Literature DB >> 24499847

Safety, efficacy and population pharmacokinetics of fixed-dose combination of artesunate-mefloquine in the treatment of acute uncomplicated Plasmodium falciparum malaria in India.

Neena Valecha, Bina Srivastava, N G Dubhashi, B H Krishnamoorthy Rao, Ashwani Kumar, S K Ghosh, Jai Prakash Narayan Singh, J R Kiechel, Bhawna Sharma, V Jullien, A P Dash, W R J Taylor, Anupkumar R Anvikar1.   

Abstract

BACKGROUND &
OBJECTIVES: India has switched over to artemisinin-based combination therapy (ACT) for the treatment of acute uncomplicated Plasmodium falciparum malaria and the ACT used in the national programme is artesunate + sulphadoxine-pyrimethamine. Since the efficacy of ACT is dependent also on the partner drug, there is a need to evaluate and deploy multiple ACTs.
METHODS: This multicentre, single-arm, open-label clinical trial was carried out to assess the efficacy, safety and population pharmacokinetics of a fixed dose combination (FDC) artesunate mefloquine (ASMQ) in P. falciparum infected, Indian adults at Panjim, Goa, and Mangalore, Karnataka between December 2007 and November 2008.
RESULTS: A total of 77 patients (males 74) were screened and enrolled: 42 at Goa and 35 at Mangalore with a median age of 25 yr (range 18-55 yr). One patient failed in treatment on D53, a PCR proven new infection, seven developed recurrent vivax parasitaemia and 11 did not have a parasitological endpoint. By per protocol analysis, the D63 cure rate was 58/59 (98.3; 95% C.I. 90.9-99.9%), and 58/58, with PCR correction. ASMQ was well-tolerated and no serious adverse events were reported. INTERPRETATION &
CONCLUSION: The study showed that the ASMQ FDC was efficacious and well-tolerated for the treatment of acute, uncomplicated P. falciparum malaria in highly endemic, chloroquine resistant areas of Goa and Mangalore. It is a viable option for India.

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Year:  2013        PMID: 24499847

Source DB:  PubMed          Journal:  J Vector Borne Dis        ISSN: 0972-9062            Impact factor:   1.688


  5 in total

Review 1.  Antimalarial drug policy in India: past, present & future.

Authors:  Anupkumar R Anvikar; Usha Arora; G S Sonal; Neelima Mishra; Bharatendu Shahi; Deepali Savargaonkar; Navin Kumar; Naman K Shah; Neena Valecha
Journal:  Indian J Med Res       Date:  2014-02       Impact factor: 2.375

2.  Comparison of artesunate-mefloquine and artemether-lumefantrine fixed-dose combinations for treatment of uncomplicated Plasmodium falciparum malaria in children younger than 5 years in sub-Saharan Africa: a randomised, multicentre, phase 4 trial.

Authors:  Sodiomon B Sirima; Bernhards Ogutu; John P A Lusingu; Ali Mtoro; Zakayo Mrango; Alphonse Ouedraogo; Jean Baptiste Yaro; Kevin Omondi Onyango; Samwel Gesase; Ernest Mnkande; James Samwel Ngocho; Isabelle Ackermann; François Aubin; Joelle Vanraes; Nathalie Strub; Gwenaelle Carn
Journal:  Lancet Infect Dis       Date:  2016-07-16       Impact factor: 25.071

3.  Efficacy of two artemisinin-based combinations for the treatment of malaria in pregnancy in India: a randomized controlled trial.

Authors:  Anupkumar R Anvikar; Irene Kuepfer; Vinitkumar Mishra; Jane Bruce; Tushar Arya; Deb Ranjan Mishra; Sanjib Mohanty; Rajesh Mohanty; Bina Srivastava; Suryakant Sharma; Neelima Mishra; Brian Greenwood; Daniel Chandramohan; Neena Valecha
Journal:  Malar J       Date:  2018-07-04       Impact factor: 2.979

4.  Population pharmacokinetics of mefloquine, administered as a fixed-dose combination of artesunate-mefloquine in Indian patients for the treatment of acute uncomplicated Plasmodium falciparum malaria.

Authors:  Vincent Jullien; Neena Valecha; Bina Srivastava; Bhawna Sharma; Jean-René Kiechel
Journal:  Malar J       Date:  2014-05-23       Impact factor: 2.979

5.  Pharmacokinetics of mefloquine administered with artesunate in patients with uncomplicated falciparum malaria from the Brazilian Amazon basin.

Authors:  Michelle V D Ferreira; José L F Vieira; Eduardo D Almeida; Juan G B Rivera; Margarete S M Gomes; André M de Siqueira
Journal:  Malar J       Date:  2018-07-16       Impact factor: 2.979

  5 in total

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