Literature DB >> 24103533

Role of the aromatase inhibitor letrozole in the management of uterine leiomyomas in premenopausal women.

Nirmala Duhan1, Shikha Madaan, Jyotsna Sen.   

Abstract

BACKGROUND: Uterine myomas are benign tumours affecting 20-40% women. Various medical and surgical therapeutic options are available but the search for an ideal medical option continues. Aromatase inhibitors have recently been reported to have a potential role in the management of oestrogen-dependent conditions like endometriosis and leiomyoma.
OBJECTIVE: To evaluate the effect of letrozole on uterine myoma size and symptomatology in perimenopausal women. STUDY
DESIGN: Prospective interventional study conducted on 30 premenopausal women aged between 30 and 55 years with menstrual or pressure symptoms and having a single intrauterine myoma of size 4 cm or more with or without one or more additional myomata each of size 2 cm or less. They received tablet letrozole 2.5 mg a day for 12 weeks, and the effect of the drug on myoma size and volume and symptomatology was studied along with the adverse effect profile and patient satisfaction.
RESULTS: The mean myoma size reduced from 5.4±1.3 cm to 4.3±0.9 cm (p<0.05) and the myoma volume exhibited a reduction of 52.45% (p=0.00) at the end of 3 months. The symptomatology score showed a significant improvement that persisted up to 3 months after cessation of therapy. No significant effect was observed on lipid profile, serum estradiol, progesterone, testosterone and FSH and LH levels during the therapy. Nausea and hot flushes were the main adverse effects observed and were self-limiting.
CONCLUSION: Letrozole significantly reduces myoma size and volume and also improves the associated symptoms. It has a good adverse effect profile and appears to be a promising medical option for management of uterine myomas.
Copyright © 2013 Elsevier Ireland Ltd. All rights reserved.

Entities:  

Keywords:  Letrozole; Medical therapy; Uterine myoma

Mesh:

Substances:

Year:  2013        PMID: 24103533     DOI: 10.1016/j.ejogrb.2013.09.010

Source DB:  PubMed          Journal:  Eur J Obstet Gynecol Reprod Biol        ISSN: 0301-2115            Impact factor:   2.435


  10 in total

Review 1.  Endocrinology of uterine fibroids: steroid hormones, stem cells, and genetic contribution.

Authors:  Molly B Moravek; Serdar E Bulun
Journal:  Curr Opin Obstet Gynecol       Date:  2015-08       Impact factor: 1.927

2.  Obligatory role of hypothalamic neuroestradiol during the estrogen-induced LH surge in female ovariectomized rhesus monkeys.

Authors:  Brian P Kenealy; Kim L Keen; James P Garcia; Lucille K Kohlenberg; Ei Terasawa
Journal:  Proc Natl Acad Sci U S A       Date:  2017-12-11       Impact factor: 11.205

Review 3.  The conservative and interventional treatment of fibroids.

Authors:  Alexander Stephan Boosz; Peter Reimer; Matthias Matzko; Thomas Römer; Andreas Müller
Journal:  Dtsch Arztebl Int       Date:  2014-12-22       Impact factor: 5.594

Review 4.  Current approaches to overcome the side effects of GnRH analogs in the treatment of patients with uterine fibroids.

Authors:  Mohamed Ali; Mohamed Raslan; Michał Ciebiera; Kornelia Zaręba; Ayman Al-Hendy
Journal:  Expert Opin Drug Saf       Date:  2021-10-20       Impact factor: 4.250

Review 5.  Ovarian steroids, stem cells and uterine leiomyoma: therapeutic implications.

Authors:  Molly B Moravek; Ping Yin; Masanori Ono; John S Coon; Matthew T Dyson; Antonia Navarro; Erica E Marsh; Debabrata Chakravarti; J Julie Kim; Jian-Jun Wei; Serdar E Bulun
Journal:  Hum Reprod Update       Date:  2014-09-08       Impact factor: 15.610

Review 6.  Role of Transforming Growth Factor β in Uterine Fibroid Biology.

Authors:  Michał Ciebiera; Marta Włodarczyk; Małgorzata Wrzosek; Błażej Męczekalski; Grażyna Nowicka; Krzysztof Łukaszuk; Magdalena Ciebiera; Aneta Słabuszewska-Jóźwiak; Grzegorz Jakiel
Journal:  Int J Mol Sci       Date:  2017-11-17       Impact factor: 5.923

Review 7.  Current medical treatment of uterine fibroids.

Authors:  Geum Seon Sohn; SiHyun Cho; Yong Man Kim; Chi-Heum Cho; Mee-Ran Kim; Sa Ra Lee
Journal:  Obstet Gynecol Sci       Date:  2018-02-13

Review 8.  Clinical Utility Of Elagolix As An Oral Treatment For Women With Uterine Fibroids: A Short Report On The Emerging Efficacy Data.

Authors:  Manuela Neri; Gian Benedetto Melis; Elena Giancane; Valerio Vallerino; Monica Pilloni; Bruno Piras; Alessandro Loddo; Anna Maria Paoletti; Valerio Mais
Journal:  Int J Womens Health       Date:  2019-10-22

Review 9.  Alternative Oral Agents in Prophylaxis and Therapy of Uterine Fibroids-An Up-to-Date Review.

Authors:  Michał Ciebiera; Krzysztof Łukaszuk; Błażej Męczekalski; Magdalena Ciebiera; Cezary Wojtyła; Aneta Słabuszewska-Jóźwiak; Grzegorz Jakiel
Journal:  Int J Mol Sci       Date:  2017-12-01       Impact factor: 5.923

10.  Gonadotropin-releasing Hormone Agonist Plus Aromatase Inhibitor in the Treatment of Uterine Leiomyoma in Near Menopause Patient: A Case Series Study.

Authors:  Sanam Moradan
Journal:  J Menopausal Med       Date:  2018-04-30
  10 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.