta Bradbury; Daniela Traini; Hui Xin Ong
Journal:  Front Bioeng Biotechnol       Date:  2020-10-23
  8 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.