Literature DB >> 24505552

A Divalent Protecting Group for Benzoxaboroles.

Brett Vanveller1, Matthew R Aronoff2, Ronald T Raines3.   

Abstract

1-Dimethylamino-8-methylaminonaphthalene is put forth as a protecting group for benzoxaboroles. The ensuing complex is fluorescent, charge-neutral, highly stable under basic conditions, stable to anhydrous acid, and readily cleavable in aqueous acid to return the free benzoxaborole.

Entities:  

Year:  2013        PMID： 24505552      PMCID： PMC3910298          DOI： 10.1039/C3RA44385J

Source DB:  PubMed          Journal:  RSC Adv        ISSN： 2046-2069            Impact factor:   3.361


  34 in total

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Authors:  Xianfeng Li; Yong-Kang Zhang; Yang Liu; Charles Z Ding; Qun Li; Yasheen Zhou; Jacob J Plattner; Stephen J Baker; Xuelei Qian; Dazhong Fan; Liang Liao; Zhi-Jie Ni; Gemma V White; Jackie E Mordaunt; Linos X Lazarides; Martin J Slater; Richard L Jarvest; Pia Thommes; Malcolm Ellis; Colin M Edge; Julia A Hubbard; Don Somers; Paul Rowland; Pamela Nassau; Bill McDowell; Tadeusz J Skarzynski; Wieslaw M Kazmierski; Richard M Grimes; Lois L Wright; Gary K Smith; Wuxin Zou; Jon Wright; Lewis E Pennicott
Journal:  Bioorg Med Chem Lett       Date:  2010-05-20       Impact factor: 2.823

2.  Chalcone-benzoxaborole hybrid molecules as potent antitrypanosomal agents.

Authors:  Zhitao Qiao; Qi Wang; Fenglong Zhang; Zhongli Wang; Tana Bowling; Bakela Nare; Robert T Jacobs; Jiong Zhang; Dazhong Ding; Yangang Liu; Huchen Zhou
Journal:  J Med Chem       Date:  2012-03-14       Impact factor: 7.446

3.  A benzoboroxole-functionalized monolithic column for the selective enrichment and separation of cis-diol containing biomolecules.

Authors:  Hengye Li; Heye Wang; Yunchun Liu; Zhen Liu
Journal:  Chem Commun (Camb)       Date:  2012-03-20       Impact factor: 6.222

4.  Label-free detection of enhanced saccharide binding at pH 7.4 to nanoparticulate benzoboroxole based receptor units.

Authors:  Soeren Schumacher; Martin Katterle; Cornelia Hettrich; Bernd-Reiner Paulke; Dennis G Hall; Frieder W Scheller; Nenad Gajovic-Eichelmann
Journal:  J Mol Recognit       Date:  2011 Nov-Dec       Impact factor: 2.137

5.  A new palladium precatalyst allows for the fast Suzuki-Miyaura coupling reactions of unstable polyfluorophenyl and 2-heteroaryl boronic acids.

Authors:  Tom Kinzel; Yong Zhang; Stephen L Buchwald
Journal:  J Am Chem Soc       Date:  2010-10-13       Impact factor: 15.419

6.  Synthesis and SAR of novel benzoxaboroles as a new class of β-lactamase inhibitors.

Authors:  Yi Xia; Kathy Cao; Yasheen Zhou; M R K Alley; Fernando Rock; Manisha Mohan; Maliwan Meewan; Stephen J Baker; Sarah Lux; Charles Z Ding; Guofeng Jia; Maureen Kully; Jacob J Plattner
Journal:  Bioorg Med Chem Lett       Date:  2011-02-12       Impact factor: 2.823

7.  Benzoboroxoles as efficient glycopyranoside-binding agents in physiological conditions: structure and selectivity of complex formation.

Authors:  Marie Bérubé; Meenakshi Dowlut; Dennis G Hall
Journal:  J Org Chem       Date:  2008-06-13       Impact factor: 4.354

8.  An antifungal agent inhibits an aminoacyl-tRNA synthetase by trapping tRNA in the editing site.

Authors:  Fernando L Rock; Weimin Mao; Anya Yaremchuk; Mikhail Tukalo; Thibaut Crépin; Huchen Zhou; Yong-Kang Zhang; Vincent Hernandez; Tsutomu Akama; Stephen J Baker; Jacob J Plattner; Lucy Shapiro; Susan A Martinis; Stephen J Benkovic; Stephen Cusack; M R K Alley
Journal:  Science       Date:  2007-06-22       Impact factor: 47.728

9.  Differentially protected benzenediboronic acids: divalent cross-coupling modules for the efficient synthesis of boron-substituted oligoarenes.

Authors:  Hiroyoshi Noguchi; Takayuki Shioda; Chih-Ming Chou; Michinori Suginome
Journal:  Org Lett       Date:  2008-01-10       Impact factor: 6.005

10.  Discovery and structure-activity study of a novel benzoxaborole anti-inflammatory agent (AN2728) for the potential topical treatment of psoriasis and atopic dermatitis.

Authors:  Tsutomu Akama; Stephen J Baker; Yong-Kang Zhang; Vincent Hernandez; Huchen Zhou; Virginia Sanders; Yvonne Freund; Richard Kimura; Kirk R Maples; Jacob J Plattner
Journal:  Bioorg Med Chem Lett       Date:  2009-03-09       Impact factor: 2.823
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  1 in total

1.  Temporal and Wash-Out Studies Identify Medicines for Malaria Venture Pathogen Box Compounds with Fast-Acting Activity against Both Trypanosoma cruzi and Trypanosoma brucei.

Authors:  Melissa L Sykes; Emily K Kennedy; Kevin D Read; Marcel Kaiser; Vicky M Avery
Journal:  Microorganisms       Date:  2022-06-25
  1 in total

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