Literature DB >> 24256886

Mechanosynthesis of pharmaceutically relevant sulfonyl-(thio)ureas.

Davin Tan1, Vjekoslav Štrukil, Cristina Mottillo, Tomislav Friščić.   

Abstract

We demonstrate the first application of mechanochemistry to conduct the synthesis of sulfonyl-(thio)ureas, including known anti-diabetic drugs tolbutamide, chlorpropamide and glibenclamide, in good to excellent isolated yields by either stoichiometric base-assisted or copper-catalysed coupling of sulfonamides and iso(thio)cyanates.

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Year:  2013        PMID： 24256886     DOI： 10.1039/c3cc47905f

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  12 in total

Review 1.  Mechanochemistry: New Tools to Navigate the Uncharted Territory of "Impossible" Reactions.

Authors:  Federico Cuccu; Lidia De Luca; Francesco Delogu; Evelina Colacino; Niclas Solin; Rita Mocci; Andrea Porcheddu
Journal:  ChemSusChem       Date:  2022-07-21       Impact factor: 9.140

2.  Redox-promoted associative assembly of metal-organic materials.

Authors:  Martin Glavinović; Feng Qi; Athanassios D Katsenis; Tomislav Friščić; Jean-Philip Lumb
Journal:  Chem Sci       Date:  2015-10-09       Impact factor: 9.825

Review 3.  Mechanochemistry: A Force of Synthesis.

Authors:  Jean-Louis Do; Tomislav Friščić
Journal:  ACS Cent Sci       Date:  2016-12-29       Impact factor: 14.553

Review 4.  Mechanochemistry as an emerging tool for molecular synthesis: what can it offer?

Authors:  Joseph L Howard; Qun Cao; Duncan L Browne
Journal:  Chem Sci       Date:  2018-03-07       Impact factor: 9.825

Review 5.  Advances in Solid-State Transformations of Coordination Bonds: From the Ball Mill to the Aging Chamber.

Authors:  Cristina Mottillo; Tomislav Friščić
Journal:  Molecules       Date:  2017-01-17       Impact factor: 4.411

6.  Mechanochemical Catalytic Transfer Hydrogenation of Aromatic Nitro Derivatives.

Authors:  Tomislav Portada; Davor Margetić; Vjekoslav Štrukil
Journal:  Molecules       Date:  2018-11-30       Impact factor: 4.411

Review 7.  Main group mechanochemistry.

Authors:  Agota A Gečiauskaitė; Felipe García
Journal:  Beilstein J Org Chem       Date:  2017-10-05       Impact factor: 2.883

8.  Mechanochemical N-alkylation of imides.

Authors:  Anamarija Briš; Mateja Đud; Davor Margetić
Journal:  Beilstein J Org Chem       Date:  2017-08-22       Impact factor: 2.883

Review 9.  Mechanochemical synthesis of thioureas, ureas and guanidines.

Authors:  Vjekoslav Štrukil
Journal:  Beilstein J Org Chem       Date:  2017-09-01       Impact factor: 2.883

10.  Mechanochemical Preparation of Active Pharmaceutical Ingredients Monitored by In Situ Raman Spectroscopy.

Authors:  Irena Sović; Stipe Lukin; Ernest Meštrović; Ivan Halasz; Andrea Porcheddu; Francesco Delogu; Pier Carlo Ricci; Fabien Caron; Thomas Perilli; Anita Dogan; Evelina Colacino
Journal:  ACS Omega       Date:  2020-10-30
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